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Publications by authors named "Kentaro Umei"

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Discovery of novel pyrazolo[1,5-a]pyridine-based EP receptor antagonists by scaffold hopping: Design, synthesis, and structure-activity relationships.
Yosuke Nishigaya, Kentaro Umei, Yoshifumi Saito, Hiroyuki Watanabe, Tatsuhiro Kondo

Bioorg Med Chem Lett· September 2017


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Identification of novel 1,2,3,6-tetrahydropyridyl-substituted benzo[d]thiazoles: Lead generation and optimization toward potent and orally active EP receptor antagonists.
Kentaro Umei, Yosuke Nishigaya, Kazuya Tatani, Yasushi Kohno, Nobuyuki Tanaka

Bioorg Med Chem· July 2017


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Novel pyrazolo[1,5-a]pyridines as orally active EP receptor antagonists: Synthesis, structure-activity relationship studies, and biological evaluation.
Kentaro Umei, Yosuke Nishigaya, Atsushi Kondo, Kazuya Tatani, Nobuyuki Tanaka

Bioorg Med Chem· May 2017


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Synthesis of Paclitaxel. 1. Synthesis of the ABC Ring of Paclitaxel by SmI2-Mediated Cyclization.
Keisuke Fukaya, Yuta Tanaka, Ayako C Sato, Keisuke Kodama, Hirohisa Yamazaki, Kentaro Umei

Org Lett· June 2015


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