Publications by authors named "Douglas Gernert"

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Modulation of TARP 8-Containing AMPA Receptors as a Novel Therapeutic Approach for Chronic Pain.
Kelly L Knopp, Rosa Maria A Simmons, Wenhong Guo, Benjamin L Adams, Kevin M Gardinier, Douglas L Gernert

J Pharmacol Exp Ther· June 2019

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Targeted Blockade of TARP-γ8-Associated AMPA Receptors: Anticonvulsant Activity with the Selective Antagonist LY3130481 (CERC-611).
Jeffrey M Witkin, Douglas A Schober, Scott D Gleason, John T Catlow, Warren J Porter, Douglas L Gernert

CNS Neurol Disord Drug Targets· March 2019

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Structural Determinants of the γ-8 TARP Dependent AMPA Receptor Antagonist.
Matthew R Lee, Kevin M Gardinier, Douglas L Gernert, Douglas A Schober, Rebecca A Wright

ACS Chem Neurosci· December 2017

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Forebrain-selective AMPA-receptor antagonism guided by TARP γ-8 as an antiepileptic mechanism.
Akihiko S Kato, Kevin D Burris, Kevin M Gardinier, Douglas L Gernert, Warren J Porter

Nat Med· December 2016

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Discovery of the First α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor Antagonist Dependent upon Transmembrane AMPA Receptor Regulatory Protein (TARP) γ-8.
Kevin M Gardinier, Douglas L Gernert, Warren J Porter, Jon K Reel, Paul L Ornstein

J Med Chem· May 2016

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Discovery of a potent, dual serotonin and norepinephrine reuptake inhibitor.
Nicolas Dreyfus, Jason K Myers, Valentina O Badescu, Oscar de Frutos, Maria Luz de la Puente, Douglas L Gernert

ACS Med Chem Lett· June 2013

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Transmembrane AMPA receptor regulatory proteins and cornichon-2 allosterically regulate AMPA receptor antagonists and potentiators.
Douglas A Schober, Martin B Gill, Hong Yu, Douglas L Gernert, Matthew W Jeffries

J Biol Chem· April 2011

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(S)-N-{3-[1-cyclopropyl-1-(2,4-difluoro-phenyl)-ethyl]-1H-indol-7-yl}-methanesulfonamide: a potent, nonsteroidal, functional antagonist of the mineralocorticoid receptor.
Michael G Bell, Douglas L Gernert, Timothy A Grese, Matthew D Belvo, Peter S Borromeo

J Med Chem· December 2007

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Design and synthesis of piperidine farnesyltransferase inhibitors with reduced glucuronidation potential.
Rieko Tanaka, Almudena Rubio, Nancy K Harn, Douglas Gernert, Timothy A Grese

Bioorg Med Chem· February 2007

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