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Publications by authors named "Moriyasu Masui"

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Discovery of NR2B-selective antagonists via scaffold hopping and pharmacokinetic profile optimization.
Kosuke Anan, Moriyasu Masui, Aya Tazawa, Minoru Tomida, Yoshihiro Haga

Bioorg Med Chem Lett· May 2019


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Rational Design of Novel 1,3-Oxazine Based β-Secretase (BACE1) Inhibitors: Incorporation of a Double Bond To Reduce P-gp Efflux Leading to Robust Aβ Reduction in the Brain.
Kouki Fuchino, Yasunori Mitsuoka, Moriyasu Masui, Noriyuki Kurose, Shuhei Yoshida

J Med Chem· June 2018


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Discovery of orally bioavailable cyclohexanol-based NR2B-selective NMDA receptor antagonists with analgesic activity utilizing a scaffold hopping approach.
Kosuke Anan, Moriyasu Masui, Shinichiro Hara, Miho Ohara, Masaharu Kume

Bioorg Med Chem Lett· September 2017


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