Publications by authors named "Mark D Rosen"

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Beyond Traditional Structure-Based Drug Design: The Role of Iron Complexation, Strain, and Water in the Binding of Inhibitors for Hypoxia-Inducible Factor Prolyl Hydroxylase 2.
Scott D Bembenek, Hariharan Venkatesan, Hillary M Peltier, Mark D Rosen, Terrance D Barrett

ACS Omega· April 2019

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Glutamatergic stimulation induces GluN2B translation by the nitric oxide-Heme-Regulated eIF2α kinase in cortical neurons.
Eva Ramos-Fernández, Marta Tajes, Gerard Ill-Raga, Lina Vargas, Arnau Busquets-García, Mark D Rosen

Oncotarget· September 2016

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Prolyl hydroxylase inhibition corrects functional iron deficiency and inflammation-induced anaemia in rats.
Terrance D Barrett, Heather L Palomino, Theresa I Brondstetter, Kimon C Kanelakis, Xiaodong Wu, Mark D Rosen

Br J Pharmacol· August 2015

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Physiological Control of Nitric Oxide in Neuronal BACE1 Translation by Heme-Regulated eIF2α Kinase HRI Induces Synaptogenesis.
Gerard Ill-Raga, Marta Tajes, Arnau Busquets-García, Eva Ramos-Fernández, Lina M Vargas, Mark D Rosen

Antioxid Redox Signal· May 2015

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Consolidation of object recognition memory requires HRI kinase-dependent phosphorylation of eIF2α in the hippocampus.
Gerard ILL-Raga, Cristiano Köhler, Andressa Radiske, Ramón H Lima, Mark D Rosen

Hippocampus· June 2013

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Pharmacological characterization of 1-(5-chloro-6-(trifluoromethoxy)-1H-benzoimidazol-2-yl)-1H-pyrazole-4-carboxylic acid (JNJ-42041935), a potent and selective hypoxia-inducible factor prolyl hydroxylase inhibitor.
Terrance D Barrett, Heather L Palomino, Theresa I Brondstetter, Kimon C Kanelakis, Xiaodong Wu, Mark D Rosen

Mol Pharmacol· June 2011

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Benzimidazole-2-pyrazole HIF Prolyl 4-Hydroxylase Inhibitors as Oral Erythropoietin Secretagogues.
Mark D Rosen, Hariharan Venkatesan, Hillary M Peltier, Scott D Bembenek, Kimon C Kanelakis

ACS Med Chem Lett· December 2010

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Terminating Catalytic Asymmetric Heck Cyclizations by Stereoselective Intramolecular Capture of η-Allylpalladium Intermediates: Total Synthesis of (-)-Spirotryprostatin B and Three Stereoisomers.
Larry E Overman, Mark D Rosen

Tetrahedron· August 2010

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Discovery of the first known small-molecule inhibitors of heme-regulated eukaryotic initiation factor 2alpha (HRI) kinase.
Mark D Rosen, Craig R Woods, Steven D Goldberg, Michael D Hack, A Dawn Bounds

Bioorg Med Chem Lett· December 2009

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Characterization of a robust enzymatic assay for inhibitors of 2-oxoglutarate-dependent hydroxylases.
Kimon C Kanelakis, Heather L Palomino, Lina Li, Jiejun Wu, Wen Yan, Mark D Rosen

J Biomol Screen· July 2009

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Discovery of potent cholecystokinin-2 receptor antagonists: elucidation of key pharmacophore elements by X-ray crystallographic and NMR conformational analysis.
Mark D Rosen, Michael D Hack, Brett D Allison, Victor K Phuong, Craig R Woods

Bioorg Med Chem· April 2008

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Synthesis and solid-phase purification of anthranilic sulfonamides as CCK-2 ligands.
Craig R Woods, Michael D Hack, Brett D Allison, Victor K Phuong, Mark D Rosen

Bioorg Med Chem Lett· December 2007

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Total synthesis of (+/-)-didehydrostemofoline (asparagamine A) and (+/-)-isodidehydrostemofoline.
Markus Brüggemann, Andrew I McDonald, Larry E Overman, Mark D Rosen, Lothar Schwink

J Am Chem Soc· December 2003

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Total Synthesis of (-)-Spirotryprostatin B and Three Stereoisomers We thank NIH NIGMS (GM-30859) for financial support, Prof. A. J. Shaka and N. D. Taylor for DPFGSE experiments, Prof. H. Osada for providing spectral data for natural 1, and Prof. R. M. Williams and P. R. Sebahar for providing spectral data and a sample of synthetic ent-21. We are also grateful to Prof. R. M. Williams and Prof. S. J. Danishefsky for open exchange of information prior to publication. NMR and mass spectra were determined at UC Irvine with instruments purchased with the assistance of the NSF and NIH shared instrumentation programs.
Larry E. Overman, Mark D. Rosen

Angew Chem Int Ed Engl· December 2000

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