Publications by authors named "Tibor Docsa"

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Regioselective Synthesis of 5-Substituted 3-(β-d-Glycopyranosyl)isoxazoles and -isoxazolines by 1,3-Dipolar Cycloaddition as Potential Anticancer Agents and Glycogen Phosphorylase Inhibitors.
Tímea Kaszás, Bence Szakács, Márta Bertalan, Tekla Blága, Faria Hameed, Tibor Docsa

Int J Mol Sci· August 2025

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Synthesis, In Silico and Kinetics Evaluation of -(β-d-glucopyranosyl)-2-arylimidazole-4(5)-carboxamides and -(β-d-glucopyranosyl)-4(5)-arylimidazole-2-carboxamides as Glycogen Phosphorylase Inhibitors.
Levente Homolya, Rachel T Mathomes, Luca Varga, Tibor Docsa, László Juhász

Int J Mol Sci· April 2024

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Stretch-Induced Down-Regulation of HCN2 Suppresses Contractile Activity.
Job Baffin Kola, Botagoz Turarova, Dora Csige, Ádám Sipos, Luca Varga, Tibor Docsa

Molecules· May 2023

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Design and Synthesis of 3-(β-d-Glucopyranosyl)-4-amino/4-guanidino Pyrazole Derivatives and Analysis of Their Glycogen Phosphorylase Inhibitory Potential.
Sándor Kun, Rachel T Mathomes, Tibor Docsa, László Somsák, Joseph M Hayes

Molecules· March 2023

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Mechanosensing in the Physiology and Pathology of the Gastrointestinal Tract.
Job Baffin Kola, Tibor Docsa, Karen Uray

Int J Mol Sci· December 2022

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The Role of Inflammatory Mediators in the Development of Gastrointestinal Motility Disorders.
Tibor Docsa, Adám Sipos, Charles S Cox, Karen Uray

Int J Mol Sci· June 2022

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Dual-Target Compounds against Type 2 : Proof of Concept for Sodium Dependent Glucose Transporter (SGLT) and Glycogen Phosphorylase (GP) Inhibitors.
Ádám Sipos, Eszter Szennyes, Nikolett Éva Hajnal, Sándor Kun, Katalin E Szabó, Tibor Docsa

Pharmaceuticals (Basel)· April 2021

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Glycogen phosphorylase inhibitor, 2,3-bis[(2E)-3-(4-hydroxyphenyl)prop-2-enamido] butanedioic acid (BF142), improves baseline insulin secretion of MIN6 insulinoma cells.
Lilla Nagy, Ferenc Béke, László Juhász, Tünde Kovács, Éva Juhász-Tóth, Tibor Docsa

PLoS One· October 2020

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CXCL1 is upregulated during the development of ileus resulting in decreased intestinal contractile activity.
Tibor Docsa, Deepa Bhattarai, Adam Sipos, Charles E Wade, Charles S Cox

Neurogastroenterol Motil· March 2020

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Glucose-based spiro-oxathiazoles as in vivo anti-hyperglycemic agents through glycogen phosphorylase inhibition.
David Goyard, Bálint Kónya, Katalin Czifrák, Paolo Larini, Fanny Demontrond, Tibor Docsa

Org Biomol Chem· February 2020

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Identification of -β-d-Glucopyranosyl Azole-Type Inhibitors of Glycogen Phosphorylase That Reduce Glycogenolysis in Hepatocytes: Design, Synthesis, Kinetics, and Studies.
Daniel Barr, Eszter Szennyes, Éva Bokor, Ziad H Al-Oanzi, Colin Moffatt, Tibor Docsa

ACS Chem Biol· July 2019

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Glucopyranosylidene-spiro-imidazolinones, a New Ring System: Synthesis and Evaluation as Glycogen Phosphorylase Inhibitors by Enzyme Kinetics and X-ray Crystallography.
Katalin E Szabó, Efthimios Kyriakis, Anna-Maria G Psarra, Aikaterini G Karra, Ádám Sipos, Tibor Docsa

