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Publications by authors named "Kenji Matsuki"

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8-(3-chloro-4-methoxybenzyl)-8H-pyrido[2,3-d]pyrimidin-7-one derivatives as potent and selective phosphodiesterase 5 inhibitors.
Toshiaki Sakamoto, Yuichi Koga, Masataka Hikota, Kenji Matsuki, Hideki Mochida

Bioorg Med Chem Lett· April 2015


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The discovery of avanafil for the treatment of erectile dysfunction: a novel pyrimidine-5-carboxamide derivative as a potent and highly selective phosphodiesterase 5 inhibitor.
Toshiaki Sakamoto, Yuichi Koga, Masataka Hikota, Kenji Matsuki, Michino Murakami

Bioorg Med Chem Lett· December 2014


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Design and synthesis of novel 5-(3,4,5-trimethoxybenzoyl)-4-aminopyrimidine derivatives as potent and selective phosphodiesterase 5 inhibitors: scaffold hopping using a pseudo-ring by intramolecular hydrogen bond formation.
Toshiaki Sakamoto, Yuichi Koga, Masataka Hikota, Kenji Matsuki, Michino Murakami

Bioorg Med Chem Lett· November 2014


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