Publications by authors named "Thierry Besson"

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Quinazoline-Derivatives of Imino-1,2,3-Dithiazoles Promote Biofilm Dispersion of .
Mathieu Gonzalez, Anne-Sophie Tareau, Daphnée de Crozals, Corentin Layec, Nathan Broudic, Thierry Besson

Pharmaceuticals (Basel)· November 2025

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DYRK1A inhibition results in MYC and ERK activation rendering KMT2A-R acute lymphoblastic leukemia cells sensitive to BCL2 inhibition.
V S S Abhinav Ayyadevara, Gerald Wertheim, Shikha Gaur, John A Chukinas, Joseph P Loftus, Thierry Besson

Leukemia· May 2025

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Novel Thiazole-Fused [4,5-] or [5,4-]Quinazolin-8-ones and Their Quinazoline Analogues: Synthesis and Biological Evaluation.
Nathan Broudic, Alexandra Pacheco-Benichou, Cécile Corbière, Blandine Baratte, Thomas Robert, Thierry Besson

Pharmaceuticals (Basel)· October 2024

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Efficacy of DYRK1A inhibitors in novel models of Down syndrome acute lymphoblastic leukemia.
Shannon L Carey-Smith, Maryam H Simad, Kunjal Panchal, Carlos Aya-Bonilla, Hannah Smolders, Thierry Besson

Haematologica· July 2024

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Design, synthesis and preliminary biological evaluation of rivastigmine-INDY hybrids as multitarget ligands against Alzheimer's disease by targeting butyrylcholinesterase and DYRK1A/CLK1 kinases.
Mihaela-Liliana Ţînţaş, Ludovic Peauger, Anaïs Barré, Cyril Papamicaël, Thierry Besson

RSC Med Chem· March 2024

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Synthesis of 2-Cyanobenzothiazoles via Pd-Catalyzed/Cu-Assisted C-H Functionalization/Intramolecular C-S Bond Formation from -Arylcyanothioformamides.
Nathan Broudic, Alexandra Pacheco-Benichou, Corinne Fruit, Thierry Besson

Molecules· December 2022

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Straightforward Access to a New Class of Dual DYRK1A/CLK1 Inhibitors Possessing a Simple Dihydroquinoline Core.
Mihaela-Liliana Ţînţaş, Ludovic Peauger, Florent Alix, Cyril Papamicaël, Thierry Besson

Molecules· December 2022

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Relieving DYRK1A repression of MKL1 confers an adult-like phenotype to human infantile megakaryocytes.
Kamaleldin E Elagib, Ashton Brock, Cara M Clementelli, Goar Mosoyan, Lorrie L Delehanty, Thierry Besson

J Clin Invest· October 2022

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Therapeutic antibody glycosylation impacts antigen recognition and immunogenicity.
Babette Wolf, Mateusz Piksa, Isabelle Beley, Agnes Patoux, Thierry Besson

Immunology· July 2022

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Review on the Synthesis and Therapeutic Potential of Pyrido[2,3-], [3,2-], [3,4-] and [4,3-]pyrimidine Derivatives.
Joana F Campos, Thierry Besson, Sabine Berteina-Raboin

Pharmaceuticals (Basel)· March 2022

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Recent Advances in Transition-Metal-Free Late-Stage C-H and N-H Arylation of Heteroarenes Using Diaryliodonium Salts.
Thierry Besson, Corinne Fruit

Pharmaceuticals (Basel)· July 2021

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Microwave-Assisted Sequential One-Pot Synthesis of 8-Substituted Pyrazolo[1,5-][1,3,5]triazines.
Jonathan Elie, Corinne Fruit, Thierry Besson

Molecules· June 2021

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Demonstration of Green Solvent Performance on O,S,N-Heterocycles Synthesis: Metal-Free Click Chemistry and Buchwald-Hartwig Coupling.
Joana F Campos, Manon Cailler, Remi Claudel, Benjamin Prot, Thierry Besson