J Med Chem· July 2019

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Glucopyranosylidene-spiro-benzo[ b][1,4]oxazinones and -benzo[ b][1,4]thiazinones: Synthesis and Investigation of Their Effects on Glycogen Phosphorylase and Plant Growth Inhibition.
Sándor Kun, Nándor Kánya, Norbert Galó, András Páhi, Attila Mándi, Tibor Docsa

J Agric Food Chem· June 2019

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Synthesis of C-β-d-glucopyranosyl derivatives of some fused azoles for the inhibition of glycogen phosphorylase.
Eszter Szennyes, Éva Bokor, Tibor Docsa, Ádám Sipos, László Somsák

Carbohydr Res· January 2019

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A multidisciplinary study of 3-(β-d-glucopyranosyl)-5-substituted-1,2,4-triazole derivatives as glycogen phosphorylase inhibitors: Computation, synthesis, crystallography and kinetics reveal new potent inhibitors.
Sándor Kun, Jaida Begum, Efthimios Kyriakis, Evgenia C V Stamati, Thomas A Barkas, Tibor Docsa

Eur J Med Chem· March 2018

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Synthesis of New C- and N-β-d-Glucopyranosyl Derivatives of Imidazole, 1,2,3-Triazole and Tetrazole, and Their Evaluation as Inhibitors of Glycogen Phosphorylase.
Sándor Kun, Éva Bokor, Ádám Sipos, Tibor Docsa, László Somsák

Molecules· March 2018

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Glycogen phosphorylase inhibition improves beta cell function.
Lilla Nagy, Judit Márton, András Vida, Gréta Kis, Éva Bokor, Tibor Docsa

Br J Pharmacol· January 2018

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Nanomolar Inhibitors of Glycogen Phosphorylase Based on β-d-Glucosaminyl Heterocycles: A Combined Synthetic, Enzyme Kinetic, and Protein Crystallography Study.
Éva Bokor, Efthimios Kyriakis, Theodora G A Solovou, Csenge Koppány, Anastassia L Kantsadi, Tibor Docsa

J Med Chem· November 2017

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Synthetic, enzyme kinetic, and protein crystallographic studies of C-β-d-glucopyranosyl pyrroles and imidazoles reveal and explain low nanomolar inhibition of human liver glycogen phosphorylase.
Anastassia L Kantsadi, Éva Bokor, Sándor Kun, George A Stravodimos, Demetra S M Chatzileontiadou, Tibor Docsa

Eur J Med Chem· November 2016

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Insulin sensitivity is modified by a glycogen phosphorylase inhibitor: glucopyranosylidene-spiro-thiohydantoin in streptozotocin-induced diabetic rats.
Tibor Docsa, Balázs Marics, József Németh, Csaba Hüse, László Somsák

Curr Top Med Chem· June 2016

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C-Glucopyranosyl-1,2,4-triazol-5-ones: synthesis and inhibition of glycogen phosphorylase.
Éva Bokor, Zsolt Széles, Tibor Docsa, Pál Gergely, László Somsák

Carbohydr Res· June 2016

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Glucose-derived spiro-isoxazolines are anti-hyperglycemic agents against type 2 diabetes through glycogen phosphorylase inhibition.
David Goyard, Bálint Kónya, Aikaterini S Chajistamatiou, Evangelia D Chrysina, Jérémy Leroy, Tibor Docsa

Eur J Med Chem· January 2016

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4(5)-Aryl-2-C-glucopyranosyl-imidazoles as New Nanomolar Glucose Analogue Inhibitors of Glycogen Phosphorylase.
Éva Bokor, Sándor Kun, Tibor Docsa, Pál Gergely, László Somsák

ACS Med Chem Lett· December 2015

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C-(2-Deoxy-d-arabino-hex-1-enopyranosyl)-oxadiazoles: synthesis of possible isomers and their evaluation as glycogen phosphorylase inhibitors.
Éva Bokor, Eszter Szennyes, Tibor Csupász, Nóra Tóth, Tibor Docsa

Carbohydr Res· August 2015

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3-Glucosylated 5-amino-1,2,4-oxadiazoles: synthesis and evaluation as glycogen phosphorylase inhibitors.
Marion Donnier-Maréchal, David Goyard, Vincent Folliard, Tibor Docsa, Pal Gergely

Beilstein J Org Chem· May 2015

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