Publications by authors named "Emilia Caselli"

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Boronate-Based Inhibitors of Penicillin-Binding Proteins: An Underestimated Avenue for Antibiotic Discovery?
Valentina Villamil, Luca Svolacchia Brusoni, Fabio Prati, Emilia Caselli, Nicolò Santi

Pharmaceuticals (Basel)· September 2025

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Resistance to oxyimino-cephalosporins conferred by an alternative mechanism of hydrolysis by the -derived cephalosporinase-33 (ADC-33), a class C β-lactamase present in carbapenem-resistant (CR).
Rachel A Powers, Bradley J Wallar, Hannah R Jarvis, Zoe X Ziegler, Cynthia M June, Emilia Caselli

mBio· June 2025

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Discovery of Boronic Acids-Based β-Lactamase Inhibitors Through In Situ Click Chemistry.
Nicolò Santi, Alessandra Piccirilli, Federico Corsini, Magdalena A Taracila, Mariagrazia Perilli, Emilia Caselli

Int J Mol Sci· April 2025

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Restoring cefepime activity against multidrug-resistant KPC-producing by combination with boronic acid inhibitors, MB076 and S02030.
Laura J Rojas, Travis B Nielsen, Paul Pantapalangkoor, Magdalena A Taracila, Maria L Introvigne, Emilia Caselli

Antimicrob Agents Chemother· March 2025

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α-Triazolylboronic Acids: A Novel Scaffold to Target FLT3 in AML.
Maria Luisa Introvigne, Lorenza Destro, Luca Mologni, Valentina Crippa, Paolo Zardi, Emilia Caselli

ChemMedChem· January 2025

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Natural protein engineering in the Ω-loop: the role of Y221 in ceftazidime and ceftolozane resistance in -derived cephalosporinase.
Andrew R Mack, Vijay Kumar, Magdalena A Taracila, Maria F Mojica, Margaret O'Shea, Emilia Caselli

Antimicrob Agents Chemother· November 2023

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Synthesis of a Novel Boronic Acid Transition State Inhibitor, MB076: A Heterocyclic Triazole Effectively Inhibits -Derived Cephalosporinase Variants with an Expanded-Substrate Spectrum.
Rachel A Powers, Cynthia M June, Micah C Fernando, Erin R Fish, Olivia L Maurer, Emilia Caselli

J Med Chem· July 2023

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Defining the minimum inhibitory concentration of 22 rifamycins in iron limited, physiologic medium against Acinetobacter baumannii, Escherichia coli, and Klebsiella pneumoniae clinical isolates.
Peggy Lu, Francesco Alletto, Bosul Lee, Elizabeth Burk, Jasmine Martinez, Emilia Caselli

PLoS One· June 2023

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Sulfonamidoboronic Acids as "Cross-Class" Inhibitors of an Expanded-Spectrum Class C Cephalosporinase, ADC-33, and a Class D Carbapenemase, OXA-24/40: Strategic Compound Design to Combat Resistance in .
Maria Luisa Introvigne, Trevor J Beardsley, Micah C Fernando, David A Leonard, Bradley J Wallar, Emilia Caselli

Antibiotics (Basel)· March 2023

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Boronic Acid Transition State Inhibitors as Potent Inactivators of KPC and CTX-M β-Lactamases: Biochemical and Structural Analyses.
Tahani A Alsenani, María Margarita Rodríguez, Barbara Ghiglione, Magdalena A Taracila, Maria F Mojica, Emilia Caselli

Antimicrob Agents Chemother· January 2023

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Insights Into the Inhibition of MOX-1 β-Lactamase by S02030, a Boronic Acid Transition State Inhibitor.
Tatsuya Ishikawa, Nayuta Furukawa, Emilia Caselli, Fabio Prati, Magdalena A Taracila

Front Microbiol· December 2021

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Straightforward synthesis of chiral non-racemic α-boryl isocyanides.
Francesco Fini, Alessandro Zanni, Maria Luisa Introvigne, Mattia Stucchi, Emilia Caselli

