Publications by authors named "Sium Habte"

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B cells from African American lupus patients exhibit an activated phenotype.
Laurence C Menard, Sium Habte, Waldemar Gonsiorek, Deborah Lee, Dana Banas

JCI Insight· June 2016

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Improving the pharmacokinetic and CYP inhibition profiles of azaxanthene-based glucocorticoid receptor modulators-identification of (S)-5-(2-(9-fluoro-2-(4-(2-hydroxypropan-2-yl)phenyl)-5H-chromeno[2,3-b]pyridin-5-yl)-2-methylpropanamido)-N-(tetrahydro-2H-pyran-4-yl)-1,3,4-thiadiazole-2-carboxamide (BMS-341).
Michael G Yang, T G Murali Dhar, Zili Xiao, Hai-Yun Xiao, James J-W Duan, Sium Habte

J Med Chem· May 2015

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Discovery of acylurea isosteres of 2-acylaminothiadiazole in the azaxanthene series of glucocorticoid receptor agonists.
Hua Gong, Michael Yang, Zili Xiao, Arthur M Doweyko, Mark Cunningham, Sium Habte

Bioorg Med Chem Lett· August 2014

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Synthesis and structure-activity relationships of novel indazolyl glucocorticoid receptor partial agonists.
John L Gilmore, James E Sheppeck, Jim Wang, T G Murali Dhar, Cullen Cavallaro, Sium F Habte

Bioorg Med Chem Lett· October 2013

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Discovery of potent and selective nonsteroidal indazolyl amide glucocorticoid receptor agonists.
James E Sheppeck, John L Gilmore, Hai-Yun Xiao, T G Murali Dhar, David Nirschl, Sium F Habte

Bioorg Med Chem Lett· October 2013

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Heterocyclic glucocorticoid receptor modulators with a 2,2-dimethyl-3-phenyl-N-(thiazol or thiadiazol-2-yl)propanamide core.
Hai-Yun Xiao, Dauh-Rurng Wu, James E Sheppeck, Sium F Habte, Mark D Cunningham

Bioorg Med Chem Lett· October 2013

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Azaxanthene based selective glucocorticoid receptor modulators: design, synthesis, and pharmacological evaluation of (S)-4-(5-(1-((1,3,4-thiadiazol-2-yl)amino)-2-methyl-1-oxopropan-2-yl)-5H-chromeno[2,3-b]pyridin-2-yl)-2-fluoro-N,N-dimethylbenzamide (BMS-776532) and its methylene homologue (BMS-791826).
David S Weinstein, Hua Gong, Arthur M Doweyko, Mark Cunningham, Sium Habte

J Med Chem· October 2011

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Dimethyl-diphenyl-propanamide derivatives as nonsteroidal dissociated glucocorticoid receptor agonists.
Bingwei V Yang, David S Weinstein, Lidia M Doweyko, Hua Gong, Wayne Vaccaro, Sium Habte

J Med Chem· December 2010

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Novel synthesis of the hexahydroimidazo[1,5b]isoquinoline scaffold: application to the synthesis of glucocorticoid receptor modulators.
Hai-Yun Xiao, Dauh-Rurng Wu, Mary F Malley, Jack Z Gougoutas, Sium F Habte

J Med Chem· February 2010

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Discovery of novel dihydro-9,10-ethano-anthracene carboxamides as glucocorticoid receptor modulators.
Bingwei V Yang, Wayne Vaccaro, Arthur M Doweyko, Lidia M Doweyko, Tram Huynh, Sium Habte

Bioorg Med Chem Lett· April 2009

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