Publications by authors named "Regis Millet"

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Characterization of the Active Enantiomer and Mapping of the Stereospecific Intermolecular Pattern of a Reference P2X7 Allosteric Antagonist.
Andrew McGown, Nicolas Renault, Amélie Barczyk, Jordan Nafie, Luciano Barluzzi, Régis Millet

ACS Pharmacol Transl Sci· February 2025

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4-Anilinoquinazoline Derivatives as the First Potent NOD1-RIPK2 Signaling Pathway Inhibitors at the Nanomolar Range.
Amélie Barczyk, Perrine Six, Morgane Rivoal, Claire Devos, Xavier Dezitter, Régis Millet

J Med Chem· November 2024

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Activity of pyridyl-pyrazolone derivatives against Trypanosoma cruzi.
Denise da Gama Jaen Batista, Ludmila Ferreira de Almeida Fiuza, Frédérique Klupsch, Krislayne Nunes da Costa, Marcos Meuser Batista, Régis Millet

Exp Parasitol· July 2024

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Receptor Interacting Ser/Thr-Protein Kinase 2 as a New Therapeutic Target.
Morgane Rivoal, Laurent Dubuquoy, Régis Millet, Natascha Leleu-Chavain

J Med Chem· November 2023

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Novel PD-L1-Targeted Phenyl-Pyrazolone Derivatives with Antioxidant Properties.
Romain Regnault, Frédérique Klupsch, Hassiba El-Bouazzati, Romain Magnez, Raphaël Le Biannic, Régis Millet

Molecules· April 2023

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Pyrazolones as inhibitors of immune checkpoint blocking the PD-1/PD-L1 interaction.
Raphaël Le Biannic, Romain Magnez, Frédérique Klupsch, Natascha Leleu-Chavain, Bryan Thiroux, Régis Millet

Eur J Med Chem· June 2022

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Antioxidant Properties and Aldehyde Reactivity of PD-L1 Targeted Aryl-Pyrazolone Anticancer Agents.
Natascha Leleu-Chavain, Romain Regnault, Hania Ahouari, Raphaël Le Biannic, Mostafa Kouach, Régis Millet

Molecules· May 2022

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A small-molecule P2RX7 activator promotes anti-tumor immune responses and sensitizes lung tumor to immunotherapy.
Laetitia Douguet, Serena Janho Dit Hreich, Jonathan Benzaquen, Laetitia Seguin, Thierry Juhel, Régis Millet

Nat Commun· January 2021

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Pyroglutamide-Based P2X7 Receptor Antagonists Targeting Inflammatory Bowel Disease.
Germain Homerin, Samir Jawhara, Xavier Dezitter, Davy Baudelet, Pierrick Dufrénoy, Régis Millet

J Med Chem· March 2020

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Benzo[d]thiazol-2(3H)-ones as new potent selective CB agonists with anti-inflammatory properties.
Natascha Leleu-Chavain, Davy Baudelet, Valéria Moas Heloire, Diana Escalante Rocha, Nicolas Renault, Régis Millet

Eur J Med Chem· March 2019

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Synthesis and biological evaluation of ferrocene-based cannabinoid receptor 2 ligands.
Supojjanee Sansook, Wei Tuo, Mélanie Bollier, Amélie Barczyk, Xavier Dezitter, Régis Millet

Future Med Chem· March 2018

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Development of novel oxazolo[5,4-d]pyrimidines as competitive CB neutral antagonists based on scaffold hopping.
Wei Tuo, Mélanie Bollier, Natascha Leleu-Chavain, Lucas Lemaire, Amélie Barczyk, Régis Millet

Eur J Med Chem· February 2018

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One- or Two-Step Synthesis of C-8 and N-9 Substituted Purines.
Mélanie Bollier, Frédérique Klupsch, Perrine Six, Laurent Dubuquoy, Nathalie Azaroual, Régis Millet

J Org Chem· January 2018

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Small scale separation of isoxazole structurally related analogues by chiral supercritical fluid chromatography.
Yasmine Zehani, Lucas Lemaire, Regis Millet, Emmanuelle Lipka

J Chromatogr A· July 2017

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Therapeutic Potential of Fatty Acid Amide Hydrolase, Monoacylglycerol Lipase, and N-Acylethanolamine Acid Amidase Inhibitors.
Wei Tuo, Natascha Leleu-Chavain, John Spencer, Supojjanee Sansook, Régis Millet

J Med Chem· January 2017

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Exploring chiral separation of 3-carboxamido-5-aryl isoxazole derivatives by supercritical fluid chromatography on amylose and cellulose tris dimethyl- and chloromethyl phenylcarbamate polysaccharide based stationary phases.
Yasmine Zehani, Lucas Lemaire, Alina Ghinet, Régis Millet, Philippe Chavatte

J Chromatogr A· October 2016

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Corrigendum to "Evaluation and comparison of three different separation techniques for analysis of retroamide enantiomers and their biological evaluation against h-P2X7 receptor" [J. Chromatogr. B 986-987 (2015) 35-43].
Davy Baudelet, Christophe Furman, Alina Ghinet, Xavier Dezitter, Sahil Adriouch, Régis Millet

J Chromatogr B Analyt Technol Biomed Life Sci· July 2016

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Design, synthesis and biological evaluation of potent FAAH inhibitors.
Wei Tuo, Natascha Leleu-Chavain, Amélie Barczyk, Nicolas Renault, Lucas Lemaire, Régis Millet

Bioorg Med Chem Lett· June 2016

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Involvement of the P2X7 purinergic receptor in inflammation: an update of antagonists series since 2009 and their promising therapeutic potential.
Davy Baudelet, Emmanuelle Lipka, Régis Millet, Alina Ghinet

Curr Med Chem· September 2015

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Evaluation and comparison of three different separation techniques for analysis of retroamide enantiomers and their biological evaluation against h-P2X7 receptor.
Davy Baudelet, Christophe Furman, Alina Ghinet, Xavier Dezitter, Sahil Adriouch, Régis Millet

J Chromatogr B Analyt Technol Biomed Life Sci· April 2015

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Conformational Restriction Leading to a Selective CB2 Cannabinoid Receptor Agonist Orally Active Against Colitis.
Jamal El Bakali, Giulio G Muccioli, Mathilde Body-Malapel, Madjid Djouina, Frédérique Klupsch, Régis Millet

ACS Med Chem Lett· February 2015

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Antagonists of the P2X7 receptor: mechanism of enantioselective recognition using highly sulfated and sulfobutylether cyclodextrins by capillary electrokinetic chromatography.
Davy Baudelet, Alina Ghinet, Christophe Furman, Xavier Dezitter, Philippe Gautret, Régis Millet

Electrophoresis· October 2014

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Enantioseparation of pyroglutamide derivatives on polysaccharide based chiral stationary phases by high-performance liquid chromatography and supercritical fluid chromatography: a comparative study.
Davy Baudelet, Nadège Schifano-Faux, Alina Ghinet, Xavier Dezitter, Florent Barbotin, Régis Millet

J Chromatogr A· October 2014

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Switching cannabinoid response from CB(2) agonists to FAAH inhibitors.
Aurélien Tourteau, Natascha Leleu-Chavain, Mathilde Body-Malapel, Virginie Andrzejak, Amélie Barczyk, Régis Millet

Bioorg Med Chem Lett· March 2014

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Therapeutical potential of CB₂ receptors in immune-related diseases.
Natascha Leleu-Chavain, Pierre Desreumaux, Philippe Chavatte, Régis Millet

Curr Mol Pharmacol· November 2013

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