Publications by authors named "Mathieu Rappas"

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Discovery of PF-07054894, a Potent Squaramide-Based CCR6 Antagonist Displaying High CXCR2 Selectivity.
Mark E Schnute, Huixian Wu, John I Trujillo, Wei Li, David Jonathan Wasilko, Mathieu Rappas

J Med Chem· October 2025

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Conformational Role of Methyl in the Potency of Cyclohexane-Substituted Squaramide CCR6 Antagonists.
Brian S Gerstenberger, Ray Unwalla, Kathleen A Farley, Philippe Nuhant, Vincent M Lombardo, Mathieu Rappas

J Med Chem· February 2025

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Structural basis for CCR6 modulation by allosteric antagonists.
David Jonathan Wasilko, Brian S Gerstenberger, Kathleen A Farley, Wei Li, Jennifer Alley, Mathieu Rappas

Nat Commun· August 2024

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Mix-and-extrude: high-viscosity sample injection towards time-resolved protein crystallography.
Mohammad Vakili, Huijong Han, Christina Schmidt, Agnieszka Wrona, Marco Kloos, Mathieu Rappas

J Appl Crystallogr· August 2023

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Advances in long-wavelength native phasing at X-ray free-electron lasers.
Karol Nass, Robert Cheng, Laura Vera, Aldo Mozzanica, Sophie Redford, Mathieu Rappas

IUCrJ· November 2020

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Comparison of Orexin 1 and Orexin 2 Ligand Binding Modes Using X-ray Crystallography and Computational Analysis.
Mathieu Rappas, Ammar A E Ali, Kirstie A Bennett, Jason D Brown, Sarah J Bucknell

J Med Chem· February 2020

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High-resolution crystal structure of parathyroid hormone 1 receptor in complex with a peptide agonist.
Janosch Ehrenmann, Jendrik Schöppe, Christoph Klenk, Mathieu Rappas, Lutz Kummer

Nat Struct Mol Biol· December 2018

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BRCT domains of the DNA damage checkpoint proteins TOPBP1/Rad4 display distinct specificities for phosphopeptide ligands.
Matthew Day, Mathieu Rappas, Katie Ptasinska, Dominik Boos, Antony W Oliver

Elife· October 2018

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Structure of the complement C5a receptor bound to the extra-helical antagonist NDT9513727.
Nathan Robertson, Mathieu Rappas, Andrew S Doré, Jason Brown, Giovanni Bottegoni

Nature· January 2018

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Corrigendum: Crystal structure of the GLP-1 receptor bound to a peptide agonist.
Ali Jazayeri, Mathieu Rappas, Alastair J H Brown, James Kean, James C Errey

Nature· August 2017

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Crystal structure of the GLP-1 receptor bound to a peptide agonist.
Ali Jazayeri, Mathieu Rappas, Alastair J H Brown, James Kean, James C Errey

Nature· June 2017

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Structural insight into allosteric modulation of protease-activated receptor 2.
Robert K Y Cheng, Cédric Fiez-Vandal, Oliver Schlenker, Karl Edman, Birte Aggeler, Mathieu Rappas

Nature· May 2017

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Intracellular allosteric antagonism of the CCR9 receptor.
Christine Oswald, Mathieu Rappas, James Kean, Andrew S Doré, James C Errey

Nature· December 2016

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Phosphorylation-dependent assembly and coordination of the DNA damage checkpoint apparatus by Rad4(TopBP1).
Meng Qu, Mathieu Rappas, Christopher P Wardlaw, Valerie Garcia, Jing-Yi Ren

Mol Cell· September 2013

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Regulation of DNA replication through Sld3-Dpb11 interaction is conserved from yeast to humans.
Dominik Boos, Luis Sanchez-Pulido, Mathieu Rappas, Laurence H Pearl, Antony W Oliver

Curr Biol· July 2011

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Structure and function of the Rad9-binding region of the DNA-damage checkpoint adaptor TopBP1.
Mathieu Rappas, Antony W Oliver, Laurence H Pearl

Nucleic Acids Res· January 2011

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Coupling sigma factor conformation to RNA polymerase reorganisation for DNA melting.
Patricia C Burrows, Nicolas Joly, Wendy V Cannon, Beatriz P Cámara, Mathieu Rappas

J Mol Biol· March 2009

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Organization of an activator-bound RNA polymerase holoenzyme.
Daniel Bose, Tillmann Pape, Patricia C Burrows, Mathieu Rappas, Siva R Wigneshweraraj

Mol Cell· November 2008

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Mechanism of homotropic control to coordinate hydrolysis in a hexameric AAA+ ring ATPase.
Jörg Schumacher, Nicolas Joly, Inaki Leoz Claeys-Bouuaert, Shaniza Abdul Aziz, Mathieu Rappas

J Mol Biol· August 2008

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Visualizing the organization and reorganization of transcription complexes for gene expression.
Patricia C Burrows, Sivaramesh Wigneshweraraj, Dan Bose, Nicolas Joly, Jörg Schumacher, Mathieu Rappas

Biochem Soc Trans· August 2008

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Modus operandi of the bacterial RNA polymerase containing the sigma54 promoter-specificity factor.
Sivaramesh Wigneshweraraj, Daniel Bose, Patricia C Burrows, Nicolas Joly, Jörg Schumacher, Mathieu Rappas

Mol Microbiol· May 2008

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Trapping of a transcription complex using a new nucleotide analogue: AMP aluminium fluoride.
Nicolas Joly, Mathieu Rappas, Martin Buck, Xiaodong Zhang

J Mol Biol· February 2008

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Dissecting the ATP hydrolysis pathway of bacterial enhancer-binding proteins.
Daniel Bose, Nicolas Joly, Tillmann Pape, Mathieu Rappas, Jorg Schumacher

Biochem Soc Trans· February 2008

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Coupling nucleotide hydrolysis to transcription activation performance in a bacterial enhancer binding protein.
Nicolas Joly, Mathieu Rappas, Siva R Wigneshweraraj, Xiaodong Zhang, Martin Buck

Mol Microbiol· November 2007

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Sensor I threonine of the AAA+ ATPase transcriptional activator PspF is involved in coupling nucleotide triphosphate hydrolysis to the restructuring of sigma 54-RNA polymerase.
Jörg Schumacher, Nicolas Joly, Mathieu Rappas, Dominic Bradley, Siva R Wigneshweraraj

J Biol Chem· March 2007

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