Publications by authors named "Hollis D Showalter"

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Optimization of Benzoxazinorifamycins to Minimize hPXR Activation for the Treatment of Tuberculosis and HIV Coinfection.
Shireen R Ashkar, Walajapet Rajeswaran, Pil H Lee, Larisa Yeomans, Claire M Thrasher, Hollis D Showalter

ACS Infect Dis· August 2022

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Optimization of Benzoxazinorifamycins to Improve RNA Polymerase Inhibition and Treatment of Tuberculosis.
Walajapet Rajeswaran, Shireen R Ashkar, Pil H Lee, Larisa Yeomans, Yeonoh Shin, Hollis D Showalter

ACS Infect Dis· August 2022

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Recent Progress in the Discovery and Development of 2-Nitroimidazooxazines and 6-Nitroimidazooxazoles to Treat Tuberculosis and Neglected Tropical Diseases.
Hollis D Showalter

Molecules· September 2020

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Synthesis and structure-activity relationships of thieno[2,3-d]pyrimidines as atypical protein kinase C inhibitors to control retinal vascular permeability and cytokine-induced edema.
Xuwen Liu, Michael W Wilson, Kun Liu, Pil Lee, Larisa Yeomans, Hollis D Showalter

Bioorg Med Chem· June 2020

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Perturbation of ubiquitin homeostasis promotes macrophage oxidative defenses.
Marie-Eve Charbonneau, Karla D Passalacqua, Susan E Hagen, Hollis D Showalter, Christiane E Wobus

Sci Rep· July 2019

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A concise synthesis of 3-substituted-7-amino-6-carboxyl-8-azachromones.
Xinmin Gan, Hollis D Showalter

Tetrahedron Lett· July 2019

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Altered Domain Structure of the Prion Protein Caused by Cu Binding and Functionally Relevant Mutations: Analysis by Cross-Linking, MS/MS, and NMR.
Alex J McDonald, Deborah R Leon, Kathleen A Markham, Bei Wu, Christian F Heckendorf, Hollis D Showalter

Structure· June 2019

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Synthesis of deuterium-labelled amlexanox and its metabolic stability against mouse, rat, and human microsomes.
Xinmin Gan, Michael W Wilson, Tyler S Beyett, Bo Wen, Duxin Sun, Hollis D Showalter

J Labelled Comp Radiopharm· May 2019

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Revisiting the role of dihydroorotate dehydrogenase as a therapeutic target for cancer.
Joseph T Madak, Armand Bankhead, Christine R Cuthbertson, Hollis D Showalter, Nouri Neamati

Pharmacol Ther· March 2019

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Design, synthesis, and biological activity of substituted 2-amino-5-oxo-5H-chromeno[2,3-b]pyridine-3-carboxylic acid derivatives as inhibitors of the inflammatory kinases TBK1 and IKKε for the treatment of obesity.
Tyler S Beyett, Xinmin Gan, Shannon M Reilly, Andrew V Gomez, Louise Chang, Hollis D Showalter

Bioorg Med Chem· November 2018

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Carboxylic Acid Derivatives of Amlexanox Display Enhanced Potency toward TBK1 and IKK and Reveal Mechanisms for Selective Inhibition.
Tyler S Beyett, Xinmin Gan, Shannon M Reilly, Louise Chang, Andrew V Gomez, Hollis D Showalter

Mol Pharmacol· October 2018

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Synthesis of CID-cleavable protein crosslinking agents containing quaternary amines for structural mass spectrometry.
Susan E Hagen, Kun Liu, Yafei Jin, Lolita Piersimoni, Philip C Andrews, Hollis D Showalter

Org Biomol Chem· September 2018

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Design, Synthesis, and Biological Evaluation of 4-Quinoline Carboxylic Acids as Inhibitors of Dihydroorotate Dehydrogenase.
Joseph T Madak, Christine R Cuthbertson, Yoshinari Miyata, Shuzo Tamura, Elyse M Petrunak, Hollis D Showalter

J Med Chem· June 2018

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Design, Synthesis, and Characterization of Brequinar Conjugates as Probes to Study DHODH Inhibition.
Joseph T Madak, Christine R Cuthbertson, Wenmin Chen, Hollis D Showalter, Nouri Neamati

Chemistry· October 2017

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Direct and Systemic Administration of a CNS-Permeant Tamoxifen Analog Reduces Amphetamine-Induced Dopamine Release and Reinforcing Effects.
Colleen Carpenter, Alexander G Zestos, Rachel Altshuler, Roderick J Sorenson, Bipasha Guptaroy, Hollis D Showalter

Neuropsychopharmacology· September 2017

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Design, synthesis, and biological activity of 5'-phenyl-1,2,5,6-tetrahydro-3,3'-bipyridine analogues as potential antagonists of nicotinic acetylcholine receptors.
Yafei Jin, Xiaoqin Huang, Roger L Papke, Emily M Jutkiewicz, Hollis D Showalter

Bioorg Med Chem Lett· September 2017

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Vesicular Glutamate Transporter Inhibitors: Structurally Modified Brilliant Yellow Analogs.
Jason Kehrl, J Christian Althaus, Hollis D Showalter, DiAndra M Rudzinski, Michael A Sutton

Neurochem Res· June 2017

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Design and synthesis of triarylacrylonitrile analogues of tamoxifen with improved binding selectivity to protein kinase C.
Colleen Carpenter, Roderick J Sorenson, Yafei Jin, Szymon Klossowski, Tomasz Cierpicki, Hollis D Showalter

Bioorg Med Chem· November 2016

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Anti-infective Activity of 2-Cyano-3-Acrylamide Inhibitors with Improved Drug-Like Properties against Two Intracellular Pathogens.
Karla D Passalacqua, Marie-Eve Charbonneau, Nicholas J Donato, Hollis D Showalter, Duxin Sun

Antimicrob Agents Chemother· July 2016

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Small molecule deubiquitinase inhibitors promote macrophage anti-infective capacity.
Marie-Eve Charbonneau, Marta J Gonzalez-Hernandez, Hollis D Showalter, Nicholas J Donato, Christiane E Wobus

PLoS One· November 2015

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Substrate-Competitive Activity-Based Profiling of Ester Prodrug Activating Enzymes.
Hao Xu, Jaimeen D Majmudar, Dahvid Davda, Phani Ghanakota, Ki H Kim, Hollis D Showalter

Mol Pharm· September 2015

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Novel carboxaldehyde mediated synthetic pathway for 5'-amino adenosine analogues.
Garrett S Gibbons, Hollis D Showalter, Zaneta Nikolovska-Coleska

Nucleosides Nucleotides Nucleic Acids· August 2015

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Targeting deubiquitinase activity with a novel small-molecule inhibitor as therapy for B-cell malignancies.
Luke F Peterson, Hanshi Sun, Yihong Liu, Harish Potu, Malathi Kandarpa, Hollis D Showalter

Blood· June 2015

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Chemical derivatives of a small molecule deubiquitinase inhibitor have antiviral activity against several RNA viruses.
Marta J Gonzalez-Hernandez, Anupama Pal, Kofi E Gyan, Marie-Eve Charbonneau, Hollis D Showalter

PLoS One· December 2014

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RecO and RecR are necessary for RecA loading in response to DNA damage and replication fork stress.
Justin S Lenhart, Eileen R Brandes, Jeremy W Schroeder, Roderick J Sorenson, Hollis D Showalter

J Bacteriol· August 2014

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