Publications by authors named "Raphael Labruere"

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Synthesis and In Vitro Pharmacological Evaluation of 5,8-Dideaza Analogs of Methotrexate.
Marta Abellán-Flos, Charles Skarbek, Dáire J Gibbons, Estelle Rascol, Ainhoa García

Molecules· June 2025

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Re-designing environmentally persistent pharmaceutical pollutant through programmed inactivation: The case of methotrexate.
Anaïs Espinosa, Estelle Rascol, Marta Abellán Flos, Charles Skarbek, Pascale Lieben

Chemosphere· November 2022

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Photodegradation of methotrexate in aqueous solution: degradation kinetics and identification of transformation products.
Anaïs Espinosa, Sylvie Nélieu, Pascale Lieben, Charles Skarbek, Raphaël Labruère

Environ Sci Pollut Res Int· January 2022

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In-Cell Generation of Anticancer Phenanthridine Through Bioorthogonal Cyclization in Antitumor Prodrug Development.
Hichem Maslah, Charles Skarbek, Catherine Gourson, Marie-Aude Plamont, Stéphanie Pethe

Angew Chem Int Ed Engl· November 2021

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Boronic acid/boronate prodrugs for cancer treatment: current status and perspectives.
Hichem Maslah, Stéphanie Pethe, Raphaël Labruère

Future Med Chem· May 2021

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Anticancer boron-containing prodrugs responsive to oxidative stress from the tumor microenvironment.
Hichem Maslah, Charles Skarbek, Stéphanie Pethe, Raphaël Labruère

Eur J Med Chem· December 2020

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Arylboronate prodrugs of doxorubicin as promising chemotherapy for pancreatic cancer.
Charles Skarbek, Silvia Serra, Hichem Maslah, Estelle Rascol, Raphaël Labruère

Bioorg Chem· October 2019

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Anti-Methicillin-Resistant Nanoantibiotics.
Raphaël Labruère, A J Sona, Edward Turos

Front Pharmacol· October 2019

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Spermine-NBD as fluorescent probe for studies of the polyamine transport system in Leishmania donovani.
Elodie Jagu, Sébastien Pomel, Stéphanie Pethe, Jean-Christophe Cintrat, Philippe M Loiseau

Bioorg Med Chem Lett· July 2019

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A chemically encoded timer for dual molecular delivery at tailored ranges and concentrations.
Silvia Serra, Ahmed Alouane, Thomas Le Saux, Steve Huvelle, Raphaël Plasson

Chem Commun (Camb)· June 2018

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Synthesis and antikinetoplastid evaluation of bis(benzyl)spermidine derivatives.
Elodie Jagu, Sébastien Pomel, Alba Diez-Martinez, Estelle Rascol, Stéphanie Pethe

Eur J Med Chem· April 2018

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Polyamine-based analogs and conjugates as antikinetoplastid agents.
Elodie Jagu, Sébastien Pomel, Stéphanie Pethe, Philippe M Loiseau, Raphaël Labruère

Eur J Med Chem· October 2017

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Synthesis and in vitro antikinetoplastid activity of polyamine-hydroxybenzotriazole conjugates.
Elodie Jagu, Sébastien Pomel, Alba Diez-Martinez, Florence Ramiandrasoa, R Luise Krauth-Siegel

Bioorg Med Chem· January 2017

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Self-immolative spacers: kinetic aspects, structure-property relationships, and applications.
Ahmed Alouane, Raphaël Labruère, Thomas Le Saux, Frédéric Schmidt, Ludovic Jullien

Angew Chem Int Ed Engl· June 2015

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Design, synthesis and in vitro antikinetoplastid evaluation of N-acylated putrescine, spermidine and spermine derivatives.
Elodie Jagu, Rachid Djilali, Sébastien Pomel, Florence Ramiandrasoa, Stéphanie Pethe

Bioorg Med Chem Lett· January 2015

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Disassembly kinetics of quinone-methide-based self-immolative spacers that contain aromatic nitrogen heterocycles.
Ahmed Alouane, Raphaël Labruère, Katherine J Silvestre, Thomas Le Saux, Frédéric Schmidt

Chem Asian J· May 2014

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Light activation for the versatile and accurate kinetic analysis of disassembly of self-immolative spacers.
Ahmed Alouane, Raphaël Labruère, Thomas Le Saux, Isabelle Aujard, Sylvie Dubruille

Chemistry· August 2013

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"Self-immolative" spacer for uncaging with fluorescence reporting.
Raphaël Labruère, Ahmed Alouane, Thomas Le Saux, Isabelle Aujard, Philippe Pelupessy

Angew Chem Int Ed Engl· September 2012

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Attenuating the size and molecular carrier capabilities of polyacrylate nanoparticles by a hydrophobic fluorine effect.
Raphaël Labruère, Edward Turos

Bioorg Med Chem· August 2012

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Poly(vinyl benzoate) nanoparticles for molecular delivery: Studies on their preparation and in vitro properties.
Raphaël Labruère, Renaud Sicard, Ryan Cormier, Edward Turos, Leigh West

J Control Release· December 2010

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Design, synthesis, and biological evaluation of the first podophyllotoxin analogues as potential vascular-disrupting agents.
Raphaël Labruère, Benoît Gautier, Marlène Testud, Johanne Seguin, Christine Lenoir

ChemMedChem· December 2010

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Design and effective synthesis of the first 4-aza-2,3-didehydropodophyllotoxin rigid aminologue: a N-methyl-4-[(3,4,5-trimethoxyphenyl)amino)]-1,2-dihydroquinoline-lactone.
Raphaël Labruère, Philippe Helissey, Stéphanie Desbène-Finck, Sylviane Giorgi-Renault

J Org Chem· May 2008

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