Publications by authors named "Stefano Tomassi"

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β-Cyclodextrin Inclusion Complexes with Model Pentapeptides: Role of the Tyrosine Position within the Peptide Chain.
Martina Dragone, Gianluca D'Abrosca, Antonia D'Aniello, Domenico Alberga, Getasew Shitaye, Stefano Tomassi

ChemistryOpen· October 2025

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Switching Roles─Exploring Concentration-Dependent Agonistic versus Antagonistic Behavior of Integrin Ligands.
Beatrice Stefanie Ludwig, Nils Krautkremer, Stefano Tomassi, Salvatore Di Maro, Francesco Saverio Di Leva

J Med Chem· February 2025

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Discovery of -substituted-2-oxoindolin benzoylhydrazines as c-MET/SMO modulators in EGFRi-resistant non-small cell lung cancer.
Stefano Tomassi, Benito Natale, Michele Roggia, Luisa Amato, Caterina De Rosa

RSC Med Chem· January 2025

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Comprehensive structural investigation of a potent and selective CXCR4 antagonist via crosslink modification.
Anna Maria Trotta, Vincenzo Mazzarella, Michele Roggia, Antonia D'Aniello, Alessandra Del Bene, Stefano Tomassi

Eur J Med Chem· December 2024

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Disulfide bond replacement with non-reducible side chain to tail macrolactamization for the development of potent and selective CXCR4 peptide antagonists endowed with flanking binding sites.
Anna Maria Trotta, Stefano Tomassi, Gaetana Di Maiolo, Caterina Ieranò, Cinzia Vetrei

Eur J Med Chem· October 2024

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A combined approach of structure-based virtual screening and NMR to interrupt the PD-1/PD-L1 axis: Biphenyl-benzimidazole containing compounds as novel PD-L1 inhibitors.
Greta Donati, Monica Viviano, Vincenzo Maria D'Amore, Alessandra Cipriano, Isidora Diakogiannaki, Stefano Tomassi

Arch Pharm (Weinheim)· March 2024

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Paper-based electrochemical device for early detection of integrin αvβ6 expressing tumors.
Stefano Cinti, Stefano Tomassi, Chiara Ciardiello, Rossella Migliorino, Marinella Pirozzi

Commun Chem· March 2024

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Specific Inhibitors of Mitochondrial Deacylase Sirtuin 4 Endowed with Cellular Activity.
Martin Pannek, Zayan Alhalabi, Daniela Tomaselli, Martina Menna, Francesco Fiorentino, Stefano Tomassi

J Med Chem· February 2024

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Irreversible inhibition of TRF2 recruiting functions by a covalent cyclic peptide induces telomeric replication stress in cancer cells.
Alexander P Sobinoff, Salvatore Di Maro, Ronnie R J Low, Rosaria Benedetti, Stefano Tomassi

Cell Chem Biol· December 2023

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Ultrasound-assisted Peptide Nucleic Acids synthesis (US-PNAS).
Alessandra Del Bene, Antonia D'Aniello, Stefano Tomassi, Francesco Merlino, Vincenzo Mazzarella

Ultrason Sonochem· May 2023

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First-in-Class Selective Inhibitors of the Lysine Acetyltransferase KAT8.
Francesco Fiorentino, Sara Sementilli, Martina Menna, Federica Turrisi, Stefano Tomassi

J Med Chem· May 2023

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Novel pyridine-containing histone deacetylase inhibitors strongly arrest proliferation, induce apoptosis and modulate miRNAs in cancer cells.
Elisabetta Di Bello, Veronica Sian, Giulio Bontempi, Clemens Zwergel, Rossella Fioravanti, Stefano Tomassi

Eur J Med Chem· February 2023

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Novel non-covalent LSD1 inhibitors endowed with anticancer effects in leukemia and solid tumor cellular models.
Martina Menna, Francesco Fiorentino, Biagina Marrocco, Alessia Lucidi, Stefano Tomassi

Eur J Med Chem· July 2022

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Tailoring the Structure of Cell Penetrating DNA and RNA Binding Nucleopeptides.
Stefano Tomassi, Caterina Ieranò, Alessandra Del Bene, Antonia D'Aniello, Maria Napolitano

Int J Mol Sci· July 2022

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Design and synthesis of Nrf2-derived hydrocarbon stapled peptides for the disruption of protein-DNA-interactions.
Bianca Wiedemann, Dominic Kamps, Laura Depta, Jörn Weisner, Jana Cvetreznik, Stefano Tomassi

PLoS One· June 2022

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CLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists.
Stefano Tomassi, Marilisa Pia Dimmito, Minying Cai, Antonia D'Aniello, Alessandra Del Bene

J Med Chem· March 2022

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A novel smaller β-defensin-derived peptide is active against multidrug-resistant bacterial strains.
Roberta Colicchio, Ersilia Nigro, Irene Colavita, Chiara Pagliuca, Salvatore Di Maro, Stefano Tomassi

FASEB J· December 2021

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Polycomb Repressive Complex 2 Modulation through the Development of EZH2-EED Interaction Inhibitors and EED Binders.
Stefano Tomassi, Annalisa Romanelli, Clemens Zwergel, Sergio Valente, Antonello Mai

J Med Chem· August 2021

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Halting the Spread of Herpes Simplex Virus-1: The Discovery of an Effective Dual αvβ6/αvβ8 Integrin Ligand.
Stefano Tomassi, Vincenzo Maria D'Amore, Francesco Saverio Di Leva, Andrea Vannini, Giacomo Quilici

J Med Chem· May 2021

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The organometallic ferrocene exhibits amplified anti-tumor activity by targeted delivery via highly selective ligands to αvβ3, αvβ6, or α5β1 integrins.
Beatrice Stefanie Ludwig, Stefano Tomassi, Salvatore Di Maro, Francesco Saverio Di Leva, Anke Benge

Biomaterials· April 2021

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Novel Peptide-Based PET Probe for Non-invasive Imaging of C-X-C Chemokine Receptor Type 4 (CXCR4) in Tumors.
Anna Maria Trotta, Michela Aurilio, Crescenzo D'Alterio, Caterina Ieranò, Daria Di Martino, Stefano Tomassi

J Med Chem· March 2021

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Characterization of water-soluble esters of nitrobenzoxadiazole-based GSTP1-1 inhibitors for cancer treatment.
Veronica Di Paolo, Chiara Fulci, Dante Rotili, Anastasia De Luca, Stefano Tomassi

Biochem Pharmacol· August 2020

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Disulfide Bond Replacement with 1,4- and 1,5-Disubstituted [1,2,3]-Triazole on C-X-C Chemokine Receptor Type 4 (CXCR4) Peptide Ligands: Small Changes that Make Big Differences.
Stefano Tomassi, Anna Maria Trotta, Caterina Ieranò, Francesco Merlino, Anna Messere

Chemistry· August 2020

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Properly Substituted Cyclic Bis-(2-bromobenzylidene) Compounds Behaved as Dual p300/CARM1 Inhibitors and Induced Apoptosis in Cancer Cells.
Rossella Fioravanti, Stefano Tomassi, Elisabetta Di Bello, Annalisa Romanelli, Andrea Maria Plateroti

Molecules· July 2020

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HOPPI-NMR: Hot-Peptide-Based Screening Assay for Inhibitors of Protein-Protein Interactions by NMR.
Diego Brancaccio, Salvatore Di Maro, Linda Cerofolini, Stefano Giuntini, Marco Fragai, Stefano Tomassi

ACS Med Chem Lett· May 2020

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