Publications by authors named "Craig Masse"

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Discovery of a Potent and Selective Tyrosine Kinase 2 Inhibitor: TAK-279.
Silvana Leit, Jeremy Greenwood, Samantha Carriero, Sayan Mondal, Robert Abel, Craig E Masse

J Med Chem· August 2023

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Potent and selective TYK2-JH1 inhibitors highly efficacious in rodent model of psoriasis.
Silvana Leit, Jeremy R Greenwood, Sayan Mondal, Samantha Carriero, Markus Dahlgren, Craig E Masse

Bioorg Med Chem Lett· October 2022

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Preclinical evaluation of tyrosine kinase 2 inhibitors for human beta-cell protection in type 1 diabetes.
Alexandra Coomans de Brachène, Angela Castela, Anne Op de Beeck, Raghavendra G Mirmira, Lorella Marselli, Craig Masse

Diabetes Obes Metab· October 2020

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TYK2 inhibition reduces type 3 immunity and modifies disease progression in murine spondyloarthritis.
Eric Gracey, Dominika Hromadová, Melissa Lim, Zoya Qaiyum, Michael Zeng, Craig Masse

J Clin Invest· April 2020

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Accelerating drug discovery through tight integration of expert molecular design and predictive scoring.
Robert Abel, Sayan Mondal, Craig Masse, Jeremy Greenwood, Geraldine Harriman

Curr Opin Struct Biol· April 2017

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Anti-leukaemic activity of the TYK2 selective inhibitor NDI-031301 in T-cell acute lymphoblastic leukaemia.
Koshi Akahane, Zhaodong Li, Julia Etchin, Alla Berezovskaya, Evisa Gjini, Craig E Masse

Br J Haematol· April 2017

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X-ray crystal structures of Escherichia coli RNA polymerase with switch region binding inhibitors enable rational design of squaramides with an improved fraction unbound to human plasma protein.
Vadim Molodtsov, Paul R Fleming, Charles J Eyermann, Andrew D Ferguson, Melinda A Foulk, Craig E Masse

J Med Chem· April 2015

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Accurate and reliable prediction of relative ligand binding potency in prospective drug discovery by way of a modern free-energy calculation protocol and force field.
Lingle Wang, Yujie Wu, Yuqing Deng, Byungchan Kim, Levi Pierce, Craig Masse

J Am Chem Soc· February 2015

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A Potent and Orally Efficacious, Hydroxyethylamine-Based Inhibitor of β-Secretase.
Matthew R Kaller, Scott S Harried, Brian Albrecht, Patricia Amarante, Safura Babu-Khan, Craig Masse

ACS Med Chem Lett· November 2012

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Discovery of aminoquinazolines as potent, orally bioavailable inhibitors of Lck: synthesis, SAR, and in vivo anti-inflammatory activity.
Erin F DiMauro, John Newcomb, Joseph J Nunes, Jean E Bemis, Christina Boucher, Craig E Masse

J Med Chem· September 2006

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Divergent structural complexity from a linear reaction sequence: synthesis of fused and spirobicyclic gamma-lactams from common synthetic precursors.
Craig E Masse, Pui Yee Ng, Yoshiyuki Fukase, María Sanchez-Roselló, Jared T Shaw

J Comb Chem· August 2006

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Cycloaddition reactions of imines with 3-thiosuccinic anhydrides: synthesis of the tricyclic core of martinellic acid.
Pui Yee Ng, Craig E Masse, Jared T Shaw

Org Lett· August 2006

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C(2)-symmetric Sc(III)-complexes as chiral Lewis acids. Catalytic enantioselective aldol additions to glyoxylate esters.
David A Evans, Craig E Masse, Jimmy Wu

Org Lett· October 2002

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A general method for the enantioselective synthesis of pantolactone derivatives.
David A Evans, Jimmy Wu, Craig E Masse, David W C MacMillan

Org Lett· October 2002

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Total Synthesis of (+)-Mycotrienol and (+)-Mycotrienin I.
James S. Panek, Craig E. Masse

J Org Chem· November 1997

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