Publications by authors named "Dimitris Georgiadis"

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Guidelines for the Design of Custom Affinity-Based Probes for Metalloproteases.
Marie Launay, Lomane Berthy, Sandra Llamas Rizo, Myrto Athina Balachouti, Dimitris Georgiadis

Methods Mol Biol· January 2026

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Targeted approach to determine the impact of cancer-associated protease variants.
Kira Bickenbach, Nele David, Tomas Koudelka, Corentin Joos, Franka Scharfenberg, Dimitris Georgiadis

Sci Adv· February 2025

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Covalent Labeling of Matrix Metalloproteases with Affinity-Based Probes Containing Tuned Reactive N-Acyl-N-Alkyl Sulfonamide Cleavable Linkers.
Laurent Devel, Carole Malgorn, Regis-William Tohon, Marie Launay, Konstantinos Patiniotis, Dimitris Georgiadis

Chembiochem· December 2024

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Discovery of the First-in-Class Inhibitors of Hypoxia Up-Regulated Protein 1 (HYOU1) Suppressing Pathogenic Fibroblast Activation.
Dimitra Papadopoulou, Vasiliki Mavrikaki, Filippos Charalampous, Christos Tzaferis, Martina Samiotaki, Dimitris Georgiadis

Angew Chem Int Ed Engl· April 2024

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Diastereoselective Synthesis of Phosphinic Dipeptide Isosteres: Domino Chirality Transfer during a Stereocontrolled P-Michael Reaction.
Angelos Lelis, Nikolaos Skoulikas, Mirto Papathanasopoulou, Kostas Voreakos, Dimitris Georgiadis

Org Lett· September 2023

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Author Correction: Conformational dynamics linked to domain closure and substrate binding explain the ERAP1 allosteric regulation mechanism.
Zachary Maben, Richa Arya, Dimitris Georgiadis, Efstratios Stratikos, Lawrence J Stern

Nat Commun· March 2023

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Phosphinic Peptides as Tool Compounds for the Study of Pharmacologically Relevant Zn-Metalloproteases.
Dimitris Georgiadis, Nikolaos Skoulikas, Athanasios Papakyriakou, Efstratios Stratikos

ACS Pharmacol Transl Sci· December 2022

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ERAP2 Inhibition Induces Cell-Surface Presentation by MOLT-4 Leukemia Cancer Cells of Many Novel and Potentially Antigenic Peptides.
Ioannis Temponeras, George Stamatakis, Martina Samiotaki, Dimitris Georgiadis, Harris Pratsinis

Int J Mol Sci· February 2022

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Inhibitor-Dependent Usage of the S1' Specificity Pocket of ER Aminopeptidase 2.
Anastasia Mpakali, Dimitris Georgiadis, Efstratios Stratikos, Petros Giastas

ACS Med Chem Lett· February 2022

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Practical Synthesis of Phosphinic Dipeptides by Tandem Esterification of Aminophosphinic and Acrylic Acids under Silylating Conditions.
Paraskevi Kokkala, Kostas Voreakos, Angelos Lelis, Konstantinos Patiniotis, Nikolaos Skoulikas, Dimitris Georgiadis

Molecules· February 2022

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Conformational dynamics linked to domain closure and substrate binding explain the ERAP1 allosteric regulation mechanism.
Zachary Maben, Richa Arya, Dimitris Georgiadis, Efstratios Stratikos, Lawrence J Stern

Nat Commun· September 2021

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Ligand-Directed Modification of Active Matrix Metalloproteases: Activity-based Probes with no Photolabile Group.
Monika Kaminska, Pierrick Bruyat, Carole Malgorn, Marion Doladilhe, Evelyne Cassar-Lajeunesse, Dimitris Georgiadis

Angew Chem Int Ed Engl· August 2021

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The ERAP1 active site cannot productively access the N-terminus of antigenic peptide precursors stably bound onto MHC class I.
George Mavridis, Anastasia Mpakali, Jerome Zoidakis, Manousos Makridakis, Antonia Vlahou, Dimitris Georgiadis

