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Publications by authors named "Chuck Locuson"

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Volumetric absorptive microsampling as an effective microsampling technique for LC-MS/MS bioanalysis of biomarkers in drug discovery.
Unnati Kapadnis, Chuck Locuson, Heidi Okamura, Gianluca De Rienzo, Cece Cotter

Bioanalysis· July 2023


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Discovery of (S)-2-cyclopentyl-N-((1-isopropylpyrrolidin2-yl)-9-methyl-1-oxo-2,9-dihydro-1H-pyrrido[3,4-b]indole-4-carboxamide (VU0453379): a novel, CNS penetrant glucagon-like peptide 1 receptor (GLP-1R) positive allosteric modulator (PAM).
Lindsey C Morris, Kellie D Nance, Patrick R Gentry, Emily L Days, C David Weaver, Chuck W Locuson

J Med Chem· December 2014


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Challenges in exploring the cytochrome P450 system as a source of variation in canine drug pharmacokinetics.
Marilyn N Martinez, Leposava Antonovic, Michael Court, Mauro Dacasto, Johanna Fink-Gremmels, Chuck Locuson

Drug Metab Rev· May 2013


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Amiodarone analog-dependent effects on CYP2C9-mediated metabolism and kinetic profiles.
Vikas Kumar, Chuck W Locuson, Yuk Y Sham, Timothy S Tracy

Drug Metab Dispos· October 2006


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