Publications by authors named "Albert Robichaud"

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Pharmacological characterization of SAGE-718, a novel positive allosteric modulator of N-methyl-d-aspartate receptors.
Jacob T Beckley, Teresa K Aman, Michael A Ackley, Tatiana M Kazdoba, Michael C Lewis, Albert J Robichaud

Br J Pharmacol· April 2024

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Novel neuroactive steroids as positive allosteric modulators of NMDA receptors: mechanism, site of action, and rescue pharmacology on GRIN variants associated with neurological conditions.
Weiting Tang, Jacob T Beckley, Jin Zhang, Rui Song, Yuchen Xu, Albert J Robichaud

Cell Mol Life Sci· January 2023

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SAGE-718: A First-in-Class -Methyl-d-Aspartate Receptor Positive Allosteric Modulator for the Potential Treatment of Cognitive Impairment.
Matthew D Hill, Maria-Jesus Blanco, Francesco G Salituro, Zhu Bai, Jacob T Beckley, Albert J Robichaud

J Med Chem· July 2022

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Preclinical characterization of zuranolone (SAGE-217), a selective neuroactive steroid GABA receptor positive allosteric modulator.
Alison L Althaus, Michael A Ackley, Gabriel M Belfort, Steven M Gee, Jing Dai, Albert J Robichaud

Neuropharmacology· December 2020

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Neuroactive Steroid -Methyl-d-aspartate Receptor Positive Allosteric Modulators: Synthesis, SAR, and Pharmacological Activity.
Daniel S La, Francesco G Salituro, Gabriel Martinez Botella, Andrew M Griffin, Zhu Bai, Albert J Robichaud

J Med Chem· August 2019

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Allosteric Modalities for Membrane-Bound Receptors: Insights from Drug Hunting for Brain Diseases.
Quinn Coughlin, Allen T Hopper, Maria-Jesus Blanco, Vijaya Tirunagaru, Albert J Robichaud

J Med Chem· July 2019

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Neuroactive Steroids. 2. 3α-Hydroxy-3β-methyl-21-(4-cyano-1H-pyrazol-1'-yl)-19-nor-5β-pregnan-20-one (SAGE-217): A Clinical Next Generation Neuroactive Steroid Positive Allosteric Modulator of the (γ-Aminobutyric Acid) Receptor.
Gabriel Martinez Botella, Francesco G Salituro, Boyd L Harrison, Richard T Beresis, Zhu Bai, Albert J Robichaud

J Med Chem· September 2017

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Anticonvulsant profile of the neuroactive steroid, SGE-516, in animal models.
Rebecca S Hammond, Alison L Althaus, Michael A Ackley, Carla Maciag, Gabriel Martinez Botella, Albert J Robichaud

Epilepsy Res· August 2017

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The synthetic neuroactive steroid SGE-516 reduces status epilepticus and neuronal cell death in a rat model of soman intoxication.
Alison L Althaus, Hilary S McCarren, Aymen Alqazzaz, Cecelia Jackson, John H McDonough, Albert J Robichaud

Epilepsy Behav· March 2017

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Rescue of deficient amygdala tonic γ-aminobutyric acidergic currents in the Fmr-/y mouse model of fragile X syndrome by a novel γ-aminobutyric acid type A receptor-positive allosteric modulator.
Brandon S Martin, Gabriel Martinez-Botella, Carlos M Loya, Francesco G Salituro, Albert J Robichaud

J Neurosci Res· June 2016

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Neuroactive Steroids. 1. Positive Allosteric Modulators of the (γ-Aminobutyric Acid)A Receptor: Structure-Activity Relationships of Heterocyclic Substitution at C-21.
Gabriel Martinez Botella, Francesco G Salituro, Boyd L Harrison, Richard T Beresis, Zhu Bai, Albert J Robichaud

J Med Chem· April 2015

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Discovery of a tetracyclic quinoxaline derivative as a potent and orally active multifunctional drug candidate for the treatment of neuropsychiatric and neurological disorders.
Peng Li, Qiang Zhang, Albert J Robichaud, Taekyu Lee, John Tomesch

J Med Chem· March 2014

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The major brain cholesterol metabolite 24(S)-hydroxycholesterol is a potent allosteric modulator of N-methyl-D-aspartate receptors.
Steven M Paul, James J Doherty, Albert J Robichaud, Gabriel M Belfort, Brian Y Chow

J Neurosci· October 2013

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Fused thiazolyl alkynes as potent mGlu5 receptor positive allosteric modulators.
Mathivanan Packiarajan, Michel Grenon, Samuel Zorn, Allen T Hopper, Andrew D White, Albert J Robichaud

Bioorg Med Chem Lett· July 2013

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Azetidinyl oxadiazoles as potent mGluR5 positive allosteric modulators.
Mathivanan Packiarajan, Christine G Mazza Ferreira, Sang-Phyo Hong, Andrew D White, Gamini Chandrasena, Albert J Robichaud

Bioorg Med Chem Lett· October 2012

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N-Aryl pyrrolidinonyl oxadiazoles as potent mGluR5 positive allosteric modulators.
Mathivanan Packiarajan, Christine G Mazza Ferreira, Sang-Phyo Hong, Andrew D White, Gamini Chandrasena, Albert J Robichaud

Bioorg Med Chem Lett· September 2012

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Novel triazines as potent and selective phosphodiesterase 10A inhibitors.
Michael S Malamas, Hans Stange, Rudolf Schindler, Hans-Joachim Lankau, Christian Grunwald, Albert Robichaud

Bioorg Med Chem Lett· September 2012

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2-(Pyrrolidin-1-yl)ethyl-3,4-dihydroisoquinolin-1(2H)-one derivatives as potent and selective histamine-3 receptor antagonists.
Dahui Zhou, Jonathan L Gross, Adedayo B Adedoyin, Suzan B Aschmies, Julie Brennan, Albert J Robichaud

J Med Chem· March 2012

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Highly potent, selective, and orally active phosphodiesterase 10A inhibitors.
Michael S Malamas, Yike Ni, James Erdei, Hans Stange, Rudolf Schindler, Albert Robichaud

J Med Chem· November 2011

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Pyrrolidin-3-yl-N-methylbenzamides as potent histamine 3 receptor antagonists.
Dahui Zhou, Jonathan L Gross, Jean Y Sze, Adedayo B Adedoyin, Mark Bowlby, Albert J Robichaud

Bioorg Med Chem Lett· October 2011

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5-HT6 medicinal chemistry.
Kevin G Liu, Albert J Robichaud

Int Rev Neurobiol· September 2011

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New pyrazolyl and thienyl aminohydantoins as potent BACE1 inhibitors: exploring the S2' region.
Michael S Malamas, Jim Erdei, Iwan Gunawan, Keith Barnes, Yu Hui, Albert Robichaud

Bioorg Med Chem Lett· September 2011

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Recent progress on the identification of metabotropic glutamate 4 receptor ligands and their potential utility as CNS therapeutics.
Albert J Robichaud, Darren W Engers, Craig W Lindsley, Corey R Hopkins

ACS Chem Neurosci· August 2011

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Tricyclic thiazolopyrazole derivatives as metabotropic glutamate receptor 4 positive allosteric modulators.
Sang-Phyo Hong, Kevin G Liu, Gil Ma, Michael Sabio, Michelle A Uberti, Albert J Robichaud

J Med Chem· July 2011

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Identification of 3-sulfonylindazole derivatives as potent and selective 5-HT(6) antagonists.
Kevin G Liu, Albert J Robichaud, Alexander A Greenfield, Jennifer R Lo, Cristina Grosanu

Bioorg Med Chem· January 2011

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