Publications by authors named "Giuseppe Meroni"

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Structure-based design of potent and selective inhibitors of the HECT ligase NEDD4.
Elena Maspero, Anna Cappa, Janine Weber, Paolo Trifirò, Raffaella Amici, Giuseppe Meroni

Commun Chem· May 2025

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A multiparametric screen uncovers FDA-approved small molecules that potentiate the nuclear mechano-dysfunctions in ATR-defective cells.
Maria Rosaria Cera, Giulia Bastianello, Divya Purushothaman, Adrian Andronache, Flora Ascione, Giuseppe Meroni

Sci Rep· December 2024

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Inhibition of the lysine demethylase LSD1 modulates the balance between inflammatory and antiviral responses against coronaviruses.
Luca Mazzarella, Fabio Santoro, Roberto Ravasio, Valeria Fumagalli, Paul E Massa, Giuseppe Meroni

Sci Signal· December 2023

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Tuning mTORC1 activity dictates the response of acute myeloid leukemia to LSD1 inhibition.
Amal Kamal Abdel-Aziz, Isabella Pallavicini, Elena Ceccacci, Giuseppe Meroni, Mona Kamal Saadeldin

Haematologica· August 2020

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Novel potent inhibitors of the histone demethylase KDM1A (LSD1), orally active in a murine promyelocitic leukemia model.
Paolo Trifirò, Anna Cappa, Silvia Brambillasca, Oronza A Botrugno, Maria Rosaria Cera, Giuseppe Meroni

Future Med Chem· July 2017

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Thieno[3,2-b]pyrrole-5-carboxamides as New Reversible Inhibitors of Histone Lysine Demethylase KDM1A/LSD1. Part 1: High-Throughput Screening and Preliminary Exploration.
Luca Sartori, Ciro Mercurio, Federica Amigoni, Anna Cappa, Giovanni Fagá, Giuseppe Meroni

J Med Chem· March 2017

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Thieno[3,2-b]pyrrole-5-carboxamides as New Reversible Inhibitors of Histone Lysine Demethylase KDM1A/LSD1. Part 2: Structure-Based Drug Design and Structure-Activity Relationship.
Paola Vianello, Luca Sartori, Federica Amigoni, Anna Cappa, Giovanni Fagá, Giuseppe Meroni

J Med Chem· March 2017

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Discovery of a Novel Inhibitor of Histone Lysine-Specific Demethylase 1A (KDM1A/LSD1) as Orally Active Antitumor Agent.
Paola Vianello, Oronza A Botrugno, Anna Cappa, Roberto Dal Zuffo, Paola Dessanti, Giuseppe Meroni

J Med Chem· February 2016

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Further insights into the SAR of α-substituted cyclopropylamine derivatives as inhibitors of histone demethylase KDM1A.
Marco Pieroni, Giannamaria Annunziato, Elisa Azzali, Paola Dessanti, Ciro Mercurio, Giuseppe Meroni

Eur J Med Chem· March 2015

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Synthesis, biological activity and mechanistic insights of 1-substituted cyclopropylamine derivatives: a novel class of irreversible inhibitors of histone demethylase KDM1A.
Paola Vianello, Oronza A Botrugno, Anna Cappa, Giuseppe Ciossani, Paola Dessanti, Giuseppe Meroni

Eur J Med Chem· October 2014

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Measurement of S-methylcysteine and S-methyl-mercapturic acid in human urine by alkyl-chloroformate extractive derivatization and isotope-dilution gas chromatography-mass spectrometry.
Federico M Rubino, Marco Pitton, Daniela Di Fabio, Giuseppe Meroni, Enzo Santaniello

Biomed Chromatogr· March 2011

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Enhanced activity or resistance of adenosine derivatives towards adenosine deaminase-catalyzed deamination: Influence of ribose modifications.
Giulio Vistoli, Alessandro Pedretti, Laura Alessandrini, Silvana Casati, Pierangela Ciuffreda, Giuseppe Meroni

Bioorg Med Chem Lett· May 2009

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Synthesis of enantiopure Delta2-isoxazoline derivatives and evaluation of their affinity and efficacy profiles at human beta-adrenergic receptor subtypes.
Clelia Dallanoce, Giuseppe Meroni, Marco De Amici, Carsten Hoffmann, Karl-Norbert Klotz

Bioorg Med Chem· July 2006

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