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Publications by authors named "Koen Buysse"

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Azepinone-Containing Tetrapeptide Analogues of Melanotropin Lead to Selective hMC4R Agonists and hMC5R Antagonist.
Olivier Van der Poorten, Krisztina Fehér, Koen Buysse, Debby Feytens, Ioanna Zoi

ACS Med Chem Lett· February 2015


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Amino triazolo diazepines (Ata) as constrained histidine mimics.
Koen Buysse, Julien Farard, Alexandros Nikolaou, Patrick Vanderheyden, Georges Vauquelin

Org Lett· December 2011


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Design of novel neurokinin 1 receptor antagonists based on conformationally constrained aromatic amino acids and discovery of a potent chimeric opioid agonist-neurokinin 1 receptor antagonist.
Steven Ballet, Debby Feytens, Koen Buysse, Nga N Chung, Carole Lemieux

J Med Chem· April 2011


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