Publications by authors named "Pierre Falson"

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Assembly of Detergents with Highly Branched Dicarboxylate Clamps for Membrane Protein Studies.
Kim-Anh Nguyen, Pierre Falson, Ahcène Boumendjel

ChemistryOpen· September 2025

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X-ray diffraction images for two membrane protein crystals presenting high anisotropy; the ABC transporter BmrA and the NADPH oxidase.
Veronica Zampieri, Annelise Vermot, Michel Thepaut, Isabelle Petit-Hartlein, Franck Fieschi, Pierre Falson

IUCrdata· July 2025

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Ligand-Based Drug Discovery Leveraging State-of-the-Art Machine Learning Methodologies Exemplified by Cdr1 Inhibitor Prediction.
The-Chuong Trinh, Pierre Falson, Viet-Khoa Tran-Nguyen, Ahcène Boumendjel

J Chem Inf Model· April 2025

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Purification and characterization of Cdr1, the drug-efflux pump conferring azole resistance in Candida species.
Jorgaq Pata, Alexis Moreno, Benjamin Wiseman, Sandrine Magnard, Idriss Lehlali, Pierre Falson

Biochimie· May 2024

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The Hydrophilic C-terminus of Yeast Plasma-membrane Na/H Antiporters Impacts Their Ability to Transport K.
Olga Zimmermannová, Diego Velázquez, Klára Papoušková, Vojtěch Průša, Viktorie Radová, Pierre Falson

J Mol Biol· February 2024

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The transport activity of the multidrug ABC transporter BmrA does not require a wide separation of the nucleotide-binding domains.
Margot Di Cesare, Elise Kaplan, Julia Rendon, Guillaume Gerbaud, Sepideh Valimehr, Pierre Falson

J Biol Chem· January 2024

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Structure, function, and inhibition of catalytically asymmetric ABC transporters: Lessons from the PDR subfamily.
Atanu Banerjee, Jorgaq Pata, Vincent Chaptal, Ahcène Boumendjel, Pierre Falson

Drug Resist Updat· November 2023

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Drug candidates targeting multidrug resistance in cancer and infections.
Marc Le Borgne, Pierre Falson, Ahcène Boumendjel

Eur J Med Chem· March 2023

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The non-Newtonian behavior of detergents during concentration is increased by macromolecules, in trans, and results in their over-concentration.
Alexia Gobet, Veronica Zampieri, Sandrine Magnard, Eva Pebay-Peyroula, Pierre Falson

Biochimie· February 2023

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Inhibitors of ABCG2-mediated multidrug resistance: Lead generation through computer-aided drug design.
Laura Goracci, Alessandra Nurisso, Emile Roussel, Basile Pérès, Vincent Chaptal, Pierre Falson

Eur J Med Chem· February 2023

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Specific Xray diffraction patterns of membrane proteins caused by secondary structure collinearity.
Juliette Martin, Xavier Robert, Patrice Gouet, Pierre Falson, Vincent Chaptal

Biochim Biophys Acta Biomembr· January 2023

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The first ADC bearing the ferroptosis inducer RSL3 as a payload with conservation of the fragile electrophilic warhead.
Kim-Anh Nguyen, Louise Conilh, Pierre Falson, Charles Dumontet, Ahcène Boumendjel

Eur J Med Chem· December 2022

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Overexpression of the ABC Transporter BmrA Within Intracellular Caveolae in Escherichia coli.
Alexia Gobet, Christine Jaxel, Sandrine Magnard, Manuel Garrigos, Stéphane Orlowski, Pierre Falson

Methods Mol Biol· July 2022

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Production and Purification of a GFP-Tagged ABC Transporter CaCdr1p.
Jorgaq Pata, Alexis Moreno, Sandrine Magnard, Atanu Banerjee, Rajendra Prasad, Pierre Falson

Methods Mol Biol· July 2022

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Spontaneous Suppressors against Debilitating Transmembrane Mutants of Mdr1 Disclose Novel Interdomain Communication via Signature Motifs of the Major Facilitator Superfamily.
Suman Sharma, Atanu Banerjee, Alexis Moreno, Archana Kumari Redhu, Pierre Falson

J Fungi (Basel)· May 2022

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Substrate-bound and substrate-free outward-facing structures of a multidrug ABC exporter.
Vincent Chaptal, Veronica Zampieri, Benjamin Wiseman, Cédric Orelle, Juliette Martin, Pierre Falson

Sci Adv· January 2022

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CryoEM reconstructions of membrane proteins solved in several amphipathic solvents, nanodisc, amphipol and detergents, yield amphipathic belts of similar sizes corresponding to a common ordered solvent layer.
Veronica Zampieri, Alexia Gobet, Xavier Robert, Pierre Falson, Vincent Chaptal

Biochim Biophys Acta Biomembr· November 2021

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The Det.Belt Server: A Tool to Visualize and Estimate Amphipathic Solvent Belts around Membrane Proteins.
Veronica Zampieri, Cécile Hilpert, Mélanie Garnier, Yannick Gestin, Sébastien Delolme, Pierre Falson

Membranes (Basel)· June 2021

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ABCG: a new fold of ABC exporters and a whole new bag of riddles!
Atanu Banerjee, Alexis Moreno, Jorgaq Pata, Pierre Falson, Rajendra Prasad

Adv Protein Chem Struct Biol· April 2021

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Uncompetitive nanomolar dimeric indenoindole inhibitors of the human breast cancer resistance pump ABCG2.
Nathalie Guragossian, Billel Belhani, Alexis Moreno, Magda Teixeira Nunes, Lucia Gonzalez-Lobato, Pierre Falson

Eur J Med Chem· February 2021

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Directed Mutational Strategies Reveal Drug Binding and Transport by the MDR Transporters of .
Atanu Banerjee, Jorgaq Pata, Suman Sharma, Brian C Monk, Pierre Falson

J Fungi (Basel)· January 2021

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Chromones bearing amino acid residues: Easily accessible and potent inhibitors of the breast cancer resistance protein ABCG2.
Emile Roussel, Alexis Moréno, Nicolas Altounian, Christian Philouze, Basile Pérès, Pierre Falson

Eur J Med Chem· September 2020

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Molecular analysis of the massive GSH transport mechanism mediated by the human Multidrug Resistant Protein 1/ABCC1.
Rachad Nasr, Doriane Lorendeau, Ruttiros Khonkarn, Lauriane Dury, Basile Pérès, Pierre Falson

Sci Rep· May 2020

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Cdr1p highlights the role of the non-hydrolytic ATP-binding site in driving drug translocation in asymmetric ABC pumps.
Atanu Banerjee, Alexis Moreno, Mohammad Firoz Khan, Remya Nair, Suman Sharma, Pierre Falson

Biochim Biophys Acta Biomembr· February 2020

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Synthesis and Anticancer Cytotoxicity of Azaaurones Overcoming Multidrug Resistance.
Szilárd Tóth, Áron Szepesi, Viet-Khoa Tran-Nguyen, Balázs Sarkadi, Katalin Német, Pierre Falson

Molecules· February 2020

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