Publications by authors named "Janos Sapi"

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Inhibition of Recruitment and Activation of Neutrophils by Pyridazinone-Scaffold-Based Compounds.
Aurélie Moniot, Julien Braux, Renaud Siboni, Christine Guillaume, Sandra Audonnet, Janos Sapi

Int J Mol Sci· June 2022

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Pyridazinone Derivatives Limit Osteosarcoma-Cells Growth In Vitro and In Vivo.
Aurélie Moniot, Julien Braux, Camille Bour, Christine Guillaume, Fabien Lamret, Janos Sapi

Cancers (Basel)· November 2021

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Conjugates of Ultrasmall Quantum Dots and Acridine Derivatives as Prospective Nanoprobes for Intracellular Investigations.
Pavel Linkov, Pavel Samokhvalov, Maria Baryshnikova, Marie Laronze-Cochard, Janos Sapi

Nanomaterials (Basel)· August 2021

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Pyridazinone derivatives as potential anti-inflammatory agents: synthesis and biological evaluation as PDE4 inhibitors.
Ingrid Allart-Simon, Aurélie Moniot, Nicolo Bisi, Miguel Ponce-Vargas, Sandra Audonnet, Janos Sapi

RSC Med Chem· April 2021

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5-Arylisothiazol-3(2H)-one-1,(1)-(di)oxides: A new class of selective tumor-associated carbonic anhydrases (hCA IX and XII) inhibitors.
Benedetta Cornelio, Marie Laronze-Cochard, Raimundo Miambo, Michela De Grandis, Rossana Riccioni, Janos Sapi

Eur J Med Chem· August 2019

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Unexpected effect of cyclodepsipeptides bearing a sulfonylhydrazide moiety towards histone deacetylase activity.
Mathieu Létévé, Céline Gonzalez, Gautier Moroy, Agathe Martinez, Jérôme Jeanblanc, Janos Sapi

Bioorg Chem· December 2018

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Synthesis and biological evaluation of pyridazinone derivatives as potential anti-inflammatory agents.
Chantal Barberot, Aurélie Moniot, Ingrid Allart-Simon, Laurette Malleret, Tatiana Yegorova, Janos Sapi

Eur J Med Chem· February 2018

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The 52 International Conference on Medicinal Chemistry (RICT 2016) of the French Medicinal Chemistry Society (SCT) Held in Caen (Normandy).
Janos Sapi, Luc Van Hijfte, Patrick Dallemagne

ChemMedChem· June 2017

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Structure-Activity Relationships of Benzenesulfonamide-Based Inhibitors towards Carbonic Anhydrase Isoform Specificity.
Avni Bhatt, Brian P Mahon, Vinicius Wilian D Cruzeiro, Benedetta Cornelio, Marie Laronze-Cochard, Janos Sapi

Chembiochem· January 2017

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Radical Smiles Rearrangement: An Update.
Ingrid Allart-Simon, Stéphane Gérard, Janos Sapi

Molecules· July 2016

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Design, Synthesis, and Use of MMP-2 Inhibitor-Conjugated Quantum Dots in Functional Biochemical Assays.
Erika Bourguet, Kristina Brazhnik, Alyona Sukhanova, Gautier Moroy, Sylvie Brassart-Pasco, Janos Sapi

Bioconjug Chem· April 2016

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4-Arylbenzenesulfonamides as Human Carbonic Anhydrase Inhibitors (hCAIs): Synthesis by Pd Nanocatalyst-Mediated Suzuki-Miyaura Reaction, Enzyme Inhibition, and X-ray Crystallographic Studies.
Benedetta Cornelio, Marie Laronze-Cochard, Mariangela Ceruso, Marta Ferraroni, Graham A Rance, Janos Sapi

J Med Chem· January 2016

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In Memoriam: Professor Camille-Georges Wermuth.
Janos Sapi

Eur J Med Chem· January 2016

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Diastereomer Interconversion via Enolization: A Case Study.
Andrea Renzetti, Antonello Di Crescenzo, Feilin Nie, Andrew D Bond, Stéphane Gérard, Janos Sapi

Chirality· November 2015

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TiCl4-promoted condensation of methyl acetoacetate, isobutyraldehyde, and indole: a theoretical and experimental study.
Andrea Renzetti, Alessandro Marrone, Stéphane Gérard, Janos Sapi, Hiroshi Nakazawa

Phys Chem Chem Phys· April 2015

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Interfacing chemical biology and drug discovery: report from the 50th International Conference on Medicinal Chemistry of the SCT (French Medicinal Chemistry Society), July 2-4, 2014, Rouen, France.
Janos Sapi, Frédéric Schmidt, Luc Van Hijfte, Pascal George

ACS Chem Biol· December 2014

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Photochemical aryl radical cyclizations to give (E)-3-ylideneoxindoles.
Michael Gurry, Ingrid Allart-Simon, Patrick McArdle, Stéphane Gérard, Janos Sapi

Molecules· September 2014

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Chemical biology: contribution to molecular therapeutic innovation--a new role for chemistry? Report from the thematic symposium organized by the SCT (French Medicinal Chemistry Society), November 26th, 2013.
Frédéric Schmidt, Pascal George, Janos Sapi

ACS Chem Biol· April 2014

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Cyclopropyl-tryptamine analogues: synthesis and biological evaluation as 5-HT(6) receptor ligands.
Claude Szalata, Jan Szymoniak, Frédéric Fabis, Sabrina Butt-Gueulle, Sylvain Rault, Janos Sapi

ChemMedChem· January 2013

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Neutrophil elastase as a target in lung cancer.
Gautier Moroy, Alain J P Alix, Janos Sapi, William Hornebeck, Erika Bourguet

Anticancer Agents Med Chem· July 2012

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First domino radical cyclisation/Smiles rearrangement combination.
Marc Pudlo, Ingrid Allart-Simon, Bernard Tinant, Stéphane Gérard, Janos Sapi

Chem Commun (Camb)· February 2012

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Inhibition of human leukocyte elastase, plasmin and matrix metalloproteinases by oleic acid and oleoyl-galardin derivative(s).
Gautier Moroy, Erika Bourguet, Martine Decarme, Janos Sapi, Alain J P Alix

Biochem Pharmacol· March 2011

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The NC1 domain of type XIX collagen inhibits melanoma cell migration.
Aida Toubal, Laurent Ramont, Christine Terryn, Sylvie Brassart-Pasco, Dominique Patigny, Janos Sapi

Eur J Dermatol· February 2011

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Synthesis and biological evaluation of new penta- and heptacyclic indolo- and quinolinocarbazole ring systems obtained via Pd(0) catalysed reductive N-heteroannulation.
Marie Laronze-Cochard, Fabien Cochard, Etienne Daras, Amélie Lansiaux, Bertrand Brassart, Janos Sapi

Org Biomol Chem· October 2010

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Condensation of beta-diester titanium enolates with carbonyl substrates: a combined DFT and experimental investigation.
Alessandro Marrone, Andrea Renzetti, Paolo De Maria, Stéphane Gérard, Janos Sapi

Chemistry· November 2009

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