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Publications by authors named "Naphtali Reyna"

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Allosteric targeting of RIPK1: discovery of novel inhibitors parallel virtual screening and structure-guided optimization.
R S K Vijayan, Matthew M Hamilton, Dana E Pfaffinger, Fernando G Alvarez, Naphtali J Reyna

RSC Med Chem· September 2025


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Discovery of IACS-9779 and IACS-70465 as Potent Inhibitors Targeting Indoleamine 2,3-Dioxygenase 1 (IDO1) Apoenzyme.
Matthew M Hamilton, Faika Mseeh, Timothy J McAfoos, Paul G Leonard, Naphtali J Reyna

J Med Chem· August 2021


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Identification of potent and selective MTH1 inhibitors.
Alessia Petrocchi, Elisabetta Leo, Naphtali J Reyna, Matthew M Hamilton, Xi Shi

Bioorg Med Chem Lett· March 2016


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Structure-Guided Design of IACS-9571, a Selective High-Affinity Dual TRIM24-BRPF1 Bromodomain Inhibitor.
Wylie S Palmer, Guillaume Poncet-Montange, Gang Liu, Alessia Petrocchi, Naphtali Reyna

J Med Chem· February 2016


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