Org Biomol Chem· August 2021

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A comprehensive and contemporary "snapshot" of β-lactamases in carbapenem resistant Acinetobacter baumannii.
Andrea M Hujer, Kristine M Hujer, David A Leonard, Rachel A Powers, Bradley J Wallar, Emilia Caselli

Diagn Microbiol Infect Dis· February 2021

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Structural Insights into Inhibition of the Acinetobacter-Derived Cephalosporinase ADC-7 by Ceftazidime and Its Boronic Acid Transition State Analog.
Brandy N Curtis, Kali A Smolen, Sara J Barlow, Emilia Caselli, Fabio Prati

Antimicrob Agents Chemother· November 2020

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α-Triazolylboronic Acids: A Promising Scaffold for Effective Inhibitors of KPCs.
Maria Luisa Introvigne, Magdalena A Taracila, Fabio Prati, Emilia Caselli, Robert A Bonomo

ChemMedChem· July 2020

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1,2,3-Triazolylmethaneboronate: A Structure Activity Relationship Study of a Class of β-Lactamase Inhibitors against Cephalosporinase.
Emilia Caselli, Francesco Fini, Maria Luisa Introvigne, Mattia Stucchi, Magdalena A Taracila

ACS Infect Dis· July 2020

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Structures of FOX-4 Cephamycinase in Complex with Transition-State Analog Inhibitors.
Scott T Lefurgy, Emilia Caselli, Magdalena A Taracila, Vladimir N Malashkevich, Beena Biju

Biomolecules· April 2020

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The β-Lactamase Inhibitor Boronic Acid Derivative SM23 as a New Anti- Biofilm.
Samuele Peppoloni, Eva Pericolini, Bruna Colombari, Diego Pinetti, Claudio Cermelli, Emilia Caselli

Front Microbiol· February 2020

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Deciphering the Evolution of Cephalosporin Resistance to Ceftolozane-Tazobactam in Pseudomonas aeruginosa.
Melissa D Barnes, Magdalena A Taracila, Joseph D Rutter, Christopher R Bethel, Ioannis Galdadas, Emilia Caselli

mBio· December 2018

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Structure-Based Analysis of Boronic Acids as Inhibitors of Acinetobacter-Derived Cephalosporinase-7, a Unique Class C β-Lactamase.
Alexandra A Bouza, Hollister C Swanson, Kali A Smolen, Alison L VanDine, Magdalena A Taracila, Emilia Caselli

ACS Infect Dis· March 2018

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Inhibition of Acinetobacter-Derived Cephalosporinase: Exploring the Carboxylate Recognition Site Using Novel β-Lactamase Inhibitors.
Emilia Caselli, Chiara Romagnoli, Rachel A Powers, Magdalena A Taracila, Alexandra A Bouza

ACS Infect Dis· March 2018

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Crystal Structures of KPC-2 and SHV-1 β-Lactamases in Complex with the Boronic Acid Transition State Analog S02030.
Nhu Q Nguyen, Nikhil P Krishnan, Laura J Rojas, Fabio Prati, Emilia Caselli

Antimicrob Agents Chemother· January 2016

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Boronic Acid Transition State Inhibitors Active against KPC and Other Class A β-Lactamases: Structure-Activity Relationships as a Guide to Inhibitor Design.
Laura J Rojas, Magdalena A Taracila, Krisztina M Papp-Wallace, Christopher R Bethel, Emilia Caselli

Antimicrob Agents Chemother· January 2016

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Click Chemistry in Lead Optimization of Boronic Acids as β-Lactamase Inhibitors.
Emilia Caselli, Chiara Romagnoli, Roza Vahabi, Magdalena A Taracila, Robert A Bonomo

J Med Chem· July 2015

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Synthesis of 1,2,3-triazol-1-yl-methaneboronic acids via click chemistry: an easy access to a new potential scaffold for protease inhibitors.
Chiara Romagnoli, Emilia Caselli, Fabio Prati

European J Org Chem· February 2015

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