Publications by authors named "Gail Mattson"

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Oxazolidinone-based allosteric modulators of mGluR5: Defining molecular switches to create a pharmacological tool box.
Hong Huang, Andrew P Degnan, Anand Balakrishnan, Amy Easton, Michael Gulianello, Gail Mattson

Bioorg Med Chem Lett· September 2016

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Synthesis and evaluation of carbamate and aryl ether substituted pyrazinones as corticotropin releasing factor-1 (CRF₁) receptor antagonists.
Vijay T Ahuja, Richard A Hartz, Thaddeus F Molski, Gail K Mattson, Kimberley A Lentz

Bioorg Med Chem Lett· May 2016

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Discovery and Preclinical Evaluation of BMS-955829, a Potent Positive Allosteric Modulator of mGluR5.
Fukang Yang, Lawrence B Snyder, Anand Balakrishnan, Jeffrey M Brown, Digavalli V Sivarao, Gail Mattson

ACS Med Chem Lett· March 2016

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Biaryls as potent, tunable dual neurokinin 1 receptor antagonists and serotonin transporter inhibitors.
Andrew P Degnan, George O Tora, Ying Han, Ramkumar Rajamani, Robert Bertekap, Gail Mattson

Bioorg Med Chem Lett· August 2015

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Heterocyclic modification of a novel bicyclo[3.1.0]hexane NPY1 receptor antagonist.
Guanglin Luo, Ling Chen, Shuanghua Hu, Yazhong Huang, Gail Mattson

Bioorg Med Chem Lett· July 2013

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Conformationally restricted homotryptamines. Part 6: indole-5-cycloalkyl methylamines as selective serotonin reuptake inhibitors.
Jonathan L Ditta, Derek J Denhart, Jeffrey A Deskus, James R Epperson, Zhaoxing Meng, Gail K Mattson, Ronald J Mattson

Bioorg Med Chem Lett· May 2013

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Potential CRF1R PET imaging agents: 1-fluoroalkylsubstituted 5-halo-3-(arylamino)pyrazin-2(1H)-ones.
Derek J Denhart, Dmitry Zuev, Jonathan L Ditta, Richard A Hartz, Vijay T Ahuja, Ronald J Mattson, Gail K Mattson

Bioorg Med Chem Lett· April 2013

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[18F](R)-5-chloro-1-(1-cyclopropyl-2-methoxyethyl)-3-(4-(2-fluoroethoxy)-2,5-dimethyl phenylamino)pyrazin-2(1H)-one: introduction of N3-phenylpyrazinones as potential CRF-R1 PET imaging agents.
Jeffrey A Deskus, Douglas D Dischino, Ronald J Mattson, Jonathan L Ditta, Michael F Parker, Gail K Mattson

Bioorg Med Chem Lett· November 2012

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Discovery of a Novel Class of Bicyclo[3.1.0]hexanylpiperazines as Noncompetitive Neuropeptide Y Y1 Antagonists.
Shuanghua Hu, Yazhong Huang, Milind Deshpande, Guanglin Luo, Marc A Bruce, Gail Mattson

ACS Med Chem Lett· March 2012

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Potential CRF1R PET imaging agents: N-fluoroalkyl-8-(6-methoxy-2-methylpyridin-3-yl)-2,7-dimethyl-N-alkylpyrazolo[1,5-a][1,3,5]triazin-4-amines.
Dmitry Zuev, Ronald J Mattson, Hong Huang, Gail K Mattson, Larisa Zueva

Bioorg Med Chem Lett· April 2011

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Conformationally restricted homotryptamines. Part 7: 3-cis-(3-aminocyclopentyl)indoles as potent selective serotonin reuptake inhibitors.
H Dalton King, Zhaoxing Meng, Jeffrey A Deskus, Charles P Sloan, Qi Gao, Gail K Mattson, Ronald J Mattson

J Med Chem· November 2010

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Synthesis and structure-activity relationships of N3-pyridylpyrazinones as corticotropin-releasing factor-1 (CRF1) receptor antagonists.
Richard A Hartz, Vijay T Ahuja, William D Schmitz, Thaddeus F Molski, Gail K Mattson

