Publications by authors named "Thierry Calmels"

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Guanidine Derivative ADS1017, a Potent Histamine H Receptor Antagonist with Promising Analgesic Activity and Satisfactory Safety Profile.
Tadeusz Karcz, Katarzyna Szczepańska, Szczepan Mogilski, Aleksandra Moroz, Agnieszka Olejarz-Maciej, Thierry Calmels

ACS Chem Neurosci· December 2024

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Dual Piperidine-Based Histamine H and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain.
Katarzyna Szczepańska, Tadeusz Karcz, Maria Dichiara, Szczepan Mogilski, Justyna Kalinowska-Tłuścik, Thierry Calmels

J Med Chem· July 2023

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Discovery of nanomolar ligands with novel scaffolds for the histamine H4 receptor by virtual screening.
Nicolas Levoin, Olivier Labeeuw, Xavier Billot, Thierry Calmels, Denis Danvy

Eur J Med Chem· January 2017

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Synthesis and evaluation of a 2-benzothiazolylphenylmethyl ether class of histamine H4 receptor antagonists.
Olivier Labeeuw, Nicolas Levoin, Xavier Billot, Denis Danvy, Thierry Calmels

Bioorg Med Chem Lett· November 2016

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Improving selectivity of dopamine D3 receptor ligands.
Marc Capet, Thierry Calmels, Nicolas Levoin, Denis Danvy, Isabelle Berrebi-Bertrand

Bioorg Med Chem Lett· February 2016

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Determination of the binding mode and interacting amino-acids for dibasic H3 receptor antagonists.
Nicolas Levoin, Olivier Labeeuw, Stéphane Krief, Thierry Calmels, Olivia Poupardin-Olivier

Bioorg Med Chem· August 2013

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Novel and highly potent histamine H3 receptor ligands. Part 3: an alcohol function to improve the pharmacokinetic profile.
Olivier Labeeuw, Nicolas Levoin, Olivia Poupardin-Olivier, Thierry Calmels, Xavier Ligneau

Bioorg Med Chem Lett· May 2013

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Novel and highly potent histamine H3 receptor ligands. Part 2: exploring the cyclohexylamine-based series.
Olivier Labeeuw, Nicolas Levoin, Olivia Poupardin-Olivier, Thierry Calmels, Xavier Ligneau

Bioorg Med Chem Lett· September 2011

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Novel and highly potent histamine H3 receptor ligands. Part 1: withdrawing of hERG activity.
Nicolas Levoin, Olivier Labeeuw, Thierry Calmels, Olivia Poupardin-Olivier, Isabelle Berrebi-Bertrand

Bioorg Med Chem Lett· September 2011

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Homology Model Versus X-ray Structure in Receptor-based Drug Design: A Retrospective Analysis with the Dopamine D3 Receptor.
Nicolas Levoin, Thierry Calmels, Stéphane Krief, Denis Danvy, Isabelle Berrebi-Bertrand

ACS Med Chem Lett· April 2011

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Synthesis and evaluation of amides surrogates of dopamine D3 receptor ligands.
Mickaël Jean, Jacques Renault, Nicolas Levoin, Denis Danvy, Thierry Calmels

Bioorg Med Chem Lett· September 2010

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Connexin 30 is expressed in the mouse sino-atrial node and modulates heart rate.
Daniel Gros, Magali Théveniau-Ruissy, Monique Bernard, Thierry Calmels, Frank Kober

Cardiovasc Res· January 2010

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Refined docking as a valuable tool for lead optimization: application to histamine H3 receptor antagonists.
Nicolas Levoin, Thierry Calmels, Olivia Poupardin-Olivier, Olivier Labeeuw, Denis Danvy

Arch Pharm (Weinheim)· October 2008

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Hybrid approach for the design of highly affine and selective dopamine D(3) receptor ligands using privileged scaffolds of biogenic amine GPCR ligands.
Britta C Sasse, Ulrich R Mach, Jukka Leppaenen, Thierry Calmels, Holger Stark

Bioorg Med Chem· December 2007

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In situ hybridization: a technique to study localization of cardiac gene expression.
Thierry P Calmels, David Mazurais

Methods Mol Biol· July 2007

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Dysregulation of connexins and inactivation of NFATc1 in the cardiovascular system of Nkx2-5 null mutants.
Laurent Dupays, Thérèse Jarry-Guichard, David Mazurais, Thierry Calmels, Seigo Izumo

J Mol Cell Cardiol· May 2005

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Parallel synthesis and dopamine D3/D2 receptor screening of novel {4-[4-(2-methoxyphenyl)piperazin-1-yl]butyl}carboxamides.
Philipp Heidler, Vida Zohrabi-Kalantari, Thierry Calmels, Marc Capet, Isabelle Berrebi-Bertrand

Bioorg Med Chem· March 2005

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Genomic organization and alternative transcripts of the human Connexin40 gene.
Laurent Dupays, David Mazurais, Catherine Rücker-Martin, Thierry Calmels, Denis Bernot

Gene· February 2003

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Cell type-specific localization of human cardiac S1P receptors.
David Mazurais, Philippe Robert, Bernard Gout, Isabelle Berrebi-Bertrand, Marie Paule Laville, Thierry Calmels

J Histochem Cytochem· May 2002

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Human p63RhoGEF, a novel RhoA-specific guanine nucleotide exchange factor, is localized in cardiac sarcomere.
Michel Souchet, Elodie Portales-Casamar, David Mazurais, Susanne Schmidt, Isabelle Léger, Thierry P G Calmels

J Cell Sci· February 2002

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