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Publications by authors named "Harry Brielmann"

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Discovery of novel 6,6-heterocycles as transient receptor potential vanilloid (TRPV1) antagonists.
Charles A Blum, Timothy Caldwell, Xiaozhang Zheng, Rajagopal Bakthavatchalam, Scott Capitosti, Harry Brielmann

J Med Chem· April 2010


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Aminoquinazolines as TRPV1 antagonists: modulation of drug-like properties through the exploration of 2-position substitution.
Charles A Blum, Xiaozhang Zheng, Harry Brielmann, Kevin J Hodgetts, Rajagopal Bakthavatchalam

Bioorg Med Chem Lett· August 2008


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From arylureas to biarylamides to aminoquinazolines: discovery of a novel, potent TRPV1 antagonist.
Xiaozhang Zheng, Kevin J Hodgetts, Harry Brielmann, Alan Hutchison, Frank Burkamp

Bioorg Med Chem Lett· October 2006


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