Publications by authors named "Angus Morrison"

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High-Throughput Screening of Potent Drug-like Molecules Targeting 17β-HSD10 for the Treatment of Alzheimer's Disease and Cancer.
Laura Aitken, Gemma Baillie, Andrew Pannifer, Angus Morrison, Louise L Major

ACS Chem Biol· July 2025

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Optimization of Cyclophilin B-Targeted Tri-vector Inhibitors for Novel MASH Treatments.
Maria-Eleni Kouridaki, Jonathan Gillespie, John Robinson, Tanya Mathie, Laura Bain, Angus Morrison

J Med Chem· March 2025

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Cell-active small molecule inhibitors validate the SNM1A DNA repair nuclease as a cancer target.
Marcin Bielinski, Lucy R Henderson, Yuliana Yosaatmadja, Lonnie P Swift, Hannah T Baddock, Angus Morrison

Chem Sci· May 2024

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The Discovery of New Inhibitors of Insulin-Regulated Aminopeptidase by a High-Throughput Screening of 400,000 Drug-like Compounds.
Johan Gising, Saman Honarnejad, Maaike Bras, Gemma L Baillie, Stuart P McElroy, Angus Morrison

Int J Mol Sci· April 2024

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Investigating the Structure-Activity Relationship of 1,2,4-Triazine G-Protein-Coupled Receptor 84 (GPR84) Antagonists.
Amit Mahindra, Laura Jenkins, Sara Marsango, Mark Huggett, Margaret Huggett, Angus Morrison

J Med Chem· August 2022

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IMI European Lead Factory - democratizing access to high-throughput screening.
Philip S Jones, Sylviane Boucharens, Stuart P McElroy, Angus Morrison, Saman Honarnejad

Nat Rev Drug Discov· April 2022

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Development of a High-Throughput Screening Assay for Small-Molecule Inhibitors of Androgen Receptor Splice Variants.
Amy E Monaghan, Alison Porter, Irene Hunter, Angus Morrison, Stuart P McElroy

Assay Drug Dev Technol· April 2022

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Standard method for performing positron emission particle tracking (PEPT) measurements of froth flotation at PEPT Cape Town.
Katie Cole, Daniel J Barker, Pablo R Brito-Parada, Andy Buffler, Kathryn Hadler, Angus J Morrison

MethodsX· March 2022

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Imitation of β-lactam binding enables broad-spectrum metallo-β-lactamase inhibitors.
Jürgen Brem, Tharindi Panduwawala, Jon Ulf Hansen, Joanne Hewitt, Edgars Liepins, Angus Morrison

Nat Chem· January 2022

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Discovery and Characterization of Novel Antagonists of the Proinflammatory Orphan Receptor GPR84.
Laura Jenkins, Sara Marsango, Sarah Mancini, Zobaer Al Mahmud, Angus Morrison

ACS Pharmacol Transl Sci· October 2021

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The identification and characterisation of autophagy inhibitors from the published kinase inhibitor sets.
Maria Zachari, Julie M Rainard, George C Pandarakalam, Lindsay Robinson, Jonathan Gillespie, Angus Morrison

Biochem J· February 2020

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Synthesis and Structure-Activity Relationships of N-(4-Benzamidino)-Oxazolidinones: Potent and Selective Inhibitors of Kallikrein-Related Peptidase 6.
Elena De Vita, Niels Smits, Helma van den Hurk, Elizabeth M Beck, Joanne Hewitt, Angus Morrison

ChemMedChem· January 2020

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Identification of A Novel Class of Benzofuran Oxoacetic Acid-Derived Ligands that Selectively Activate Cellular EPAC1.
Elizabeth M Beck, Euan Parnell, Angela Cowley, Alison Porter, Jonathan Gillespie, Angus Morrison

Cells· November 2019

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In Vitro Assay Development and HTS of Small-Molecule Human ABAD/17β-HSD10 Inhibitors as Therapeutics in Alzheimer's Disease.
Laura Aitken, Gemma Baillie, Andrew Pannifer, Angus Morrison, Philip S Jones

SLAS Discov· July 2017

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The importance of triaging in determining the quality of output from high-throughput screening.
Philip Jones, Stuart McElroy, Angus Morrison, Andrew Pannifer

Future Med Chem· July 2016

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Total syntheses of multiple cladiellin natural products by use of a completely general strategy.
J Stephen Clark, Raphaëlle Berger, Stewart T Hayes, Hans Martin Senn, Louis J Farrugia, Angus J Morrison

J Org Chem· January 2013

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Modified Shapiro reactions with bismesitylmagnesium as an efficient base reagent.
William J Kerr, Angus J Morrison, Marek Pazicky, Tina Weber

Org Lett· May 2012

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Low brain penetrant CB1 receptor agonists for the treatment of neuropathic pain.
Julia M Adam, John K Clark, Keneth Davies, Kathryn Everett, Ruth Fields, Angus Morrison

Bioorg Med Chem Lett· April 2012

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Design, synthesis and structure-activity relationships of (indo-3-yl) heterocyclic derivatives as agonists of the CB1 receptor. Discovery of a clinical candidate.
Paul Ratcliffe, Julia M Adam, James Baker, Roberta Bursi, Robert Campbell, Angus Morrison

Bioorg Med Chem Lett· April 2011

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Discovery of potent and orally bioavailable heterocycle-based cannabinoid CB1 receptor agonists.
Takao Kiyoi, Julia M Adam, John K Clark, Keneth Davies, Anna-Marie Easson, Angus J Morrison

Bioorg Med Chem Lett· March 2011

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Design, synthesis, and structure-activity relationships of indole-3-heterocycles as agonists of the CB1 receptor.
Angus J Morrison, Julia M Adam, James A Baker, Robert A Campbell, John K Clark

Bioorg Med Chem Lett· January 2011

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Enantioselective total syntheses of three cladiellins (eunicellins): a general approach to the entire family of natural products.
J Stephen Clark, Raphaëlle Berger, Stewart T Hayes, Lynne H Thomas, Angus J Morrison

Angew Chem Int Ed Engl· December 2010

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Trapping of palindromic ligands within native transthyretin prevents amyloid formation.
Simon E Kolstoe, Palma P Mangione, Vittorio Bellotti, Graham W Taylor, Glenys A Tennent, Angus J Morrison

Proc Natl Acad Sci U S A· November 2010

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Plagiarizing proteins: enhancing efficiency in asymmetric hydrogen-bonding catalysis through positive cooperativity.
Christopher R Jones, G Dan Pantoş, Angus J Morrison, Martin D Smith

Angew Chem Int Ed Engl· December 2009

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A nonpeptidic reverse turn that promotes parallel sheet structure stabilized by C-H...O hydrogen bonds in a cyclopropane gamma-peptide.
Christopher R Jones, M Khurram N Qureshi, Fiona R Truscott, Shang-Te Danny Hsu, Angus J Morrison

Angew Chem Int Ed Engl· October 2008

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