Publications by authors named "David M Perrin"

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Baited SELEX: Drug-Directed Selection of Aptamers to PSMA for Targeting of Prostate Cancer Xenografts in Mice.
Kun Liu, Nicole Robinson, Emirhan Tekoglu, Jerome Lozada, Ivan Pak Lok Yu, David M Perrin

J Am Chem Soc· November 2025

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Synthesis and Preclinical Evaluation of Dual-Mode Fluorescent F-PET Tracers Targeting PSMA.
Jerome Lozada, Helen Merkens, Juliette Froelich, Ruyin Astoria Tai, Kuo-Shyan Lin, David M Perrin

J Med Chem· August 2025

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Chemoselective, regioselective, and positionally selective fluorogenic stapling of unprotected peptides for cellular uptake and direct cell imaging.
Naysilla L Dayanara, Juliette Froelich, Pascale Roome, David M Perrin

Chem Sci· January 2025

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Synthesis of (2,3,4)-Dihydroxyisoleucine for Use in Amatoxin Synthesis.
Shambhu Deo Chandra, Shanal Gunasekera, Benjamin Philipp Noichl, Brian O Patrick, David M Perrin

J Org Chem· September 2024

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5-Hydroxypyrroloindoline Affords Tryptathionine and 2,2'-bis-Indole Peptide Staples: Application to Melanotan-II.
Mihajlo Todorovic, Antoine Blanc, Zhou Wang, Jerome Lozada, Juliette Froelich, David M Perrin

Chemistry· April 2024

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Diphenylphosphinylhydroxylamine (DPPH) Affords Late-Stage S-imination to access free-NH Sulfilimines and Sulfoximines.
Shanal Gunasekera, Alla Pryyma, Jimin Jung, Rebekah Greenwood, Brian O Patrick, David M Perrin

Angew Chem Int Ed Engl· March 2024

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Toward tryptathionine-stapled one-bead-one-compound (OBOC) libraries: solid phase synthesis of a bioactive octretoate analog.
Antoine Blanc, Mihajlo Todorovic, Iulia Dude, Helen Merkens, François Bénard, David M Perrin

Org Biomol Chem· October 2023

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Imidazolium-methylene-trifluoroborate: A novel radioprosthetic group validated with preclinical F-Positron Emission Tomography imaging of Prostate Specific Membrane Antigen in mice.
Jerome Lozada, Hsiou-Ting Kuo, Wen Xuan Lin, Kuo-Shyan Lin, François Bénard, David M Perrin

J Labelled Comp Radiopharm· May 2023

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Salt Metathesis: Tetrafluoroborate Anion Rapidly Fluoridates Organoboronic Acids to give Organotrifluoroborates.
Jerome Lozada, Wen Xuan Lin, Rosana M Cao-Shen, Ruyin Astoria Tai, David M Perrin

Angew Chem Int Ed Engl· April 2023

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The "Ins and Outs" of Prostate Specific Membrane Antigen (PSMA) as Specific Target in Prostate Cancer Therapy.
Felipe Eltit, Nicole Robinson, Pak Lok Ivan Yu, Mitali Pandey, Jerome Lozada, David M Perrin

Adv Exp Med Biol· April 2023

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Rationally Designed Amanitins Achieve Enhanced Cytotoxicity.
Mihajlo Todorovic, Paul Rivollier, Antonio A W L Wong, Zhou Wang, Alla Pryyma, David M Perrin

J Med Chem· August 2022

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Selection of M -Independent RNA-Cleaving DNAzymes with Side-Chains Mimicking Arginine and Lysine.
Somdeb Paul, Antonio A W L Wong, Leo T Liu, David M Perrin

Chembiochem· March 2022

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Synthesis and preliminary evaluation of octreotate conjugates of bioactive synthetic amatoxins for targeting somatostatin receptor (sstr2) expressing cells.
Alla Pryyma, Kaveh Matinkhoo, Yong Jia Bu, Helen Merkens, Zhengxing Zhang, David M Perrin

RSC Chem Biol· January 2022

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Chiral Benzothiazole Monofluoroborate Featuring Chiroptical and Oxygen-Sensitizing Properties: Synthesis and Photophysical Studies.
Omar Sadek, Laura Abad Galán, Frédéric Gendron, Bruno Baguenard, Stephan Guy, David M Perrin

J Org Chem· September 2021

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Synthesis and evaluation of "", a photocaged amatoxin prodrug for light-activated RNA Pol II inhibition and cell death.
Kaveh Matinkhoo, Alla Pryyma, Antonio A W L Wong, David M Perrin

Chem Commun (Camb)· September 2021

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Design, Synthesis, and Biochemical Evaluation of Alpha-Amanitin Derivatives Containing Analogs of the trans-Hydroxyproline Residue for Potential Use in Antibody-Drug Conjugates.
Kaveh Matinkhoo, Antonio A W L Wong, Chido M Hambira, Brandon Kato, Charlie Wei, David M Perrin

Chemistry· July 2021

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FlICk (fluorescent isoindole crosslinking) for peptide stapling.
Mihajlo Todorovic, David M Perrin

Methods Enzymol· June 2021

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Scaling Amatoxin Synthesis with an Improved Route to (2,3,4)-Dihydroxyisoleucine Exemplified by a Toxic, Clickable α-Amanitin Analogue.
Chido M Hambira, Kaveh Matinkhoo, Alla Pryyma, Brian O Patrick, David M Perrin

J Org Chem· April 2021

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Rapid, High-Yielding Solid-Phase Synthesis of Cathepsin-B Cleavable Linkers for Targeted Cancer Therapeutics.
Alla Pryyma, Shanal Gunasekera, Joshua Lewin, David M Perrin

Bioconjug Chem· December 2020

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A hypothesis for examining dihydroxyacetone, the active component in sunless tanning products, as a topical prophylactic against SARS-COV-2 transmission.
David M Perrin

Med Hypotheses· November 2020

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Meeting key synthetic challenges in amanitin synthesis with a new cytotoxic analog: 5'-hydroxy-6'-deoxy-amanitin.
Alla Pryyma, Kaveh Matinkhoo, Antonio A W L Wong, David M Perrin

Chem Sci· October 2020

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Synthesis and F-radiolabeling of thymidine AMBF conjugates.
Antonio A W L Wong, Jerome Lozada, Mathieu L Lepage, Chengcheng Zhang, Helen Merkens, David M Perrin

RSC Med Chem· May 2020

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Toward F-Labeled Theranostics: A Single Agent that Can Be Labeled with F, Cu, or Lu.
Mathieu L Lepage, Hsiou-Ting Kuo, Áron Roxin, Sungjoon Huh, Zhengxing Zhang, David M Perrin

Chembiochem· April 2020

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Pharmacokinetics, radiation dosimetry, acute toxicity and automated synthesis of [F]AmBF-TATE.
Joseph Lau, Jinhe Pan, Etienne Rousseau, Carlos F Uribe, Sudhakara Reddy Seelam, David M Perrin

EJNMMI Res· March 2020

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Synthesis and Activation of Bench-Stable 3a-Fluoropyrroloindolines as Latent Electrophiles for the Synthesis of C-2-Thiol-Substituted Tryptophans and C-3a-Substituted Pyrroloindolines.
Alla Pryyma, Yong Jia Bu, Yonnie Wai, Brian O Patrick, David M Perrin

Org Lett· October 2019

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