Publications by authors named "Eric Marsault"

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Discovery of a CCR2-targeting pepducin therapy for chronic pain.
Élora Midavaine, Rebecca L Brouillette, Elizabeth Théberge, Christine E Mona, Sakeen W Kashem, Éric Marsault

Pharmacol Res· July 2024

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Localized apelin-17 analogue-bicelle interactions as a facilitator of membrane-catalyzed receptor recognition and binding.
Trần Thanh Tâm Phạm, Alexandre Murza, Éric Marsault, John P Frampton, Jan K Rainey

Biochim Biophys Acta Biomembr· March 2024

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Insights on Structure-Passive Permeability Relationship in Pyrrole and Furan-Containing Macrocycles.
Huy M Ly, Michael Desgagné, Duc Tai Nguyen, Christian Comeau, Ulrike Froehlich, Éric Marsault

J Med Chem· March 2024

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Apelin stimulation of the vascular skeletal muscle stem cell niche enhances endogenous repair in dystrophic mice.
Emmeran Le Moal, Yuguo Liu, Jasmin Collerette-Tremblay, Simon Dumontier, Paul Fabre, Eric Marsault

Sci Transl Med· March 2024

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Optimization of Ketobenzothiazole-Based Type II Transmembrane Serine Protease Inhibitors to Block H1N1 Influenza Virus Replication.
Éloïc Colombo, Antoine Désilets, Malihe Hassanzadeh, Gabriel Lemieux, Isabelle Marois, Eric Marsault

ChemMedChem· January 2024

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Beyond Rule-of-five: Permeability Assessment of Semipeptidic Macrocycles.
Marion L'Exact, Christian Comeau, Alix Bourhis, Olivier Boisvert, Ulrike Fröhlich, Éric Marsault

Biochim Biophys Acta Biomembr· October 2023

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Apelin prevents diabetes-induced poor collateral vessel formation and blood flow reperfusion in ischemic limb.
Stéphanie Robillard, Kien Trân, Marie-Sophie Lachance, Tristan Brazeau, Elizabeth Boisvert, Éric Marsault

Front Cardiovasc Med· August 2023

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Signaling Modulation via Minimal C-Terminal Modifications of Apelin-13.
Léa Théroux, Robin Van Den Hauwe, Kien Trân, Justin Fournier, Michael Desgagné, Eric Marsault

ACS Pharmacol Transl Sci· February 2023

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A TMPRSS2 inhibitor acts as a pan-SARS-CoV-2 prophylactic and therapeutic.
Tirosh Shapira, I Abrrey Monreal, Sébastien P Dion, David W Buchholz, Brian Imbiakha, Eric Marsault

Nature· May 2022

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Size-Reduced Macrocyclic Analogues of [Pyr]-apelin-13 Showing Negative Gα Bias Still Produce Prolonged Cardiac Effects.
Kien Tran, Xavier Sainsily, Jérôme Côté, David Coquerel, Pierre Couvineau, Éric Marsault

J Med Chem· January 2022

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Apelin-13 in septic shock: effective in supporting hemodynamics in sheep but compromised by enzymatic breakdown in patients.
David Coquerel, Julie Lamoureux, Frédéric Chagnon, Kien Trân, Michael Sage, Eric Marsault

Sci Rep· November 2021

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Pharmacodynamic and pharmacokinetic profiles of a neurotensin receptor type 2 (NTS2) analgesic macrocyclic analog.
Magali Chartier, Michael Desgagné, Marc Sousbie, Charles Rumsby, Lucie Chevillard, Éric Marsault

Biomed Pharmacother· September 2021

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Elabela Protects Spontaneously Hypertensive Rats From Hypertension and Cardiorenal Dysfunctions Exacerbated by Dietary High-Salt Intake.
Xavier Sainsily, David Coquerel, Hugo Giguère, Lauralyne Dumont, Kien Tran, Éric Marsault

Front Pharmacol· July 2021

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Constraining the Side Chain of C-Terminal Amino Acids in Apelin-13 Greatly Increases Affinity, Modulates Signaling, and Improves the Pharmacokinetic Profile.
Kien Trân, Robin Van Den Hauwe, Xavier Sainsily, Pierre Couvineau, Jérôme Côté, Éric Marsault

J Med Chem· May 2021

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Modulation of the Passive Permeability of Semipeptidic Macrocycles: N- and C-Methylations Fine-Tune Conformation and Properties.
Christian Comeau, Benjamin Ries, Thomas Stadelmann, Jacob Tremblay, Sylvain Poulet, Éric Marsault

J Med Chem· May 2021

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A novel highly potent inhibitor of TMPRSS2-like proteases blocks SARS-CoV-2 variants of concern and is broadly protective against infection and mortality in mice.
Tirosh Shapira, I Abrrey Monreal, Sébastien P Dion, Mason Jager, Antoine Désilets, Eric Marsault

bioRxiv· May 2021

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Gαi-biased apelin analog protects against isoproterenol-induced myocardial dysfunction in rats.
David Coquerel, Eugénie Delile, Lauralyne Dumont, Frédéric Chagnon, Alexandre Murza, Eric Marsault

Am J Physiol Heart Circ Physiol· April 2021

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Design, Structural Optimization, and Characterization of the First Selective Macrocyclic Neurotensin Receptor Type 2 Non-opioid Analgesic.
Magali Chartier, Michael Desgagné, Marc Sousbie, Jérôme Côté, Jean-Michel Longpré, Eric Marsault

J Med Chem· February 2021

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Structure-Activity Relationship and Bioactivity of Short Analogues of ELABELA as Agonists of the Apelin Receptor.
Kien Trân, Alexandre Murza, Xavier Sainsily, Eugénie Delile, Pierre Couvineau, Éric Marsault

J Med Chem· January 2021

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Inhibitors of type II transmembrane serine proteases in the treatment of diseases of the respiratory tract - A review of patent literature.
Alexandre Murza, Sébastien P Dion, Pierre-Luc Boudreault, Antoine Désilets, Richard Leduc, Éric Marsault

Expert Opin Ther Pat· November 2020

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Structure-Permeability Relationship of Semipeptidic Macrocycles-Understanding and Optimizing Passive Permeability and Efflux Ratio.
Antoine Le Roux, Émilie Blaise, Pierre-Luc Boudreault, Christian Comeau, Annie Doucet, Eric Marsault

J Med Chem· July 2020

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Cell-penetrating pepducins targeting the neurotensin receptor type 1 relieve pain.
Rebecca L Brouillette, Élie Besserer-Offroy, Christine E Mona, Magali Chartier, Sandrine Lavenus, Éric Marsault

Pharmacol Res· May 2020

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Bactericidal Activity of the Bacterial ATP Synthase Inhibitor Tomatidine and the Combination of Tomatidine and Aminoglycoside Against Persistent and Virulent Forms of .
Jean-Philippe Langlois, Guillaume Millette, Isabelle Guay, Alexis Dubé-Duquette, Suzanne Chamberland, Éric Marsault

Front Microbiol· May 2020

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Discovery and Development of TMPRSS6 Inhibitors Modulating Hepcidin Levels in Human Hepatocytes.
François Béliveau, Aarti Tarkar, Sébastien P Dion, Antoine Désilets, Mariana Gabriela Ghinet, Éric Marsault

Cell Chem Biol· November 2019

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L-type prostaglandin D synthase regulates the trafficking of the PGD DP1 receptor by interacting with the GTPase Rab4.
Chantal Binda, Samuel Génier, Jade Degrandmaison, Samuel Picard, Louis Fréchette, Eric Marsault

J Biol Chem· November 2019

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