Publications by authors named "Fa-Xiang Ding"

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Structure Guided Discovery of Novel Pan Metallo-β-Lactamase Inhibitors with Improved Gram-Negative Bacterial Cell Penetration.
Shuzhi Dong, Zhiqiang Zhao, Haiqun Tang, Guoqing Li, Jianping Pan, Fa-Xiang Ding

J Med Chem· March 2024

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Orally Bioavailable Macrocyclic Peptide That Inhibits Binding of PCSK9 to the Low Density Lipoprotein Receptor.
Douglas G Johns, Louis-Charles Campeau, Puja Banka, An Bautmans, Tjerk Bueters, Fa-Xiang Ding

Circulation· July 2023

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Discovery of MK-8153, a Potent and Selective ROMK Inhibitor and Novel Diuretic/Natriuretic.
Jinlong Jiang, Fa-Xiang Ding, Xiaoyan Zhou, Thomas J Bateman, Shuzhi Dong

J Med Chem· June 2021

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Discovery of a potent and selective ROMK inhibitor with improved pharmacokinetic properties based on an octahydropyrazino[2,1-c][1,4]oxazine scaffold.
Yuping Zhu, Reynalda K de Jesus, Haifeng Tang, Shawn P Walsh, Jinlong Jiang, Fa-Xiang Ding

Bioorg Med Chem Lett· December 2016

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Guided reconstitution of membrane protein fragments.
Leah S Cohen, Boris Arshava, Sarah Kauffman, Elizabeth Mathew, Katrina E Fracchiolla, Fa-Xiang Ding

Biopolymers· January 2014

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NMR mapping of RANTES surfaces interacting with CCR5 using linked extracellular domains.
Einat Schnur, Naama Kessler, Yuri Zherdev, Eran Noah, Tali Scherf, Fa-Xiang Ding

FEBS J· May 2013

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Synergism between a CD4-mimic peptide and antibodies elicited by a constrained V3 peptide.
Adi Moseri, Subramanyam Tantry, Fa-Xiang Ding, Fred Naider, Jacob Anglister

AIDS Res Hum Retroviruses· April 2013

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Functional fusions of T4 lysozyme in the third intracellular loop of a G protein-coupled receptor identified by a random screening approach in yeast.
Elizabeth Mathew, Fa-Xiang Ding, Fred Naider, Mark E Dumont

Protein Eng Des Sel· January 2013

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Discovery of benzodihydroisofurans as novel, potent, bioavailable and brain-penetrant prolylcarboxypeptidase inhibitors.
Hong C Shen, Fa-Xiang Ding, Jinlong Jiang, Andreas Verras, Renee M Chabin

Bioorg Med Chem Lett· February 2012

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The conformation and orientation of a 27-residue CCR5 peptide in a ternary complex with HIV-1 gp120 and a CD4-mimic peptide.
Einat Schnur, Eran Noah, Inbal Ayzenshtat, Hasmik Sargsyan, Tatsuya Inui, Fa-Xiang Ding

J Mol Biol· July 2011

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Differential interactions of fluorescent agonists and antagonists with the yeast G protein coupled receptor Ste2p.
Elizabeth Mathew, Anshika Bajaj, Sara M Connelly, Hasmik Sargsyan, Fa-Xiang Ding

J Mol Biol· June 2011

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Discovery of benzimidazole pyrrolidinyl amides as prolylcarboxypeptidase inhibitors.
Hong C Shen, Fa-Xiang Ding, Changyou Zhou, Yusheng Xiong, Andreas Verras

Bioorg Med Chem Lett· March 2011

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Identification of residue-to-residue contact between a peptide ligand and its G protein-coupled receptor using periodate-mediated dihydroxyphenylalanine cross-linking and mass spectrometry.
George K E Umanah, Liyin Huang, Fa-xiang Ding, Boris Arshava, Adam R Farley

J Biol Chem· December 2010

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Design of potent IGF1-R inhibitors related to bis-azaindoles.
Conception Nemecek, William A Metz, Sylvie Wentzler, Fa-Xiang Ding, Corinne Venot

Chem Biol Drug Des· August 2010

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Binding of fluorinated phenylalanine alpha-factor analogues to Ste2p: evidence for a cation-pi binding interaction between a peptide ligand and its cognate G protein-coupled receptor.
Subramanyam Tantry, Fa-Xiang Ding, Mark Dumont, Jeffrey M Becker, Fred Naider

Biochemistry· June 2010

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Anthranilic acid replacements in a niacin receptor agonist.
Darby Schmidt, Abigail Smenton, Subharekha Raghavan, Hong Shen, Fa-Xiang Ding

Bioorg Med Chem Lett· June 2010

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Discovery of pyrazolyl propionyl cyclohexenamide derivatives as full agonists for the high affinity niacin receptor GPR109A.
Fa-Xiang Ding, Hong C Shen, Larrisa C Wilsie, Mihajlo L Krsmanovic, Andrew K Taggart

Bioorg Med Chem Lett· June 2010

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Discovery of a biaryl cyclohexene carboxylic acid (MK-6892): a potent and selective high affinity niacin receptor full agonist with reduced flushing profiles in animals as a preclinical candidate.
Hong C Shen, Fa-Xiang Ding, Subharekha Raghavan, Qiaolin Deng, Silvi Luell

J Med Chem· March 2010

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A strategy of employing aminoheterocycles as amide mimics to identify novel, potent and bioavailable soluble epoxide hydrolase inhibitors.
Hong C Shen, Fa-Xiang Ding, Qiaolin Deng, Suoyu Xu, Xinchun Tong

Bioorg Med Chem Lett· October 2009

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Discovery of 3,3-disubstituted piperidine-derived trisubstituted ureas as highly potent soluble epoxide hydrolase inhibitors.
Hong C Shen, Fa-Xiang Ding, Qiaolin Deng, Suoyu Xu, Hsuan-Shen Chen

Bioorg Med Chem Lett· September 2009

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HIV-1 peptide vaccine candidates: selecting constrained V3 peptides with highest affinity to antibody 447-52D.
Brenda Mester, Revital Manor, Amit Mor, Boris Arshava, Osnat Rosen, Fa-Xiang Ding

Biochemistry· August 2009

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Discovery of a highly potent, selective, and bioavailable soluble epoxide hydrolase inhibitor with excellent ex vivo target engagement.
Hong C Shen, Fa-Xiang Ding, Siyi Wang, Qiaolin Deng, Xiaoping Zhang

J Med Chem· August 2009

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Discovery of spirocyclic secondary amine-derived tertiary ureas as highly potent, selective and bioavailable soluble epoxide hydrolase inhibitors.
Hong C Shen, Fa-Xiang Ding, Siyi Wang, Suoyu Xu, Hsuan-shen Chen

Bioorg Med Chem Lett· July 2009

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Mimicking the structure of the V3 epitope bound to HIV-1 neutralizing antibodies.
Amit Mor, Eugenia Segal, Brenda Mester, Boris Arshava, Osnat Rosen, Fa-Xiang Ding

Biochemistry· April 2009

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Discovery of novel tricyclic full agonists for the G-protein-coupled niacin receptor 109A with minimized flushing in rats.
Hong C Shen, Fa-Xiang Ding, Qiaolin Deng, Larissa C Wilsie, Mihajlo L Krsmanovic

J Med Chem· April 2009

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