Publications by authors named "Giorgio Pochetti"

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Cytosolic localization and in vitro assembly of human de novo thymidylate synthesis complex.
Sharon Spizzichino, Dalila Boi, Giovanna Boumis, Roberta Lucchi, Francesca Romana Liberati, Giorgio Pochetti

FEBS J· March 2022

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PHA-680626 Is an Effective Inhibitor of the Interaction between Aurora-A and N-Myc.
Dalila Boi, Fani Souvalidou, Davide Capelli, Federica Polverino, Grazia Marini, Giorgio Pochetti

Int J Mol Sci· December 2021

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Discovery of Novel Chemical Series of OXA-48 β-Lactamase Inhibitors by High-Throughput Screening.
Barbara Garofalo, Federica Prati, Rosa Buonfiglio, Isabella Coletta, Noemi D'Atanasio, Giorgio Pochetti

Pharmaceuticals (Basel)· June 2021

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A Novel N-Substituted Valine Derivative with Unique Peroxisome Proliferator-Activated Receptor γ Binding Properties and Biological Activities.
Franck Peiretti, Roberta Montanari, Davide Capelli, Bernadette Bonardo, Cécilia Colson, Giorgio Pochetti

J Med Chem· November 2020

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Bone-Seeking Matrix Metalloproteinase Inhibitors for the Treatment of Skeletal Malignancy.
Antonio Laghezza, Luca Piemontese, Leonardo Brunetti, Alessia Caradonna, Mariangela Agamennone, Giorgio Pochetti

Pharmaceuticals (Basel)· June 2020

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Insights into PPARγ Phosphorylation and Its Inhibition Mechanism.
Roberta Montanari, Davide Capelli, Keiko Yamamoto, Hirono Awaishima, Kimina Nishikata, Giorgio Pochetti

J Med Chem· May 2020

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Surface Plasmon Resonance as a Tool for Ligand Binding Investigation of Engineered GPR17 Receptor, a G Protein Coupled Receptor Involved in Myelination.
Davide Capelli, Chiara Parravicini, Giorgio Pochetti, Roberta Montanari, Caterina Temporini

Front Chem· January 2020

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Identification of the First PPARα/γ Dual Agonist Able To Bind to Canonical and Alternative Sites of PPARγ and To Inhibit Its Cdk5-Mediated Phosphorylation.
Antonio Laghezza, Luca Piemontese, Carmen Cerchia, Roberta Montanari, Davide Capelli, Giorgio Pochetti

J Med Chem· September 2018

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Affinity-based separation methods for the study of biological interactions: The case of peroxisome proliferator-activated receptors in drug discovery.
Caterina Temporini, Gloria Brusotti, Giorgio Pochetti, Gabriella Massolini, Enrica Calleri

Methods· August 2018

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Betulinic acid is a PPARγ antagonist that improves glucose uptake, promotes osteogenesis and inhibits adipogenesis.
Gloria Brusotti, Roberta Montanari, Davide Capelli, Giulia Cattaneo, Antonio Laghezza, Giorgio Pochetti

Sci Rep· July 2017

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Catechol-based matrix metalloproteinase inhibitors with additional antioxidative activity.
Marilena Tauro, Antonio Laghezza, Fulvio Loiodice, Luca Piemontese, Alessia Caradonna, Giorgio Pochetti

J Enzyme Inhib Med Chem· February 2017

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Structural basis for PPAR partial or full activation revealed by a novel ligand binding mode.
Davide Capelli, Carmen Cerchia, Roberta Montanari, Fulvio Loiodice, Paolo Tortorella, Giorgio Pochetti

Sci Rep· October 2016

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Screening of saponins and sapogenins from Medicago species as potential PPARγ agonists and X-ray structure of the complex PPARγ/caulophyllogenin.
Roberta Montanari, Davide Capelli, Aldo Tava, Andrea Galli, Antonio Laghezza, Giorgio Pochetti

