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Publications by authors named "Peter M Syka"

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Discovery of orally available tetrahydroquinoline-based glucocorticoid receptor agonists.
Andrew R Hudson, Robert I Higuchi, Steven L Roach, Mark E Adams, Angela Vassar, Peter M Syka

Bioorg Med Chem Lett· March 2011


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Nonsteroidal 2,3-dihydroquinoline glucocorticoid receptor agonists with reduced PEPCK activation.
Andrew R Hudson, Robert I Higuchi, Steven L Roach, Lino J Valdez, Mark E Adams, Peter M Syka

Bioorg Med Chem Lett· March 2011


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Tetrahydroquinolin-3-yl carbamate glucocorticoid receptor agonists with reduced PEPCK activation.
Steven L Roach, Robert I Higuchi, Andrew R Hudson, Angie Vassar, Virginia H S Grant, Peter M Syka

Bioorg Med Chem Lett· March 2011


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Tetrahydroquinoline glucocorticoid receptor agonists: discovery of a 3-hydroxyl for improving receptor selectivity.
Steven L Roach, Robert I Higuchi, Andrew R Hudson, Mark E Adams, Peter M Syka

Bioorg Med Chem Lett· January 2011


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