Publications by authors named "Eric Valeur"

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Glucagon Like Peptide 1 Receptor Agonists for Targeted Delivery of Antisense Oligonucleotides to Pancreatic Beta Cell.
Laurent Knerr, Thazha P Prakash, Richard Lee, William J Drury Iii, Mehran Nikan, Eric Valeur

J Am Chem Soc· March 2021

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A protein tertiary structure mimetic modulator of the Hippo signalling pathway.
Hélène Adihou, Ranganath Gopalakrishnan, Tim Förster, Stéphanie M Guéret, Raphael Gasper, Eric Valeur

Nat Commun· October 2020

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Discovery of 4-((2,4)-4-Ethoxy-1-((5-methoxy-7-methyl-1-indol-4-yl)methyl)piperidin-2-yl)benzoic Acid (LNP023), a Factor B Inhibitor Specifically Designed To Be Applicable to Treating a Diverse Array of Complement Mediated Diseases.
Nello Mainolfi, Takeru Ehara, Rajeshri G Karki, Karen Anderson, Aengus Mac Sweeney, Eric Valeur

J Med Chem· June 2020

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Macrocyclic Modalities Combining Peptide Epitopes and Natural Product Fragments.
Stéphanie M Guéret, Sasikala Thavam, Rodrigo J Carbajo, Marco Potowski, Niklas Larsson, Eric Valeur

J Am Chem Soc· March 2020

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Late-Stage Functionalization of Histidine in Unprotected Peptides.
Anaïs F M Noisier, Magnus J Johansson, Laurent Knerr, Martin A Hayes, William J Drury, Eric Valeur

Angew Chem Int Ed Engl· December 2019

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Emerging modes-of-action in drug discovery.
Eric Valeur, Frank Narjes, Christian Ottmann, Alleyn T Plowright

Medchemcomm· September 2019

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Small-molecule factor B inhibitor for the treatment of complement-mediated diseases.
Anna Schubart, Karen Anderson, Nello Mainolfi, Holger Sellner, Takeru Ehara, Eric Valeur

Proc Natl Acad Sci U S A· April 2019

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New Modalities, Technologies, and Partnerships in Probe and Lead Generation: Enabling a Mode-of-Action Centric Paradigm.
Eric Valeur, Patrick Jimonet

J Med Chem· October 2018

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Inhibition of low-density lipoprotein receptor degradation with a cyclic peptide that disrupts the homodimerization of IDOL E3 ubiquitin ligase.
Eilidh K Leitch, Nagarajan Elumalai, Maria Fridén-Saxin, Göran Dahl, Paul Wan, Eric Valeur

Chem Sci· July 2018

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Structure-based design and synthesis of macrocyclic human rhinovirus 3C protease inhibitors.
Kenji Namoto, Finton Sirockin, Holger Sellner, Christian Wiesmann, Frederic Villard, Eric Valeur

Bioorg Med Chem Lett· March 2018

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Directing evolution: the next revolution in drug discovery?
Andrew M Davis, Alleyn T Plowright, Eric Valeur

Nat Rev Drug Discov· October 2017

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New Modalities for Challenging Targets in Drug Discovery.
Eric Valeur, Stéphanie M Guéret, Hélène Adihou, Ranganath Gopalakrishnan, Malin Lemurell

Angew Chem Int Ed Engl· August 2017

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Targeted delivery for regenerative medicines: an untapped opportunity for drug conjugates.
Eric Valeur, Laurent Knerr, Maria Ölwegård-Halvarsson, Malin Lemurell

Drug Discov Today· June 2017

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Therapeutic Potential of Foldamers: From Chemical Biology Tools To Drug Candidates?
Ranganath Gopalakrishnan, Andrey I Frolov, Laurent Knerr, William J Drury, Eric Valeur

J Med Chem· November 2016

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Structure-based design of 7-azaindole-pyrrolidine amides as inhibitors of 11β-hydroxysteroid dehydrogenase type I.
Eric Valeur, Serge Christmann-Franck, Franck Lepifre, Denis Carniato, Daniel Cravo

Bioorg Med Chem Lett· September 2012

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Isoindolinone inhibitors of the murine double minute 2 (MDM2)-p53 protein-protein interaction: structure-activity studies leading to improved potency.
Ian R Hardcastle, Junfeng Liu, Eric Valeur, Anna Watson, Shafiq U Ahmed

J Med Chem· March 2011

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Discovery and structure-guided drug design of inhibitors of 11beta-hydroxysteroid-dehydrogenase type I based on a spiro-carboxamide scaffold.
Franck Lepifre, Serge Christmann-Franck, Didier Roche, Caroline Leriche, Denis Carniato, Eric Valeur

Bioorg Med Chem Lett· July 2009

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Discovery and structure-activity relationships of pentanedioic acid diamides as potent inhibitors of 11beta-hydroxysteroid dehydrogenase type I.
Didier Roche, Denis Carniato, Caroline Leriche, Franck Lepifre, Serge Christmann-Franck, Eric Valeur

Bioorg Med Chem Lett· May 2009

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Amide bond formation: beyond the myth of coupling reagents.
Eric Valeur, Mark Bradley

Chem Soc Rev· February 2009

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Analysis of chemical shift changes reveals the binding modes of isoindolinone inhibitors of the MDM2-p53 interaction.
Christiane Riedinger, Jane A Endicott, Stuart J Kemp, Lynette A Smyth, Anna Watson, Eric Valeur

J Am Chem Soc· November 2008

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PS-IIDQ: an efficient polymer-supported amide coupling reagent.
Eric Valeur, Mark Bradley

Chem Commun (Camb)· March 2005

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