Publications by authors named "Jean-Denis Docquier"

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Sustainable Joullié-Ugi and Continuous Flow Implementation Led to Novel Captopril-Inspired Broad-Spectrum Metallo-β-Lactamase Inhibitors.
Antonella Ilenia Alfano, Sveva Pelliccia, Simona Barone, Luigi Cutarella, Sacha Michèle Idriss Cancade, Jean Denis Docquier

J Med Chem· August 2025

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SAND: a comprehensive annotation of class D β-lactamases using structural alignment-based numbering.
Fedaa Attana, Soobin Kim, James Spencer, Bogdan I Iorga, Jean-Denis Docquier

Antimicrob Agents Chemother· July 2025

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Synthesis of β-lactam-zidovudine pronucleosides as potential selective narrow-spectrum antibacterial agents.
Miyanou Rosales-Hurtado, Fanny Faure, Filomena Sannio, Federica Verdirosa, Georges Feller, Jean-Denis Docquier

Org Biomol Chem· January 2025

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Extract as a Source of Antimicrobial Compounds: A Circular Bioeconomy Approach.
Roberta Barletta, Alfonso Trezza, Michela Geminiani, Luisa Frusciante, Tommaso Olmastroni, Jean-Denis Docquier

Mar Drugs· November 2024

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4-Trifluoromethyl bithiazoles as broad-spectrum antimicrobial agents for virus-related bacterial infections or co-infections.
Francesca Barbieri, Vincent Carlen, Maria Grazia Martina, Filomena Sannio, Sacha Cancade, Jean-Denis Docquier

RSC Med Chem· May 2024

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An update on antibacterial AlkylGuanidino Ureas: Design of new derivatives, synergism with colistin and data analysis of the whole library.
Claudia Ardino, Filomena Sannio, Giulio Poli, Salvatore Galati, Elena Dreassi, Jean-Denis Docquier

Eur J Med Chem· April 2024

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Perturbation and resilience of the gut microbiome up to 3 months after β-lactams exposure in healthy volunteers suggest an important role of microbial β-lactamases.
Camille d'Humières, Margot Delavy, Laurie Alla, Farid Ichou, Emilie Gauliard, Jean-Denis Docquier

Microbiome· March 2024

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Aurones and derivatives as promising New Delhi metallo-β-lactamase (NDM-1) inhibitors.
Jérémy Caburet, Federica Verdirosa, Matis Moretti, Brayan Roulier, Giorgia Simoncelli, Jean-Denis Docquier

Bioorg Med Chem· January 2024

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Benzenesulfonamide derivatives as carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships.
Marialuigia Fantacuzzi, Ilaria D'Agostino, Simone Carradori, Francesco Liguori, Fabrizio Carta, Jean-Denis Docquier

J Enzyme Inhib Med Chem· December 2023

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Structure-Based Optimization of 1,2,4-Triazole-3-Thione Derivatives: Improving Inhibition of NDM-/VIM-Type Metallo-β-Lactamases and Synergistic Activity on Resistant Bacteria.
Matteo Bersani, Mariacristina Failla, Filippo Vascon, Eleonora Gianquinto, Laura Bertarini, Jean-Denis Docquier

Pharmaceuticals (Basel)· December 2023

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Nucleoside Derivatives of 2,6-Diaminopurine Antivirals: Base-Modified Nucleosides with Broad-Spectrum Antimicrobial Properties.
Maria Grazia Martina, Federica Giammarino, Ilaria Vicenti, Elisabetta Groaz, Jef Rozenski, Jean Denis Docquier

ChemMedChem· August 2023

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Zidovudine-β-Lactam Pronucleoside Strategy for Selective Delivery into Gram-Negative Bacteria Triggered by β-Lactamases.
Miyanou Rosales-Hurtado, Filomena Sannio, Lindita Lari, Federica Verdirosa, Georges Feller, Jean-Denis Docquier