Sci Rep· June 2016

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On the metabolically active form of metaglidasen: improved synthesis and investigation of its peculiar activity on peroxisome proliferator-activated receptors and skeletal muscles.
Antonio Laghezza, Roberta Montanari, Antonio Lavecchia, Luca Piemontese, Giorgio Pochetti

ChemMedChem· March 2015

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Structural basis of the transactivation deficiency of the human PPARγ F360L mutant associated with familial partial lipodystrophy.
Clorinda Lori, Alessandra Pasquo, Roberta Montanari, Davide Capelli, Valerio Consalvi, Giorgio Pochetti

Acta Crystallogr D Biol Crystallogr· July 2014

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LT175 is a novel PPARα/γ ligand with potent insulin-sensitizing effects and reduced adipogenic properties.
Federica Gilardi, Marco Giudici, Nico Mitro, Omar Maschi, Uliano Guerrini, Giorgio Pochetti

J Biol Chem· March 2014

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Design and biophysical characterization of atrazine-sensing peptides mimicking the Chlamydomonas reinhardtii plastoquinone binding niche.
Viviana Scognamiglio, Pasquale Stano, Fabio Polticelli, Amina Antonacci, Maya Dimova Lambreva, Giorgio Pochetti

Phys Chem Chem Phys· August 2013

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Synthesis, biological evaluation and molecular investigation of fluorinated peroxisome proliferator-activated receptors α/γ dual agonists.
Giuseppe Fracchiolla, Antonio Laghezza, Luca Piemontese, Mariagiovanna Parente, Antonio Lavecchia, Giorgio Pochetti

Bioorg Med Chem· March 2012

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Structural insight into peroxisome proliferator-activated receptor gamma binding of two ureidofibrate-like enantiomers by molecular dynamics, cofactor interaction analysis, and site-directed mutagenesis.
Giorgio Pochetti, Nico Mitro, Antonio Lavecchia, Federica Gilardi, Neva Besker

J Med Chem· June 2010

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New 2-aryloxy-3-phenyl-propanoic acids as peroxisome proliferator-activated receptors alpha/gamma dual agonists with improved potency and reduced adverse effects on skeletal muscle function.
Giuseppe Fracchiolla, Antonio Laghezza, Luca Piemontese, Paolo Tortorella, Fernando Mazza, Giorgio Pochetti

J Med Chem· October 2009

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Extra binding region induced by non-zinc chelating inhibitors into the S1' subsite of matrix metalloproteinase 8 (MMP-8).
Giorgio Pochetti, Roberta Montanari, Christian Gege, Carine Chevrier, Arthur G Taveras

J Med Chem· February 2009

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Crystal structure of the peroxisome proliferator-activated receptor gamma (PPARgamma) ligand binding domain complexed with a novel partial agonist: a new region of the hydrophobic pocket could be exploited for drug design.
Roberta Montanari, Fulvio Saccoccia, Elena Scotti, Maurizio Crestani, Cristina Godio, Giorgio Pochetti

J Med Chem· December 2008

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Insights into the mechanism of partial agonism: crystal structures of the peroxisome proliferator-activated receptor gamma ligand-binding domain in the complex with two enantiomeric ligands.
Giorgio Pochetti, Cristina Godio, Nico Mitro, Donatella Caruso, Andrea Galmozzi

J Biol Chem· June 2007

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Stereoselectivity by enantiomeric inhibitors of matrix metalloproteinase-8: new insights from molecular dynamics simulations.
Massimiliano Aschi, Neva Besker, Nazzareno Re, Giorgio Pochetti, Cecilia Coletti

J Med Chem· January 2007

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Structural insight into the stereoselective inhibition of MMP-8 by enantiomeric sulfonamide phosphonates.
Giorgio Pochetti, Enrico Gavuzzo, Cristina Campestre, Mariangela Agamennone, Paolo Tortorella

J Med Chem· February 2006

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