Publications by authors named "Naoki Tarui"

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[The quick screening of binding compounds and proteins for drug discovery and pharmacological research].
Naoki Tarui

Nihon Yakurigaku Zasshi· November 2024

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Discovery, synthesis, and structure-activity relations of 3,4-dihydro-1H-spiro(naphthalene-2,2'-piperidin)-1-ones as potassium-competitive acid blockers.
Toshihiro Imaeda, Koji Ono, Kazuo Nakai, Yasunobu Hori, Jun Matsukawa, Naoki Tarui

Bioorg Med Chem· July 2017

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Structure-based design of a new series of N-(piperidin-3-yl)pyrimidine-5-carboxamides as renin inhibitors.
Yasuhiro Imaeda, Michiko Tawada, Shinkichi Suzuki, Masaki Tomimoto, Mitsuyo Kondo, Naoki Tarui

Bioorg Med Chem· November 2016

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Novel approach of fragment-based lead discovery applied to renin inhibitors.
Michiko Tawada, Shinkichi Suzuki, Yasuhiro Imaeda, Hideyuki Oki, Gyorgy Snell, Naoki Tarui

Bioorg Med Chem· November 2016

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Synthetic studies of five-membered heteroaromatic derivatives as potassium-competitive acid blockers (P-CABs).
Yasuyoshi Arikawa, Atsushi Hasuoka, Haruyuki Nishida, Keizo Hirase, Nobuhiro Inatomi, Naoki Tarui

Bioorg Med Chem Lett· February 2016

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Molecular modeling, design, synthesis, and biological activity of 1H-pyrrolo[2,3-c]pyridine-7-amine derivatives as potassium-competitive acid blockers.
Yasuyoshi Arikawa, Atsushi Hasuoka, Keizo Hirase, Nobuhiro Inatomi, Fumihiko Sato, Naoki Tarui

Chem Pharm Bull (Tokyo)· May 2015

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Generating thermostabilized agonist-bound GPR40/FFAR1 using virus-like particles and a label-free binding assay.
Yoshihiko Hirozane, Takashi Motoyaji, Takamitsu Maru, Kengo Okada, Naoki Tarui

Mol Membr Biol· August 2014

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Physicochemically and pharmacokinetically stable nonapeptide KISS1 receptor agonists with highly potent testosterone-suppressive activity.
Taiji Asami, Naoki Nishizawa, Hisanori Matsui, Yoshihiro Takatsu, Atsuko Suzuki, Naoki Tarui

J Med Chem· July 2014

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Design, synthesis, and biological evaluation of novel investigational nonapeptide KISS1R agonists with testosterone-suppressive activity.
Taiji Asami, Naoki Nishizawa, Hisanori Matsui, Kimiko Nishibori, Yoshihiro Ishibashi, Naoki Tarui

J Med Chem· November 2013

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Serum stability of selected decapeptide agonists of KISS1R using pseudopeptides.
Taiji Asami, Naoki Nishizawa, Yoshihiro Ishibashi, Kimiko Nishibori, Masaharu Nakayama, Naoki Tarui

Bioorg Med Chem Lett· October 2012

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Discovery, synthesis, and biological evaluation of novel pyrrole derivatives as highly selective potassium-competitive acid blockers.
Haruyuki Nishida, Atsushi Hasuoka, Yasuyoshi Arikawa, Osamu Kurasawa, Keizo Hirase, Naoki Tarui

Bioorg Med Chem· June 2012

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Discovery of a novel pyrrole derivative 1-[5-(2-fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine fumarate (TAK-438) as a potassium-competitive acid blocker (P-CAB).
Yasuyoshi Arikawa, Haruyuki Nishida, Osamu Kurasawa, Atsushi Hasuoka, Keizo Hirase, Naoki Tarui

J Med Chem· May 2012

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High-throughput screening of potassium-competitive acid blockers.
Mitsuyo Kondo, Makiko Kawamoto, Atsushi Hasuoka, Masahiro Kajino, Nobuhiro Inatomi, Naoki Tarui

J Biomol Screen· February 2012

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Novel 3-phenylpiperidine-4-carboxamides as highly potent and orally long-acting neurokinin-1 receptor antagonists with reduced CYP3A induction.
Junya Shirai, Hideyuki Sugiyama, Shinji Morimoto, Hironobu Maezaki, Yasuharu Yamamoto, Naoki Tarui

Bioorg Med Chem· January 2012

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Design, structure-activity relationship, and highly efficient asymmetric synthesis of 3-phenyl-4-benzylaminopiperidine derivatives as novel neurokinin-1 receptor antagonists.
Junya Shirai, Takeshi Yoshikawa, Masayuki Yamashita, Yasuharu Yamamoto, Makiko Kawamoto, Naoki Tarui

Bioorg Med Chem· November 2011

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3-benzhydryl-4-piperidones as novel neurokinin-1 receptor antagonists and their efficient synthesis.
Junya Shirai, Masayoshi Yamaoka, Eikoh Imamiya, Minoru Nakamura, Naoki Tarui

Bioorg Med Chem· September 2011

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A noncompetitive BACE1 inhibitor TAK-070 ameliorates Abeta pathology and behavioral deficits in a mouse model of Alzheimer's disease.
Hiroaki Fukumoto, Hideki Takahashi, Naoki Tarui, Junji Matsui, Taisuke Tomita

J Neurosci· August 2010

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Kinetic resolution of an indan derivative using Bacillus sp. SUI-12: synthesis of a key intermediate of the melatonin receptor agonist TAK-375.
Naoki Tarui, Yoichi Nagano, Takeshi Sakane, Kiyoharu Matsumoto, Mitsuru Kawada

J Biosci Bioeng· November 2005

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Kinetic resolutions of indan derivatives using bacteria.
Naoki Tarui, Hayao Watanabe, Kohji Fukatsu, Shigenori Ohkawa, Kazuo Nakahama

Biosci Biotechnol Biochem· February 2002

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Microbial enantioselective ester hydrolysis for the preparation of optically active 4,1-benzoxazepine-3-acetic acid derivatives as squalene synthase inhibitors.
Naoki Tarui, Kazuo Nakahama, Yoichi Nagano, Motowo Izawa, Kiyoharu Matsumoto

Chem Pharm Bull (Tokyo)· January 2002

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