Publications by authors named "Gregory A Gfesser"

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Discovery of Orally Efficacious Bridged Piperazines as smTNF Modulators.
Zhiguo Bian, Robert G Schmidt, Noel S Wilson, David B Duignan, Eric Breinlinger, Gregory A Gfesser

J Med Chem· July 2025

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Discovery and SAR of 4-aminopyrrolidine-2-carboxylic acid correctors of CFTR for the treatment of cystic fibrosis.
Marc J C Scanio, Xenia B Searle, Bo Liu, John R Koenig, Robert J Altenbach, Gregory A Gfesser

Bioorg Med Chem Lett· September 2022

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Lithioarene Cycliacylation and Pd-Catalyzed Aminoethylation/Cyclization to Access Electronically Diverse Saturated Isoquinoline Derivatives.
Marek Buchman, Elliot P Farney, Stephen N Greszler, Robert J Altenbach, Gregory A Gfesser

J Org Chem· January 2022

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Discovery of ABBV/GLPG-3221, a Potent Corrector of CFTR for the Treatment of Cystic Fibrosis.
Marc J C Scanio, Xenia B Searle, Bo Liu, John R Koenig, Robert Altenbach, Gregory A Gfesser

ACS Med Chem Lett· November 2019

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Synthesis and Pharmacology of (Pyridin-2-yl)methanol Derivatives as Novel and Selective Transient Receptor Potential Vanilloid 3 Antagonists.
Arthur Gomtsyan, Robert G Schmidt, Erol K Bayburt, Gregory A Gfesser, Eric A Voight

J Med Chem· May 2016

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Discovery of 4-(5-(4-chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744) as a novel positive allosteric modulator of the alpha7 nicotinic acetylcholine receptor.
Ramin Faghih, Sujatha M Gopalakrishnan, Jens Halvard Gronlien, John Malysz, Clark A Briggs, Gregory A Gfesser

J Med Chem· May 2009

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Advances in the discovery of novel positive allosteric modulators of the alpha7 nicotinic acetylcholine receptor.
Ramin Faghih, Gregory A Gfesser, Murali Gopalakrishnan

Recent Pat CNS Drug Discov· June 2007

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Novel heterocyclic-substituted benzofuran histamine H3 receptor antagonists: in vitro properties, drug-likeness, and behavioral activity.
Marlon Cowart, Gregory A Gfesser, Kaitlin E Browman, Ramin Faghih, Thomas R Miller

Biochem Pharmacol· April 2007

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Synthesis and SAR of 5-amino- and 5-(aminomethyl)benzofuran histamine H3 receptor antagonists with improved potency.
Minghua Sun, Chen Zhao, Gregory A Gfesser, Christine Thiffault, Thomas R Miller

J Med Chem· October 2005

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5-(3-Bromophenyl)-7-(6-morpholin-4-ylpyridin-3-yl)pyrido[2,3-d]pyrimidin-4-ylamine: structure-activity relationships of 7-substituted heteroaryl analogs as non-nucleoside adenosine kinase inhibitors.
Mark A Matulenko, Chih-Hung Lee, Meiqun Jiang, Robin R Frey, Marlon D Cowart, Gregory A Gfesser

Bioorg Med Chem· June 2005

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Structure-activity relationships of arylbenzofuran H3 receptor antagonists.
Gregory A Gfesser, Ramin Faghih, Youssef L Bennani, Michael P Curtis, Timothy A Esbenshade

Bioorg Med Chem Lett· May 2005

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4-(2-[2-(2(R)-methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl)benzonitrile and related 2-aminoethylbenzofuran H3 receptor antagonists potently enhance cognition and attention.
Marlon Cowart, Ramin Faghih, Michael P Curtis, Gregory A Gfesser, Youssef L Bennani

J Med Chem· January 2005

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Structure-activity relationships of non-imidazole H(3) receptor ligands. Part 3: 5-Substituted 3-phenyl-1,2,4-oxadiazoles as potent antagonists.
Gregory A Gfesser, Henry Zhang, Jurgen Dinges, Gerard B Fox, Jia Bao Pan

Bioorg Med Chem Lett· February 2004

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Adenosine kinase inhibitors: polar 7-substitutent of pyridopyrimidine derivatives improving their locomotor selectivity.
Guo Zhu Zheng, Yue Mao, Chih-Hung Lee, John K Pratt, John R Koenig, Gregory A Gfesser

Bioorg Med Chem Lett· September 2003

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Synthesis and structure-activity relationships of 5-heteroatom-substituted pyridopyrimidines as adenosine kinase inhibitors.
Gregory A Gfesser, Erol K Bayburt, Marlon Cowart, Stanley DiDomenico, Arthur Gomtsyan

Eur J Med Chem· March 2003

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