Molecules· February 2021

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DYRK1A regulates B cell acute lymphoblastic leukemia through phosphorylation of FOXO1 and STAT3.
Rahul S Bhansali, Malini Rammohan, Paul Lee, Anouchka P Laurent, Qiang Wen, Thierry Besson

J Clin Invest· January 2021

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Microwave-Assisted Synthesis of Potential Bioactive Benzo-, Pyrido- or Pyrazino-thieno[3,2-]pyrimidin-4-amine Analogs of MPC-6827.
Yvonnick Loidreau, Marie-Renée Nourrisson, Corinne Fruit, Cécile Corbière, Pascal Marchand, Thierry Besson

Pharmaceuticals (Basel)· August 2020

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Exploring Kinase Inhibition Properties of 9-pyrimido[5,4-]- and [4,5-]indol-4-amine Derivatives.
Yvonnick Loidreau, Carole Dubouilh-Benard, Marie-Renée Nourrisson, Nadège Loaëc, Laurent Meijer, Thierry Besson

Pharmaceuticals (Basel)· May 2020

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Biological Characterization of 8-Cyclopropyl-2-(pyridin-3-yl)thiazolo[5,4-]quinazolin-9(8)-one, a Promising Inhibitor of DYRK1A.
Corinne Fruit, Florence Couly, Rahul Bhansali, Malini Rammohan, Mattias F Lindberg, Thierry Besson

Pharmaceuticals (Basel)· December 2019

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26th Annual GP2A Medicinal Chemistry Conference & 32nd Journées Franco-Belges de Pharmacochimie.
Patrick Dallemagne, Christophe Rochais, Pascal Marchand, Thierry Besson

Pharmaceuticals (Basel)· May 2019

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Development of Kinase Inhibitors via Metal-Catalyzed C⁻H Arylation of 8-Alkyl-thiazolo[5,4-]-quinazolin-9-ones Designed by Fragment-Growing Studies.
Florence Couly, Marine Harari, Carole Dubouilh-Benard, Laetitia Bailly, Emilie Petit, Thierry Besson

Molecules· August 2018

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Synthesis of 2-Mercapto-(2-Oxoindolin-3-Ylidene)Acetonitriles from 3-(4-Chloro-5-1,2,3-Dithiazol-5-Ylidene)Indolin-2-ones.
Boris Letribot, Régis Delatouche, Hervé Rouillard, Antoine Bonnet, Jean-René Chérouvrier, Thierry Besson

Molecules· June 2018

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Dual-specificity tyrosine phosphorylation-regulated kinase 1A (DYRK1A) inhibitors: a survey of recent patent literature.
Thu Lan Nguyen, Corinne Fruit, Yann Hérault, Laurent Meijer, Thierry Besson

Expert Opin Ther Pat· November 2017

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An Unusual Binding Model of the Methyl 9-Anilinothiazolo[5,4-f] quinazoline-2-carbimidates (EHT 1610 and EHT 5372) Confers High Selectivity for Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases.
Apirat Chaikuad, Julien Diharce, Martin Schröder, Alicia Foucourt, Bertrand Leblond, Thierry Besson

J Med Chem· November 2016

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Pd-Catalyzed and Copper Assisted Regioselective Sequential C2 and C7 Arylation of Thiazolo[5,4-f]quinazolin-9(8H)-one with Aryl Halides.
Marine Harari, Florence Couly, Corinne Fruit, Thierry Besson

Org Lett· July 2016

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Synthesis of Bioactive 2-(Arylamino)thiazolo[5,4-f]-quinazolin-9-ones via the Hügershoff Reaction or Cu- Catalyzed Intramolecular C-S Bond Formation.
Damien Hédou, Carole Dubouilh-Benard, Nadège Loaëc, Laurent Meijer, Corinne Fruit, Thierry Besson

Molecules· June 2016

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Synthesis of Thiazolo[5,4-f]quinazolin-9(8H)-ones as Multi-Target Directed Ligands of Ser/Thr Kinases.
Damien Hédou, Julien Godeau, Nadège Loaëc, Laurent Meijer, Corinne Fruit, Thierry Besson

Molecules· April 2016

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