Publications by authors named "Celine M'Kadmi"

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Design and characterization of a triazole-based growth hormone secretagogue receptor modulator inhibiting the glucoregulatory and feeding actions of ghrelin.
Sylvie Péraldi-Roux, Morgane Bayle, Céline M'Kadmi, Marjorie Damian, Justine Vaillé

Biochem Pharmacol· August 2022

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Concerted conformational dynamics and water movements in the ghrelin G protein-coupled receptor.
Maxime Louet, Marina Casiraghi, Marjorie Damian, Mauricio Gs Costa, Pedro Renault, Céline M'Kadmi

Elife· September 2021

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Allosteric modulation of ghrelin receptor signaling by lipids.
Marjorie Damian, Maxime Louet, Antoniel Augusto Severo Gomes, Céline M'Kadmi, Séverine Denoyelle

Nat Commun· June 2021

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Development of Nonpeptidic Inverse Agonists of the Ghrelin Receptor (GHSR) Based on the 1,2,4-Triazole Scaffold.
Khoubaib Ben Haj Salah, Mathieu Maingot, Anne-Laure Blayo, Céline M'Kadmi, Marjorie Damian

J Med Chem· October 2020

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Development of a novel fluorescent ligand of growth hormone secretagogue receptor based on the N-Terminal Leap2 region.
Franco Barrile, Céline M'Kadmi, Pablo N De Francesco, Agustina Cabral, Guadalupe García Romero

Mol Cell Endocrinol· December 2019

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Structure and dynamics of G protein-coupled receptor-bound ghrelin reveal the critical role of the octanoyl chain.
Guillaume Ferré, Maxime Louet, Oliver Saurel, Bartholomé Delort, Georges Czaplicki, Céline M'Kadmi

Proc Natl Acad Sci U S A· August 2019

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N-Terminal Liver-Expressed Antimicrobial Peptide 2 (LEAP2) Region Exhibits Inverse Agonist Activity toward the Ghrelin Receptor.
Céline M'Kadmi, Agustina Cabral, Franco Barrile, Julien Giribaldi, Sonia Cantel

J Med Chem· January 2019

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GHSR-D2R heteromerization modulates dopamine signaling through an effect on G protein conformation.
Marjorie Damian, Véronique Pons, Pedro Renault, Céline M'Kadmi, Bartholomé Delort

Proc Natl Acad Sci U S A· April 2018

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Evidence Supporting a Role for Constitutive Ghrelin Receptor Signaling in Fasting-Induced Hyperphagia in Male Mice.
Gimena Fernandez, Agustina Cabral, María F Andreoli, Alexandra Labarthe, Céline M'Kadmi

Endocrinology· February 2018

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Conditional and Reversible Activation of Class A and B G Protein-Coupled Receptors Using Tethered Pharmacology.
Tom Podewin, Julia Ast, Johannes Broichhagen, Nicholas H F Fine, Daniela Nasteska, Celine M'Kadmi

ACS Cent Sci· February 2018

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Cardioprotective Angiotensin-(1-7) Peptide Acts as a Natural-Biased Ligand at the Angiotensin II Type 1 Receptor.
Ségolène Galandrin, Colette Denis, Cédric Boularan, Jacky Marie, Céline M'Kadmi

Hypertension· December 2016

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Quantitative MALDI-MS Binding Assays: An Alternative to Radiolabeling.
Maxime Rossato, Guillaume Miralles, Céline M'Kadmi, Mathieu Maingot, Muriel Amblard

ChemMedChem· December 2016

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New ligands of the ghrelin receptor based on the 1,2,4-triazole scaffold by introduction of a second chiral center.
Mathieu Maingot, Anne-Laure Blayo, Séverine Denoyelle, Céline M'Kadmi, Marjorie Damian

Bioorg Med Chem Lett· May 2016

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The novel nonapeptide acein targets angiotensin converting enzyme in the brain and induces dopamine release.
Jérémie Neasta, Charlène Valmalle, Anne-Claire Coyne, Eric Carnazzi, Gilles Subra, Céline M'Kadmi

Br J Pharmacol· April 2016

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Detergent-free Isolation of Functional G Protein-Coupled Receptors into Nanometric Lipid Particles.
Christel Logez, Marjorie Damian, Céline Legros, Clémence Dupré, Mélody Guéry, Céline M'Kadmi

Biochemistry· January 2016

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Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling.
Céline M'Kadmi, Jean-Philippe Leyris, Lauriane Onfroy, Céline Galés, Aude Saulière

J Biol Chem· November 2015

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A new way to silicone-based peptide polymers.
Said Jebors, Jeremie Ciccione, Soultan Al-Halifa, Benjamin Nottelet, Christine Enjalbal, Céline M'Kadmi

Angew Chem Int Ed Engl· March 2015

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Ghrelin receptor conformational dynamics regulate the transition from a preassembled to an active receptor:Gq complex.
Marjorie Damian, Sophie Mary, Mathieu Maingot, Céline M'Kadmi, Didier Gagne

Proc Natl Acad Sci U S A· February 2015

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New trisubstituted 1,2,4-triazoles as ghrelin receptor antagonists.
Anne-Laure Blayo, Mathieu Maingot, Babette Aicher, Céline M'Kadmi, Peter Schmidt

Bioorg Med Chem Lett· January 2015

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Gastrin releasing peptide receptor-directed radioligands based on a bombesin antagonist: synthesis, (111)in-labeling, and preclinical profile.
Panteleimon J Marsouvanidis, Berthold A Nock, Bouchra Hajjaj, Jean-Alain Fehrentz, Luc Brunel, Céline M'Kadmi

J Med Chem· March 2013

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The 1,2,4-triazole as a scaffold for the design of ghrelin receptor ligands: development of JMV 2959, a potent antagonist.
Aline Moulin, Luc Brunel, Damien Boeglin, Luc Demange, Johanne Ryan, Céline M'Kadmi

Amino Acids· February 2013

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α-tocopherol and α-tocopheryl phosphate interact with the cannabinoid system in the rodent hippocampus.
Nadine Crouzin, Marie-Céleste de Jesus Ferreira, Catherine Cohen-Solal, Céline M'Kadmi, Nicole Bernad

Free Radic Biol Med· November 2011

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Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a.
Jean-Philippe Leyris, Thomas Roux, Eric Trinquet, Pascal Verdié, Jean-Alain Fehrentz, Céline M'kadmi

Anal Biochem· January 2011

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Involvement of tryptophan W276 and of two surrounding amino acid residues in the high constitutive activity of the ghrelin receptor GHS-R1a.
Catherine Gozé, Gilbert Bergé, Céline M'Kadmi, Nicolas Floquet, Didier Gagne

Eur J Pharmacol· September 2010

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Activation of the ghrelin receptor is described by a privileged collective motion: a model for constitutive and agonist-induced activation of a sub-class A G-protein coupled receptor (GPCR).
Nicolas Floquet, Céline M'Kadmi, David Perahia, Didier Gagne, Gilbert Bergé

J Mol Biol· January 2010

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