Publications by authors named "Luca Pinzi"

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Design, synthesis and biological activity of glycoconjugated ADAMTS5 exosite inhibitors: applications in osteoarthritis and ovarian cancer models.
Doretta Cuffaro, Sophie Blagg, Kazuhiro Yamamoto, Luca Pinzi, Rachele Bacchetti

Sci Rep· December 2025

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Design, synthesis, and biological evaluation of chalcone derivatives as selective Monoamine Oxidase-B inhibitors with potential neuroprotective effects.
Giorgio Facchetti, Sara Marchese, Valentina Coccè, Luisa Doneda, Giulio Alessandri, Luca Pinzi

Eur J Med Chem· November 2025

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Improving Machine Learning Classification Predictions through SHAP and Features Analysis Interpretation.
Leonardo Bernal, Giulio Rastelli, Luca Pinzi

J Chem Inf Model· November 2025

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Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer.
Andrea Citarella, Silvia Belluti, Davide Bonanni, Davide Moi, Isabella Piccinini, Luca Pinzi

J Med Chem· August 2025

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Selective imaging probes for differential detection of pathological tau polymorphs in tauopathies.
Nicolò Bisi, Luca Pinzi, Giulio Rastelli

Drug Discov Today· May 2025

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Exploring Biological Targets of Magnolol and Honokiol and their Nature-Inspired Synthetic Derivatives: In Silico Identification and Experimental Validation of Estrogen Receptors.
Annachiara Tinivella, Jerome C Nwachukwu, Luca Pinzi, Maria Antonietta Dettori, Davide Fabbri

J Nat Prod· November 2024

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Searching for Novel HDAC6/Hsp90 Dual Inhibitors with Anti-Prostate Cancer Activity: In Silico Screening and In Vitro Evaluation.
Luca Pinzi, Silvia Belluti, Isabella Piccinini, Carol Imbriano, Giulio Rastelli

Pharmaceuticals (Basel)· August 2024

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Early Diagnosis of Neurodegenerative Diseases: What Has Been Undertaken to Promote the Transition from PET to Fluorescence Tracers.
Nicolò Bisi, Luca Pinzi, Giulio Rastelli, Nicolò Tonali

Molecules· February 2024

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Quantitative live cell imaging of a tauopathy model enables the identification of a polypharmacological drug candidate that restores physiological microtubule interaction.
Luca Pinzi, Christian Conze, Nicolo Bisi, Gabriele Dalla Torre, Ahmed Soliman

Nat Commun· February 2024

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Structure-activity exploration of a small-molecule allosteric inhibitor of T790M/L858R double mutant EGFR.
Francesca Foschi, Annachiara Tinivella, Valentina Crippa, Luca Pinzi, Luca Mologni

J Enzyme Inhib Med Chem· December 2023

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Discovery of a Potent Dual Inhibitor of Aromatase and Aldosterone Synthase.
Annachiara Tinivella, Marta Banchi, Guido Gambacorta, Federica Borghi, Paola Orlandi, Luca Pinzi

ACS Pharmacol Transl Sci· December 2023

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Discovery of potent pyrrolo-pyrimidine and purine HDAC inhibitors for the treatment of advanced prostate cancer.
Davide Moi, Davide Bonanni, Silvia Belluti, Pasquale Linciano, Andrea Citarella, Luca Pinzi

Eur J Med Chem· November 2023

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Trends and Applications in Computationally Driven Drug Repurposing.
Luca Pinzi, Giulio Rastelli

Int J Mol Sci· November 2023

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Insights into the Structural Conformations of the Tau Protein in Different Aggregation Status.
Luca Pinzi, Nicolò Bisi, Claudia Sorbi, Silvia Franchini, Nicolò Tonali

Molecules· June 2023

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Identification of Promising Drug Candidates against Prostate Cancer through Computationally-Driven Drug Repurposing.
Leonardo Bernal, Luca Pinzi, Giulio Rastelli

Int J Mol Sci· February 2023

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Design, synthesis, biological evaluation and crystal structure determination of dual modulators of carbonic anhydrases and estrogen receptors.
Annachiara Tinivella, Jerome C Nwachukwu, Andrea Angeli, Francesca Foschi, Anna Laura Benatti, Luca Pinzi

Eur J Med Chem· January 2023

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Development of machine learning classifiers to predict compound activity on prostate cancer cell lines.
Davide Bonanni, Luca Pinzi, Giulio Rastelli

J Cheminform· November 2022

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Dual Targeting Strategies on Histone Deacetylase 6 (HDAC6) and Heat Shock Protein 90 (Hsp90).
Davide Bonanni, Andrea Citarella, Davide Moi, Luca Pinzi, Elisa Bergamini

Curr Med Chem· May 2022

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On the development of B-Raf inhibitors acting through innovative mechanisms.
Luca Pinzi

F1000Res· May 2022

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Synthesis of potent and selective HDAC6 inhibitors led to unexpected opening of a quinazoline ring.
Davide Moi, Andrea Citarella, Davide Bonanni, Luca Pinzi, Daniele Passarella

RSC Adv· April 2022

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Identification of potential biological targets of oxindole scaffolds via repositioning strategies.
Annachiara Tinivella, Luca Pinzi, Guido Gambacorta, Ian Baxendale, Giulio Rastelli

F1000Res· March 2022

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Inhibitors of histone deacetylase 6 based on a novel 3-hydroxy-isoxazole zinc binding group.
Pasquale Linciano, Luca Pinzi, Silvia Belluti, Ugo Chianese, Rosaria Benedetti

J Enzyme Inhib Med Chem· December 2021

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Design and Synthesis of Hsp90 Inhibitors with B-Raf and PDHK1 Multi-Target Activity.
Luca Pinzi, Francesca Foschi, Michael S Christodoulou, Daniele Passarella, Giulio Rastelli

ChemistryOpen· December 2021

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Chemoinformatics Analyses of Tau Ligands Reveal Key Molecular Requirements for the Identification of Potential Drug Candidates against Tauopathies.
Luca Pinzi, Annachiara Tinivella, Giulio Rastelli

Molecules· August 2021

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Hydroxamic Acid Derivatives: From Synthetic Strategies to Medicinal Chemistry Applications.
Andrea Citarella, Davide Moi, Luca Pinzi, Davide Bonanni, Giulio Rastelli

ACS Omega· August 2021

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