Publications by authors named "Kurt A Josef"

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Discovery of (1R,6S)-5-[4-(1-cyclobutyl-piperidin-4-yloxy)-phenyl]-3,4-diaza-bicyclo[4.1.0]hept-4-en-2-one (R,S-4a): histamine H(3) receptor inverse agonist demonstrating potent cognitive enhancing and wake promoting activity.
Robert L Hudkins, Kurt A Josef, Nadine C Becknell, Lisa D Aimone, Jacquelyn A Lyons

Bioorg Med Chem Lett· March 2014

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Synthesis of constrained benzocinnolinone analogues of CEP-26401 (irdabisant) as potent, selective histamine H3 receptor inverse agonists.
Kurt A Josef, Lisa D Aimone, Jacquelyn Lyons, Rita Raddatz, Robert L Hudkins

Bioorg Med Chem Lett· June 2012

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4-phenoxypiperidine pyridazin-3-one histamine H(3) receptor inverse agonists demonstrating potent and robust wake promoting activity.
Robert L Hudkins, Allison L Zulli, Reddeppa reddy Dandu, Ming Tao, Kurt A Josef

Bioorg Med Chem Lett· February 2012

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4,5-dihydropyridazin-3-one derivatives as histamine H₃ receptor inverse agonists.
Robert L Hudkins, Lisa D Aimone, Reddeppa Reddy Dandu, Derek Dunn, John A Gruner, Kurt A Josef

Bioorg Med Chem Lett· January 2012

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Identification of pyridazin-3-one derivatives as potent, selective histamine H₃ receptor inverse agonists with robust wake activity.
Robert L Hudkins, Lisa D Aimone, Thomas R Bailey, Robert J Bendesky, Reddeppa Reddy Dandu, Kurt A Josef

Bioorg Med Chem Lett· September 2011

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Mixed-lineage kinase 1 and mixed-lineage kinase 3 subtype-selective dihydronaphthyl[3,4-a]pyrrolo[3,4-c]carbazole-5-ones: optimization, mixed-lineage kinase 1 crystallography, and oral in vivo activity in 1-methyl-4-phenyltetrahydropyridine models.
Robert L Hudkins, James L Diebold, Ming Tao, Kurt A Josef, Chung Ho Park

J Med Chem· September 2008

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