Sci Rep· August 2021

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A Carbodiimide-Mediated P-C Bond-Forming Reaction: Mild Amidoalkylation of -Nucleophiles by Boc-Aminals.
Paraskevi Kokkala, Thayalan Rajeshkumar, Anastasia Mpakali, Efstratios Stratikos, Konstantinos D Vogiatzis, Dimitris Georgiadis

Org Lett· March 2021

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A Reliable Enantioselective Route to Mono-Protected N1-Cbz Piperazic Acid Building Block.
Evanthia Papadaki, Dimitris Georgiadis, Michail Tsakos

Molecules· December 2020

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The Discovery of Insulin-Regulated Aminopeptidase (IRAP) Inhibitors: A Literature Review.
Dimitris Georgiadis, Angeliki Ziotopoulou, Eleni Kaloumenou, Angelos Lelis, Antonia Papasava

Front Pharmacol· September 2020

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A systematic re-examination of processing of MHCI-bound antigenic peptide precursors by endoplasmic reticulum aminopeptidase 1.
George Mavridis, Richa Arya, Alexander Domnick, Jerome Zoidakis, Manousos Makridakis, Dimitris Georgiadis

J Biol Chem· May 2020

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Mechanism for antigenic peptide selection by endoplasmic reticulum aminopeptidase 1.
Petros Giastas, Anastasia Mpakali, Athanasios Papakyriakou, Aggelos Lelis, Paraskevi Kokkala, Dimitris Georgiadis

Proc Natl Acad Sci U S A· December 2019

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Novel Matrix Metalloproteinase 12 Selective Radiotracers for Vascular Molecular Imaging.
Jakub Toczek, Thomas Bordenave, Kiran Gona, Hye-Yeong Kim, Fabrice Beau, Dimitris Georgiadis

J Med Chem· November 2019

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Inhibitors of ER Aminopeptidase 1 and 2: From Design to Clinical Application.
Dimitris Georgiadis, Anastasia Mpakali, Despoina Koumantou, Efstratios Stratikos

Curr Med Chem· September 2019

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Editing the immunopeptidome of melanoma cells using a potent inhibitor of endoplasmic reticulum aminopeptidase 1 (ERAP1).
Despoina Koumantou, Eilon Barnea, Adrian Martin-Esteban, Zachary Maben, Athanasios Papakyriakou, Dimitris Georgiadis

Cancer Immunol Immunother· August 2019

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Late-Stage Diversification of Phosphinic Dehydroalanine Pseudopeptides Based on a Giese-Type Radical C-Alkylation Strategy.
Kostas Voreakos, Laurent Devel, Dimitris Georgiadis

Org Lett· June 2019

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Synthesis and Structural/Functional Characterization of Selective M14 Metallocarboxypeptidase Inhibitors Based on Phosphinic Pseudopeptide Scaffold: Implications on the Design of Specific Optical Probes.
Giovanni Covaleda, Pablo Gallego, Josep Vendrell, Dimitris Georgiadis, Julia Lorenzo

J Med Chem· February 2019

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Ligand-Induced Conformational Change of Insulin-Regulated Aminopeptidase: Insights on Catalytic Mechanism and Active Site Plasticity.
Anastasia Mpakali, Emmanuel Saridakis, Karl Harlos, Yuguang Zhao, Paraskevi Kokkala, Dimitris Georgiadis

J Med Chem· April 2017

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Critical Role of Interdomain Interactions in the Conformational Change and Catalytic Mechanism of Endoplasmic Reticulum Aminopeptidase 1.
Athanasios Stamogiannos, Zachary Maben, Athanasios Papakyriakou, Anastasia Mpakali, Paraskevi Kokkala, Dimitris Georgiadis

Biochemistry· March 2017

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