Publications by authors named "Andrew Beekman"

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Screening herbal and natural product libraries to aid discovery of novel allosteric modulators of human P2X7.
Stefan Bidula, Waraporn Piyasirananda, Hanna Bielecka, Lučka Bibič, Andrew Beekman

Purinergic Signal· April 2025

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Peptide design to control protein-protein interactions.
Suzanne P van Wier, Andrew M Beekman

Chem Soc Rev· February 2025

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Carbonyl reductase 1: a novel regulator of blood pressure in Down syndrome.
Alexandra J Malbon, Alicja Czopek, Andrew M Beekman, Zoë R Goddard, Aileen Boyle

Biosci Rep· February 2025

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Light-activated azobenzene peptide inhibitor of the PD-1/PD-L1 interaction.
Deanne Hayward, Zoë R Goddard, Marco M D Cominetti, Mark Searcey, Andrew M Beekman

Chem Commun (Camb)· August 2024

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Borylation iridium catalysed C-H activation: a new concise route to duocarmycin derivatives.
Marco M D Cominetti, Zoë R Goddard, Bethany R Hood, Andrew M Beekman, Maria A O'Connell

Org Biomol Chem· July 2024

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Strategies for converting turn-motif and cyclic peptides to small molecules for targeting protein-protein interactions.
Deanne Hayward, Andrew M Beekman

RSC Chem Biol· March 2024

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Insights into the Structure-Activity Relationship of Glycosides as Positive Allosteric Modulators Acting on P2X7 Receptors.
Waraporn Piyasirananda, Andrew Beekman, A Ganesan, Stefan Bidula, Leanne Stokes

Mol Pharmacol· February 2021

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peptide-directed ligand design complements experimental peptide-directed binding for protein-protein interaction modulator discovery.
Lesley Ann Howell, Andrew Michael Beekman

RSC Chem Biol· February 2021

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Peptide directed phthalocyanine-gold nanoparticles for selective photodynamic therapy of EGFR overexpressing cancers.
Zoë Rachael Goddard, Andrew Michael Beekman, Marco M D Cominetti, Maria A O'Connell, Isabelle Chambrier

RSC Med Chem· November 2020

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A Peptide-Duocarmycin Conjugate Targeting the Thomsen-Friedenreich Antigen Has Potent and Selective Antitumor Activity.
Oliver Charles Cartwright, Andrew Michael Beekman, Marco M D Cominetti, David A Russell, Mark Searcey

Bioconjug Chem· July 2020

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A small molecule drug conjugate (SMDC) of DUPA and a duocarmycin built on the solid phase.
Andrew Michael Beekman, Marco M D Cominetti, Oliver Charles Cartwright, Dale L Boger, Mark Searcey

Medchemcomm· December 2019

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Identification of selective protein-protein interaction inhibitors using efficient peptide-directed ligand design.
Andrew M Beekman, Marco M D Cominetti, Samuel J Walpole, Saurabh Prabhu, Maria A O'Connell

Chem Sci· April 2019

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Rac1 plays a role in CXCL12 but not CCL3-induced chemotaxis and Rac1 GEF inhibitor NSC23766 has off target effects on CXCR4.
Shirley C Mills, Lesley Howell, Andrew Beekman, Leanne Stokes, Anja Mueller

Cell Signal· January 2018

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Peptide-Directed Binding for the Discovery of Modulators of α-Helix-Mediated Protein-Protein Interactions: Proof-of-Concept Studies with the Apoptosis Regulator Mcl-1.
Andrew Michael Beekman, Maria Anne O'Connell, Lesley Ann Howell

Angew Chem Int Ed Engl· August 2017

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Identification of Small-Molecule Inhibitors of the Antiapoptotic Protein Myeloid Cell Leukaemia-1 (Mcl-1).
Andrew M Beekman, Maria A O'Connell, Lesley A Howell

ChemMedChem· April 2016

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Small-Molecule and Peptide Inhibitors of the Pro-Survival Protein Mcl-1.
Andrew M Beekman, Lesley A Howell

ChemMedChem· April 2016

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Discovery and Synthesis of Boletopsins 13 and 14, Brominated Fungal Metabolites of Terrestrial Origin.
Andrew M Beekman, Stewart W Wossa, Oromo Kevo, Paul Ma, Russell A Barrow

J Nat Prod· August 2015

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Syntheses of the fungal metabolites boletopsins 7, 11, and 12 from the Papua New Guinea medicinal mushroom Boletopsis sp.
Andrew M Beekman, Russell A Barrow

J Org Chem· February 2014

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Stereochemical assignment of the fungal metabolites pestalotiopsones D and E through enantiopure synthesis.
Andrew Michael Beekman, Russell Allan Barrow

J Nat Prod· November 2013

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First syntheses of the biologically active fungal metabolites pestalotiopsones A, B, C and F.
Andrew Michael Beekman, Edwin Castillo Martinez, Russell Allan Barrow

Org Biomol Chem· February 2013

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