Publications by authors named "Anne Valade"

Claim this Profile
D
Discovery and Characterization of a Novel Series of Chloropyrimidines as Covalent Inhibitors of the Kinase MSK1.
Adrian Hall, Jan Abendroth, Madison J Bolejack, Tom Ceska, Sylvie Dell'Aiera, Anne Valade

ACS Med Chem Lett· July 2022

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
C
Crystal structure of dopamine D1 receptor in complex with G protein and a non-catechol agonist.
Bingfa Sun, Dan Feng, Matthew Ling-Hon Chu, Inbar Fish, Silvia Lovera, Anne Valade

Nat Commun· June 2021

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
N
Novel Strategies To Activate the Dopamine D Receptor: Recent Advances in Orthosteric Agonism and Positive Allosteric Modulation.
Adrian Hall, Laurent Provins, Anne Valade

J Med Chem· January 2019

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
A
Alkene protection against acid using a bromide substituent: application in a total synthesis of (-)-6,7-dideoxysqualestatin H5.
Hasanain A A Almohseni, Hamad H Al Mamari, Anne Valade, Herman O Sintim, David M Hodgson

Chem Commun (Camb)· May 2018

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
M
Measuring brain synaptic vesicle protein 2A with positron emission tomography and [F]UCB-H.
Mohamed Ali Bahri, Alain Plenevaux, Joël Aerts, Christine Bastin, Guillaume Becker, Anne Valade

Alzheimers Dement (N Y)· November 2017

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
D
Discovery and development of SV2A PET tracers: Potential for imaging synaptic density and clinical applications.
Joel Mercier, Laurent Provins, Anne Valade

Drug Discov Today Technol· November 2017

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
E
Evaluation of 18F-UCB-H as a novel PET tracer for synaptic vesicle protein 2A in the brain.
Geoffrey I Warnock, Joël Aerts, Mohamed Ali Bahri, Florian Bretin, Christian Lemaire, Anne Valade

J Nucl Med· August 2014

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
D
Discovery of heterocyclic nonacetamide synaptic vesicle protein 2A (SV2A) ligands with single-digit nanomolar potency: opening avenues towards the first SV2A positron emission tomography (PET) ligands.
Joël Mercier, Laurence Archen, Véronique Bollu, Stéphane Carré, Yves Evrard, Anne Valade

ChemMedChem· April 2014

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
P
Preclinical radiation dosimetry for the novel SV2A radiotracer [18F]UCB-H.
Florian Bretin, Geoffrey Warnock, Mohamed Ali Bahri, Joël Aerts, Nathalie Mestdagh, Anne Valade

EJNMMI Res· May 2013

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
L
Lead optimization of thiazolo[5,4-c]piperidines: 3-cyclobutoxy linker as a key spacer for H(3)R inverse agonists.
Laurent Provins, Frédéric Denonne, Sylvain Célanire, Bernard Christophe, Sabine Defays, Anne Valade

ChemMedChem· December 2012

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
P
Primary amino acid derivatives: substitution of the 4'-N'-benzylamide site in (R)-N'-benzyl 2-amino-3-methylbutanamide, (R)-N'-benzyl 2-amino-3,3-dimethylbutanamide, and (R)-N'-benzyl 2-amino-3-methoxypropionamide provides potent anticonvulsants with pain-attenuating properties.
Amber M King, Christophe Salomé, Elise Salomé-Grosjean, Marc De Ryck, Rafal Kaminski, Anne Valade

J Med Chem· October 2011

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
D
Defining the structural parameters that confer anticonvulsant activity by the site-by-site modification of (R)-N'-benzyl 2-amino-3-methylbutanamide.
Amber M King, Marc De Ryck, Rafal Kaminski, Anne Valade, James P Stables

J Med Chem· October 2011

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
P
Primary amino acid derivatives: compounds with anticonvulsant and neuropathic pain protection activities.
Amber M King, Christophe Salomé, Jason Dinsmore, Elise Salomé-Grosjean, Marc De Ryck, Anne Valade

J Med Chem· July 2011

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
T
Two galactosyltransferases' selection of different binders from the same uridine-based dynamic combinatorial library.
Anne Valade, Dominique Urban, Jean-Marie Beau

J Comb Chem· March 2007

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis
T
Target-assisted selection of galactosyltransferase binders from dynamic combinatorial libraries. An unexpected solution with restricted amounts of the enzyme.
Anne Valade, Dominique Urban, Jean-Marie Beau

Chembiochem· July 2006

Social Media Activity not collected for this article yet.

Sign Up to Request Social Media Analysis