Publications by authors named "Robert Aversa"

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Discovery of Selective and Orally Bioavailable Heterobifunctional Degraders of Cyclin-Dependent Kinase 2.
Philip N Collier, Xiaozhang Zheng, Melissa Ford, Matthew Weiss, Dapeng Chen, Robert J Aversa

J Med Chem· September 2025

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CDK2 heterobifunctional degraders co-degrade CDK2 and cyclin E resulting in efficacy in CCNE1-amplified and overexpressed cancers.
Nicholas Kwiatkowski, Tong Liang, Zhe Sha, Philip N Collier, Annan Yang, Robert Aversa

Cell Chem Biol· April 2025

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Design and Discovery of -(3-(2-(2-Hydroxyethoxy)-6-morpholinopyridin-4-yl)-4-methylphenyl)-2-(trifluoromethyl)isonicotinamide, a Selective, Efficacious, and Well-Tolerated RAF Inhibitor Targeting RAS Mutant Cancers: The Path to the Clinic.
Savithri Ramurthy, Benjamin R Taft, Robert J Aversa, Paul A Barsanti, Matthew T Burger

J Med Chem· March 2020

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USP7 inhibits Wnt/β-catenin signaling through promoting stabilization of Axin.
Lei Ji, Bo Lu, Raffaella Zamponi, Olga Charlat, Robert Aversa

Nat Commun· September 2019

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Antitumor Properties of RAF709, a Highly Selective and Potent Inhibitor of RAF Kinase Dimers, in Tumors Driven by Mutant RAS or BRAF.
Wenlin Shao, Yuji M Mishina, Yun Feng, Giordano Caponigro, Vesselina G Cooke, Robert Aversa

Cancer Res· March 2018

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Design and Discovery of N-(2-Methyl-5'-morpholino-6'-((tetrahydro-2H-pyran-4-yl)oxy)-[3,3'-bipyridin]-5-yl)-3-(trifluoromethyl)benzamide (RAF709): A Potent, Selective, and Efficacious RAF Inhibitor Targeting RAS Mutant Cancers.
Gisele A Nishiguchi, Alice Rico, Huw Tanner, Robert J Aversa, Benjamin R Taft

J Med Chem· June 2017

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Structure-Based Drug Design of Novel Potent and Selective Tetrahydropyrazolo[1,5-a]pyrazines as ATR Inhibitors.
Paul A Barsanti, Robert J Aversa, Xianming Jin, Yue Pan, Yipin Lu

ACS Med Chem Lett· January 2015

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Structure-Based Drug Design of Novel, Potent, and Selective Azabenzimidazoles (ABI) as ATR Inhibitors.
Paul A Barsanti, Yue Pan, Yipin Lu, Rama Jain, Matthew Cox, Robert J Aversa

ACS Med Chem Lett· January 2015

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Maitotoxin: An Inspiration for Synthesis.
K C Nicolaou, Robert J Aversa

Isr J Chem· April 2011

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Synthesis of the C'D'E'F' domain of maitotoxin.
K C Nicolaou, Jae Hong Seo, Tsuyoshi Nakamura, Robert J Aversa

J Am Chem Soc· January 2011

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Synthesis of the ABCDEFG ring system of maitotoxin.
K C Nicolaou, Robert J Aversa, Jian Jin, Fatima Rivas

J Am Chem Soc· May 2010

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The continuing saga of the marine polyether biotoxins.
K C Nicolaou, Michael O Frederick, Robert J Aversa

Angew Chem Int Ed Engl· October 2008

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Chemical Synthesis of the GHIJKLMNO Ring System of Maitotoxin.
K C Nicolaou, Michael O Frederick, Antonio C B Burtoloso, Ross M Denton, Fatima Rivas, Robert J Aversa

J Am Chem Soc· June 2008

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Chemical synthesis of the GHIJK ring system and further experimental support for the originally assigned structure of maitotoxin.
K C Nicolaou, Kevin P Cole, Michael O Frederick, Robert J Aversa, Ross M Denton

Angew Chem Int Ed Engl· January 2008

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