Publications by authors named "Adel A Rashad"

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Selective and brain-penetrant ACSS2 inhibitors target breast cancer brain metastatic cells.
Emily M Esquea, Lorela Ciraku, Riley G Young, Jessica Merzy, Alexandra N Talarico, Adel A Rashad

Front Pharmacol· May 2024

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Discovery of novel brain permeable human ACSS2 inhibitors for blocking breast cancer brain metastatic growth.
Emily Esquea, Lorela Ciraku, Riley G Young, Jessica Merzy, Alexandra N Talarico, Adel Ahmed Rashad

bioRxiv· December 2023

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Discovery of a first-in-class inhibitor of sulfide:quinone oxidoreductase that protects against adverse cardiac remodelling and heart failure.
Michael R Jackson, Kristie D Cox, Simon D P Baugh, Luke Wakeen, Adel A Rashad

Cardiovasc Res· June 2022

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Synthesis and evaluation of potent novel inhibitors of human sulfide:quinone oxidoreductase.
Simon D P Baugh, Michael R Jackson, Adel Ahmed Rashad, Allen B Reitz, Patrick Y S Lam

Bioorg Med Chem Lett· December 2021

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Altered Env conformational dynamics as a mechanism of resistance to peptide-triazole HIV-1 inactivators.
Shiyu Zhang, Andrew P Holmes, Alexej Dick, Adel A Rashad, Lucía Enríquez Rodríguez

Retrovirology· October 2021

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Bioactive Polyphenolic Compounds Showing Strong Antiviral Activities against Severe Acute Respiratory Syndrome Coronavirus 2.
Ahmed Kandeil, Ahmed Mostafa, Omnia Kutkat, Yassmin Moatasim, Ahmed A Al-Karmalawy, Adel A Rashad

Pathogens· June 2021

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Peptide Triazole Thiol Irreversibly Inactivates Metastable HIV-1 Env by Accessing Conformational Triggers Intrinsic to Virus-Cell Entry.
Charles Gotuaco Ang, Erik Carter, Ann Haftl, Shiyu Zhang, Adel A Rashad

Microorganisms· June 2021

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FDA-Approved Drugs with Potent In Vitro Antiviral Activity against Severe Acute Respiratory Syndrome Coronavirus 2.
Ahmed Mostafa, Ahmed Kandeil, Yaseen A M M Elshaier, Omnia Kutkat, Yassmin Moatasim, Adel A Rashad

Pharmaceuticals (Basel)· December 2020

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Click Chemistry for Cyclic Peptide Drug Design.
Adel Ahmed Rashad

Methods Mol Biol· March 2020

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Metastable HIV-1 Surface Protein Env Sensitizes Cell Membranes to Transformation and Poration by Dual-Acting Virucidal Entry Inhibitors.
Charles G Ang, Md Alamgir Hossain, Marg Rajpara, Harry Bach, Kriti Acharya, Adel A Rashad

Biochemistry· February 2020

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Pharmacokinetic stability of macrocyclic peptide triazole HIV-1 inactivators alone and in liposomes.
Rachna Aneja, Antonella Grigoletto, Aakansha Nangarlia, Adel A Rashad, Steven Wrenn

J Pept Sci· April 2019

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Field-Based Affinity Optimization of a Novel Azabicyclohexane Scaffold HIV-1 Entry Inhibitor.
Megan E Meuser, Adel A Rashad, Gabriel Ozorowski, Alexej Dick, Andrew B Ward

Molecules· April 2019

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Kinetic Characterization of Novel HIV-1 Entry Inhibitors: Discovery of a Relationship between Off-Rate and Potency.
Megan E Meuser, Michael B Murphy, Adel A Rashad, Simon Cocklin

Molecules· August 2018

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Exploring Modifications of an HIV-1 Capsid Inhibitor: Design, Synthesis, and Mechanism of Action.
Jimmy P Xu, Ashwanth C Francis, Megan E Meuser, Marie Mankowski, Roger G Ptak, Adel A Rashad

J Drug Des Res· August 2018

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Bifunctional Chimera That Coordinately Targets Human Immunodeficiency Virus 1 Envelope gp120 and the Host-Cell CCR5 Coreceptor at the Virus-Cell Interface.
Adel A Rashad, Li-Rui Song, Andrew P Holmes, Kriti Acharya, Shiyu Zhang

J Med Chem· June 2018

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Chemical optimization of macrocyclic HIV-1 inactivators for improving potency and increasing the structural diversity at the triazole ring.
Adel A Rashad, Kriti Acharya, Ann Haftl, Rachna Aneja, Alexej Dick

Org Biomol Chem· September 2017

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Recognition of HIV-inactivating peptide triazoles by the recombinant soluble Env trimer, BG505 SOSIP.664.
Kriti Acharya, Adel A Rashad, Francesca Moraca, Per Johan Klasse, John P Moore

Proteins· May 2017

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Lytic Inactivation of Human Immunodeficiency Virus by Dual Engagement of gp120 and gp41 Domains in the Virus Env Protein Trimer.
Bibek Parajuli, Kriti Acharya, Reina Yu, Brendon Ngo, Adel A Rashad

Biochemistry· November 2016

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Peptide triazole inactivators of HIV-1: how do they work and what is their potential?
Irwin Chaiken, Adel A Rashad

Future Med Chem· September 2016

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Short Communication: Inhibition of DC-SIGN-Mediated HIV-1 Infection by Complementary Actions of Dendritic Cell Receptor Antagonists and Env-Targeting Virus Inactivators.
Sergey Pustylnikov, Rajnish S Dave, Zafar K Khan, Vanessa Porkolab, Adel A Rashad

AIDS Res Hum Retroviruses· January 2016

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Impact of HIV-1 Membrane Cholesterol on Cell-Independent Lytic Inactivation and Cellular Infectivity.
Ramalingam Venkat Kalyana Sundaram, Huiyuan Li, Lauren Bailey, Adel A Rashad, Rachna Aneja

Biochemistry· January 2016

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Disulfide Sensitivity in the Env Protein Underlies Lytic Inactivation of HIV-1 by Peptide Triazole Thiols.
Lauren D Bailey, Ramalingam Venkat Kalyana Sundaram, Huiyuan Li, Caitlin Duffy, Rachna Aneja, Adel A Rashad

ACS Chem Biol· December 2015

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Macrocyclic Envelope Glycoprotein Antagonists that Irreversibly Inactivate HIV-1 before Host Cell Encounter.
Adel A Rashad, Ramalingam Venkat Kalyana Sundaram, Rachna Aneja, Caitlin Duffy, Irwin Chaiken

J Med Chem· September 2015

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Peptide Triazole Inactivators of HIV-1 Utilize a Conserved Two-Cavity Binding Site at the Junction of the Inner and Outer Domains of Env gp120.
Rachna Aneja, Adel A Rashad, Huiyuan Li, Ramalingam Venkat Kalyana Sundaram, Caitlin Duffy

J Med Chem· May 2015

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Facile Synthesis and Preliminary Structure-Activity Analysis of New Sulfonamides Against Trypanosoma brucei.
Adel A Rashad, Amy J Jones, Vicky M Avery, Jonathan Baell, Paul A Keller

ACS Med Chem Lett· May 2014

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