Publications by authors named "Michael D Bartberger"

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Divergent Catalysis: Catalytic Asymmetric [4+2] Cycloaddition of Palladium Enolates.
Kaylin N Flesch, Alexander Q Cusumano, Peng-Jui Chen, Christian Santiago Strong, Stephen R Sardini, Michael D Bartberger

J Am Chem Soc· May 2023

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Ir-Catalyzed Asymmetric Allylic Alkylation of Dialkyl Malonates Enabling the Construction of Enantioenriched All-Carbon Quaternary Centers.
Farbod A Moghadam, Elliot F Hicks, Zachary P Sercel, Alexander Q Cusumano, Michael D Bartberger

J Am Chem Soc· May 2022

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Iridium-catalyzed asymmetric -selective hydrogenation of 1,3-disubstituted isoquinolines.
Alexia N Kim, Aurapat Ngamnithiporn, Michael D Bartberger, Brian M Stoltz

Chem Sci· March 2022

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Systematic Study of the Glutathione Reactivity of -Phenylacrylamides: 2. Effects of Acrylamide Substitution.
Adam Birkholz, David J Kopecky, Laurie P Volak, Michael D Bartberger, Yuping Chen

J Med Chem· October 2020

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Enantioselective synthesis of highly oxygenated acyclic quaternary center-containing building blocks palladium-catalyzed decarboxylative allylic alkylation of cyclic siloxyketones.
Aurapat Ngamnithiporn, Toshihiko Iwayama, Michael D Bartberger, Brian M Stoltz

Chem Sci· September 2020

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The development of a structurally distinct series of BACE1 inhibitors via the (Z)-fluoro-olefin amide bioisosteric replacement.
Michael Frohn, Longbin Liu, Aaron C Siegmund, Wenyuan Qian, Albert Amegadzie, Michael D Bartberger

Bioorg Med Chem Lett· July 2020

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Enantioselective total synthesis of (-)-myrifabral A and B.
Tyler J Fulton, Anthony Y Chen, Michael D Bartberger, Brian M Stoltz

Chem Sci· April 2020

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Discovery of AM-6494: A Potent and Orally Efficacious β-Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitor with in Vivo Selectivity over BACE2.
Liping H Pettus, Matthew P Bourbeau, Jodi Bradley, Michael D Bartberger, Kui Chen

J Med Chem· March 2020

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Mechanistic Insights into the Racemization of Fused Cyclopropyl Isoxazolines.
Kyle W Quasdorf, Adam B Birkholz, Michael D Bartberger, John Colyer, Stephen Osgood

Org Lett· March 2020

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Iridium-Catalyzed Enantioselective and Diastereoselective Hydrogenation of 1,3-Disubstituted Isoquinolines.
Alexia N Kim, Aurapat Ngamnithiporn, Eric R Welin, Martin T Daiger, Christian U Grünanger, Michael D Bartberger

ACS Catal· March 2020

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Discovery of a Covalent Inhibitor of KRAS (AMG 510) for the Treatment of Solid Tumors.
Brian A Lanman, Jennifer R Allen, John G Allen, Albert K Amegadzie, Kate S Ashton, Michael D Bartberger

J Med Chem· January 2020

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Incorporation of a chiral gem-disubstituted nitrogen heterocycle yields an oxazolidinone antibiotic with reduced mitochondrial toxicity.
Alexander W Sun, Philip L Bulterys, Michael D Bartberger, Peter A Jorth, Brendan M O'Boyle

Bioorg Med Chem Lett· September 2019

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Discovery of -(1-Acryloylazetidin-3-yl)-2-(1-indol-1-yl)acetamides as Covalent Inhibitors of KRAS.
Youngsook Shin, Joon Won Jeong, Ryan P Wurz, Pragathi Achanta, Tara Arvedson, Michael D Bartberger

ACS Med Chem Lett· September 2019

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Discovery of TRPM8 Antagonist ( S)-6-(((3-Fluoro-4-(trifluoromethoxy)phenyl)(3-fluoropyridin-2-yl)methyl)carbamoyl)nicotinic Acid (AMG 333), a Clinical Candidate for the Treatment of Migraine.
Daniel B Horne, Kaustav Biswas, James Brown, Michael D Bartberger, Jeffrey Clarine

J Med Chem· September 2018

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Diastereoselective synthesis of fused cyclopropyl-3-amino-2,4-oxazine β-amyloid cleaving enzyme (BACE) inhibitors and their biological evaluation.
Jonathan D Low, Michael D Bartberger, Yuan Cheng, Doug Whittington, Quifen Xue

Bioorg Med Chem Lett· April 2018

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Enantioselective Pd-Catalyzed Decarboxylative Allylic Alkylation of Thiopyranones. Access to Acyclic, Stereogenic α-Quaternary Ketones.
Eric J Alexy, Scott C Virgil, Michael D Bartberger, Brian M Stoltz

Org Lett· October 2017

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Development of 2-aminooxazoline 3-azaxanthene β-amyloid cleaving enzyme (BACE) inhibitors with improved selectivity against Cathepsin D.
Jonathan D Low, Michael D Bartberger, Kui Chen, Yuan Cheng, Mark R Fielden

Medchemcomm· June 2017

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Correction to Fragment-Linking Approach Using F NMR Spectroscopy To Obtain Highly Potent and Selective Inhibitors of β-Secretase.
John B Jordan, Douglas A Whittington, Michael D Bartberger, E Allen Sickmier, Kui Chen

J Med Chem· April 2017

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The chemical biology of HNO signaling.
Christopher L Bianco, John P Toscano, Michael D Bartberger, Jon M Fukuto

Arch Biochem Biophys· March 2017

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Telescoped Process to Manufacture 6,6,6-Trifluorofucose via Diastereoselective Transfer Hydrogenation: Scalable Access to an Inhibitor of Fucosylation Utilized in Monoclonal Antibody Production.
Michal M Achmatowicz, John G Allen, Matthew M Bio, Michael D Bartberger, Christopher J Borths

J Org Chem· June 2016

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Application of 1,1-ADEQUATE, HMBC, and Density Functional Theory To Determine Regioselectivity in the Halogenation of Pyridine N-Oxides.
Tsang-Lin Hwang, Michael D Bartberger, Ying Chen

Org Lett· May 2016

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Fragment-Linking Approach Using (19)F NMR Spectroscopy To Obtain Highly Potent and Selective Inhibitors of β-Secretase.
John B Jordan, Douglas A Whittington, Michael D Bartberger, E Allen Sickmier, Kui Chen

J Med Chem· April 2016

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Stacking with No Planarity?
Hakan Gunaydin, Michael D Bartberger

ACS Med Chem Lett· April 2016

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Discovery of the imidazole-derived GPR40 agonist AM-3189.
Zhihua Ma, Daniel C-H Lin, Rajiv Sharma, Jinqian Liu, Liusheng Zhu, Michael D Bartberger

Bioorg Med Chem Lett· January 2016

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Systematic Study of the Glutathione (GSH) Reactivity of N-Arylacrylamides: 1. Effects of Aryl Substitution.
Victor J Cee, Laurie P Volak, Yuping Chen, Michael D Bartberger, Chris Tegley

J Med Chem· December 2015

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