Bioorg Med Chem Lett· March 2010

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Synthesis and hSERT activity of homotryptamine analogs. Part 6: [3+2] dipolar cycloaddition of 3-vinylindoles.
Lawrence R Marcin, Ronald J Mattson, Qi Gao, Dedong Wu, Thaddeus F Molski, Gail K Mattson

Bioorg Med Chem Lett· February 2010

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Conformationally restricted homotryptamines. Part 5: 3-(trans-2-aminomethylcyclopentyl)indoles as potent selective serotonin reuptake inhibitors.
Derek J Denhart, Jeffrey A Deskus, Jonathan L Ditta, Qi Gao, H Dalton King, Gail K Mattson, Ronald J Mattson

Bioorg Med Chem Lett· August 2009

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Synthesis, structure-activity relationships, and in vivo evaluation of N3-phenylpyrazinones as novel corticotropin-releasing factor-1 (CRF1) receptor antagonists.
Richard A Hartz, Vijay T Ahuja, Argyrios G Arvanitis, Maria Rafalski, Eddy W Yue, Gail K Mattson, Ronald J Mattson

J Med Chem· July 2009

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Pharmacological characterization and appetite suppressive properties of BMS-193885, a novel and selective neuropeptide Y(1) receptor antagonist.
Ildiko Antal-Zimanyi, Marc A Bruce, Karen L Leboulluec, Lawrence G Iben, Gail K Mattson

Eur J Pharmacol· August 2008

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Ex vivo assessment of binding site occupancy of monoamine reuptake inhibitors: methodology and biological significance.
Kelly Lengyel, Rick Pieschl, Todd Strong, Thaddeus Molski, Gail Mattson

Neuropharmacology· July 2008

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Conformationally restricted homotryptamines. Part 4: Heterocyclic and naphthyl analogs of a potent selective serotonin reuptake inhibitor.
H Dalton King, Derek J Denhart, Jeffrey A Deskus, Jonathan L Ditta, James R Epperson, Gail K Mattson, Ronald J Mattson

Bioorg Med Chem Lett· October 2007

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Conformationally restricted homotryptamines 3. Indole tetrahydropyridines and cyclohexenylamines as selective serotonin reuptake inhibitors.
Jeffrey A Deskus, James R Epperson, Charles P Sloan, Joseph A Cipollina, Pierre Dextraze, Gail K Mattson, Ronald J Mattson

Bioorg Med Chem Lett· June 2007

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Synthesis and evaluation of 5,5-diphenylimidazolones as potent human neuropeptide Y5 receptor antagonists.
Kevin W Gillman, Mendi A Higgins, Graham S Poindexter, Marc Browning, Wendy J Clarke, Gail K Mattson

Bioorg Med Chem· August 2006

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Conformationally restricted homotryptamines. 2. Indole cyclopropylmethylamines as selective serotonin reuptake inhibitors.
Ronald J Mattson, John D Catt, Derek J Denhart, Jeffrey A Deskus, Jonathan L Ditta, Gail K Mattson

J Med Chem· September 2005

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Homotryptamines as potent and selective serotonin reuptake inhibitors (SSRIs).
William D Schmitz, Derek J Denhart, Allison B Brenner, Jonathan L Ditta, Ronald J Mattson, Gail K Mattson

Bioorg Med Chem Lett· March 2005

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Isosteric N-arylpiperazine replacements in a series of dihydropyridine NPY1 receptor antagonists.
Guanglin Luo, Gail K Mattson, Marc A Bruce, Henry Wong, Brian J Murphy

Bioorg Med Chem Lett· December 2004

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Application of solution-phase parallel synthesis to preparation of trisubstituted 1,2,4-triazoles.
Scott W Martin, Jeffrey L Romine, Ling Chen, Gail Mattson, Ildiko A Antal-Zimanyi

J Comb Chem· June 2004

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beta-alanine dipeptides as MC4R agonists.
Réjean Ruel, Timothy F Herpin, Lawrence Iben, Guanglin Luo, Alain Martel, Gail Mattson

Bioorg Med Chem Lett· December 2003

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