Publications by authors named "Gilberto Spadoni"

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N-Acylaminoethyltetrahydroquinolines: A new class of melatonin receptor ligands with in vivo activity on glioblastoma.
Annalida Bedini, Francesca Galvani, Gian Marco Elisi, Laura Scalvini, Michele Mari, Gilberto Spadoni

Eur J Med Chem· February 2026

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Industrial and academic approaches to the search for alternative melatonin receptor ligands: An historical survey.
Annalida Bedini, Jean A Boutin, Céline Legros, Darius P Zlotos, Gilberto Spadoni

J Pineal Res· May 2024

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Binding and unbinding of potent melatonin receptor ligands: Mechanistic simulations and experimental evidence.
Annalida Bedini, Gian Marco Elisi, Fabiola Fanini, Michele Retini, Laura Scalvini, Gilberto Spadoni

J Pineal Res· March 2024

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NAAA-regulated lipid signaling in monocytes controls the induction of hyperalgesic priming in mice.
Yannick Fotio, Alex Mabou Tagne, Erica Squire, Hye-Lim Lee, Connor M Phillips, Gilberto Spadoni

Nat Commun· February 2024

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2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT and MT receptors.
Michele Mari, Gian Marco Elisi, Annalida Bedini, Simone Lucarini, Michele Retini, Gilberto Spadoni

Eur J Med Chem· December 2022

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Radiosynthesis and Evaluation of Four Positron Emission Tomography Tracer Candidates for Imaging of Melatonin Receptors.
Hussein Bdair, Thomas A Singleton, Karen Ross, Dean Jolly, Min Su Kang, Gilberto Spadoni

ACS Chem Neurosci· May 2022

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In silico drug discovery of melatonin receptor ligands with therapeutic potential.
Gian Marco Elisi, Laura Scalvini, Alessio Lodola, Annalida Bedini, Gilberto Spadoni

Expert Opin Drug Discov· April 2022

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Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma.
Riccardo Castelli, Sara Taranto, Lucia Furiassi, Nicole Bozza, Giuseppe Marseglia, Gilberto Spadoni

Eur J Med Chem· October 2021

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N-(Anilinoethyl)amide Melatonergic Ligands with Improved Water Solubility and Metabolic Stability.
Francesca Ferlenghi, Michele Mari, Gabriella Gobbi, Gian Marco Elisi, Marco Mor, Gilberto Spadoni

ChemMedChem· October 2021

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NAAA-regulated lipid signaling governs the transition from acute to chronic pain.
Yannick Fotio, Kwang-Mook Jung, Francesca Palese, Andre Obenaus, Alex Mabou Tagne, Gilberto Spadoni

Sci Adv· October 2021

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New classes of potent heparanase inhibitors from ligand-based virtual screening.
Daniele Pala, Laura Scalvini, Gian Marco Elisi, Alessio Lodola, Marco Mor, Gilberto Spadoni

J Enzyme Inhib Med Chem· December 2020

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Chiral Recognition of Flexible Melatonin Receptor Ligands Induced by Conformational Equilibria.
Gian Marco Elisi, Annalida Bedini, Laura Scalvini, Caterina Carmi, Silvia Bartolucci, Gilberto Spadoni

Molecules· September 2020

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-Acylethanolamine Acid Amidase (NAAA): Structure, Function, and Inhibition.
Daniele Piomelli, Laura Scalvini, Yannick Fotio, Alessio Lodola, Gilberto Spadoni

J Med Chem· July 2020

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Antidepressant-like effects of pharmacological inhibition of FAAH activity in socially isolated female rats.
Luca Carnevali, Rosario Statello, Federica Vacondio, Francesca Ferlenghi, Gilberto Spadoni

Eur Neuropsychopharmacol· March 2020

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New Antimicrobials Targeting Bacterial RNA Polymerase Holoenzyme Assembly Identified with an BRET-Based Discovery Platform.
Sara Sartini, Elisabetta Levati, Martina Maccesi, Matteo Guerra, Gilberto Spadoni

ACS Chem Biol· August 2019

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Melatonin MT and MT Receptors Exhibit Distinct Effects in the Modulation of Body Temperature across the Light/Dark Cycle.
Martha López-Canul, Seung Hyun Min, Luca Posa, Danilo De Gregorio, Annalida Bedini, Gilberto Spadoni

Int J Mol Sci· May 2019

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Design, Synthesis, and Biological Activity of Hydrogen Peroxide Responsive Arylboronate Melatonin Hybrids.
Annalida Bedini, Alessandra Fraternale, Rita Crinelli, Michele Mari, Silvia Bartolucci, Gilberto Spadoni

Chem Res Toxicol· January 2019

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Identification of Bivalent Ligands with Melatonin Receptor Agonist and Fatty Acid Amide Hydrolase (FAAH) Inhibitory Activity That Exhibit Ocular Hypotensive Effect in the Rabbit.
Gilberto Spadoni, Annalida Bedini, Lucia Furiassi, Michele Mari, Marco Mor

J Med Chem· September 2018

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Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands.
Silvia Rivara, Laura Scalvini, Alessio Lodola, Marco Mor, Daniel-Henri Caignard, Gilberto Spadoni

J Med Chem· April 2018

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Antiproliferative and pro-apoptotic activity of melatonin analogues on melanoma and breast cancer cells.
Giuliana Gatti, Valeria Lucini, Silvana Dugnani, Angela Calastretti, Gilberto Spadoni

Oncotarget· September 2017

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Cardioprotective effects of fatty acid amide hydrolase inhibitor URB694, in a rodent model of trait anxiety.
Luca Carnevali, Federica Vacondio, Stefano Rossi, Emilio Macchi, Gilberto Spadoni

Sci Rep· December 2015

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Antidepressant-like activity and cardioprotective effects of fatty acid amide hydrolase inhibitor URB694 in socially stressed Wistar Kyoto rats.
Luca Carnevali, Federica Vacondio, Stefano Rossi, Sergio Callegari, Emilio Macchi, Gilberto Spadoni

Eur Neuropsychopharmacol· November 2015

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Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines.
Gilberto Spadoni, Annalida Bedini, Simone Lucarini, Michele Mari, Daniel-Henri Caignard

J Med Chem· September 2015

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Pharmacokinetic and pharmacodynamic evaluation of ramelteon : an insomnia therapy.
Gilberto Spadoni, Annalida Bedini, Simone Lucarini, Marco Mor, Silvia Rivara

Expert Opin Drug Metab Toxicol· July 2015

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Iridium-catalyzed direct synthesis of tryptamine derivatives from indoles: exploiting n-protected β-amino alcohols as alkylating agents.
Silvia Bartolucci, Michele Mari, Annalida Bedini, Giovanni Piersanti, Gilberto Spadoni

J Org Chem· March 2015

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