ACS Infect Dis· August 2023

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The impact of counterions in biological activity: case study of antibacterial alkylguanidino ureas.
Claudia Ardino, Filomena Sannio, Carolina Pasero, Lorenzo Botta, Elena Dreassi, Jean-Denis Docquier

Mol Divers· June 2023

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Discovering NDM-1 inhibitors using molecular substructure embeddings representations.
Thomas Papastergiou, Jérôme Azé, Sandra Bringay, Maxime Louet, Pascal Poncelet, Jean-Denis Docquier

J Integr Bioinform· June 2023

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Discovery and Optimization of a Novel Macrocyclic Amidinourea Series Active as Acidic Mammalian Chitinase Inhibitors.
Lorenzo Jacopo Ilic Balestri, Claudia Immacolata Trivisani, Francesco Orofino, Diego Fiorucci, Giuseppina Ivana Truglio, Jean-Denis Docquier

ACS Med Chem Lett· April 2023

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Peptaibol Analogs Show Potent Antibacterial Activity against Multidrug Resistant Opportunistic Pathogens.
Chiara Dalla Torre, Filomena Sannio, Mattia Battistella, Jean-Denis Docquier, Marta De Zotti

Int J Mol Sci· April 2023

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Chemical Optimization of Selective LasB Elastase Inhibitors and Their Impact on LasB-Mediated Activation of IL-1β in Cellular and Animal Infection Models.
Martin J Everett, David T Davies, Simon Leiris, Nicolas Sprynski, Agustina Llanos, Jean-Denis Docquier

ACS Infect Dis· February 2023

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Lunaemycins, New Cyclic Hexapeptide Antibiotics from the Cave Moonmilk-Dweller MM109.
Loïc Martinet, Aymeric Naômé, Lucas C D Rezende, Déborah Tellatin, Bernard Pignon, Jean-Denis Docquier

Int J Mol Sci· January 2023

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A Clinical Study Provides the First Direct Evidence That Interindividual Variations in Fecal β-Lactamase Activity Affect the Gut Mycobiota Dynamics in Response to β-Lactam Antibiotics.
Margot Delavy, Charles Burdet, Natacha Sertour, Savannah Devente, Jean-Denis Docquier

mBio· December 2022

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Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum Metallo-β-lactamase Inhibitors Showing Potent Synergistic Activity on VIM- and NDM-1-Producing Clinical Isolates.
Alice Legru, Federica Verdirosa, Yen Vo-Hoang, Giusy Tassone, Filippo Vascon, Jean-Denis Docquier

J Med Chem· December 2022

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Optimization of Pyrazole Compounds as Antibiotic Adjuvants Active against Colistin- and Carbapenem-Resistant .
Filomena Sannio, Antonella Brizzi, Rosita Del Prete, Marialuce Avigliano, Tiziana Simone, Jean-Denis Docquier

Antibiotics (Basel)· December 2022

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A fragment-based drug discovery strategy applied to the identification of NDM-1 β-lactamase inhibitors.
Jérémy Caburet, Benjamin Boucherle, Sofiane Bourdillon, Giorgia Simoncelli, Federica Verdirosa, Jean-Denis Docquier

Eur J Med Chem· October 2022

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1,2,4-Triazole-3-thione analogues with an arylakyl group at position 4 as metallo-β-lactamase inhibitors.
Laurent Gavara, Federica Verdirosa, Laurent Sevaille, Alice Legru, Giuseppina Corsica, Jean-Denis Docquier

Bioorg Med Chem· October 2022

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Towards Innovative Antibacterial Correctors for Cystic Fibrosis Targeting the Lung Microbiome with a Multifunctional Effect.
Maria Grazia Martina, Filomena Sannio, Emmanuele Crespan, Marialaura Pavone, Alice Simoncini, Jean-Denis Docquier

ChemMedChem· September 2022

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Editorial: Structural and Biochemical Aspects of the Interaction of β-Lactamases With State-of-the-Art Inhibitors.
Krisztina M Papp-Wallace, Jean-Denis Docquier, Frederic Kerff, Pablo Power

Front Microbiol· February 2022

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