Publications by authors named "Peter P Roller"

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A dual-readout F2 assay that combines fluorescence resonance energy transfer and fluorescence polarization for monitoring bimolecular interactions.
Yuhong Du, Zaneta Nikolovska-Coleska, Min Qui, Lian Li, Iestyn Lewis, Peter P Roller

Assay Drug Dev Technol· August 2011

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Discovery of thioether-bridged cyclic pentapeptides binding to Grb2-SH2 domain with high affinity.
Sheng Jiang, Chenzhong Liao, Lakshman Bindu, Biaolin Yin, Karen W Worthy, Peter P Roller

Bioorg Med Chem Lett· May 2009

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Interaction of a cyclic, bivalent smac mimetic with the x-linked inhibitor of apoptosis protein.
Zaneta Nikolovska-Coleska, Jennifer L Meagher, Sheng Jiang, Chao-Yie Yang, Su Qiu, Peter P Roller

Biochemistry· September 2008

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Design and characterization of bivalent Smac-based peptides as antagonists of XIAP and development and validation of a fluorescence polarization assay for XIAP containing both BIR2 and BIR3 domains.
Zaneta Nikolovska-Coleska, Jennifer L Meagher, Sheng Jiang, Steven A Kawamoto, Wei Gao, Peter P Roller

Anal Biochem· March 2008

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Design, synthesis, and characterization of a potent, nonpeptide, cell-permeable, bivalent Smac mimetic that concurrently targets both the BIR2 and BIR3 domains in XIAP.
Haiying Sun, Zaneta Nikolovska-Coleska, Jianfeng Lu, Jennifer L Meagher, Chao-Yie Yang, Peter P Roller

J Am Chem Soc· December 2007

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Design and synthesis of paclitaxel conjugated with an ErbB2-recognizing peptide, EC-1.
Peng Li, Sheng Jiang, Stephanie C Pero, Lyn Oligino, David N Krag, Peter P Roller

Biopolymers· November 2007

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Design and synthesis of novel and potent inhibitors of the type II transmembrane serine protease, matriptase, based upon the sunflower trypsin inhibitor-1.
Peng Li, Sheng Jiang, Sheau-Ling Lee, Cheng Yong Lin, Michael D Johnson, Peter P Roller

J Med Chem· November 2007

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Structure-based design of flavonoid compounds as a new class of small-molecule inhibitors of the anti-apoptotic Bcl-2 proteins.
Guozhi Tang, Ke Ding, Zaneta Nikolovska-Coleska, Chao-Yie Yang, Su Qiu, Peter P Roller

J Med Chem· July 2007

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Pyrogallol-based molecules as potent inhibitors of the antiapoptotic Bcl-2 proteins.
Guozhi Tang, Chao-Yie Yang, Zaneta Nikolovska-Coleska, Jie Guo, Su Qiu, Peter P Roller

J Med Chem· April 2007

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Design and synthesis of redox stable analogues of sunflower trypsin inhibitors (SFTI-1) on solid support, potent inhibitors of matriptase.
Sheng Jiang, Peng Li, Sheau-Ling Lee, Cheng Yong Lin, Ya-Qiu Long, Peter P Roller

Org Lett· January 2007

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Structure-based design of potent Grb2-SH2 domain antagonists not relying on phosphotyrosine mimics.
Sheng Jiang, Peng Li, Megan L Peach, Lakshman Bindu, Karen W Worthy, Peter P Roller

Biochem Biophys Res Commun· October 2006

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Structure-based design of potent small-molecule inhibitors of anti-apoptotic Bcl-2 proteins.
Guoping Wang, Zaneta Nikolovska-Coleska, Chao-Yie Yang, Renxiao Wang, Guozhi Tang, Peter P Roller

J Med Chem· October 2006

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Design and concise synthesis of fully protected analogues of l-gamma-carboxyglutamic acid.
Sheng Jiang, Peng Li, Christopher C Lai, James A Kelley, Peter P Roller

J Org Chem· September 2006

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New HIV-1 reverse transcriptase inhibitors based on a tricyclic benzothiophene scaffold: synthesis, resolution, and inhibitory activity.
Krzysztof Krajewski, Yijun Zhang, Damon Parrish, Jeffrey Deschamps, Peter P Roller

Bioorg Med Chem Lett· June 2006

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Structure-based design of spiro-oxindoles as potent, specific small-molecule inhibitors of the MDM2-p53 interaction.
Ke Ding, Yipin Lu, Zaneta Nikolovska-Coleska, Guoping Wang, Su Qiu, Peter P Roller

J Med Chem· June 2006

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Discovery of a novel nonphosphorylated pentapeptide motif displaying high affinity for Grb2-SH2 domain by the utilization of 3'-substituted tyrosine derivatives.
Yan-Li Song, Megan L Peach, Peter P Roller, Su Qiu, Shaomeng Wang

J Med Chem· March 2006

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Small nonphosphorylated Grb2-SH2 domain antagonists evaluated by surface plasmon resonance technology.
Feng-Di T Lung, Chiung-Wen Chang, Meng-Chin Chong, Chien-Chung Liou, Peng Li, Peter P Roller

Biopolymers· December 2005

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Structure-based design of potent non-peptide MDM2 inhibitors.
Ke Ding, Yipin Lu, Zaneta Nikolovska-Coleska, Su Qiu, Yousong Ding, Peter P Roller

J Am Chem Soc· July 2005

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Binding affinity difference induced by the stereochemistry of the sulfoxide bridge of the cyclic peptide inhibitors of Grb2-SH2 domain: NMR studies for the structural origin.
Yan-hong Shi, Yan-Li Song, Dong-hai Lin, Jinzhi Tan, Peter P Roller

Biochem Biophys Res Commun· May 2005

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Structure-based design, synthesis and biochemical testing of novel and potent Smac peptido-mimetics.
Haiying Sun, Zaneta Nikolovska-Coleska, Jianyong Chen, Chao-Yie Yang, York Tomita, Peter P Roller

Bioorg Med Chem Lett· February 2005

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Structure-based design of potent, conformationally constrained Smac mimetics.
Haiying Sun, Zaneta Nikolovska-Coleska, Chao-Yie Yang, Liang Xu, Meilan Liu, Peter P Roller

J Am Chem Soc· December 2004

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Synthesis and HIV-1 integrase inhibitory activity of dimeric and tetrameric analogs of indolicidin.
Krzysztof Krajewski, Christophe Marchand, Ya-Qiu Long, Yves Pommier, Peter P Roller

Bioorg Med Chem Lett· November 2004

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Structure-based discovery of nonpeptidic small organic compounds to block the T cell response to myelin basic protein.
Niklas K U Koehler, Chao-Yie Yang, Judith Varady, Yipin Lu, Xiong-Wu Wu, Peter P Roller

J Med Chem· October 2004

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Development and optimization of a binding assay for the XIAP BIR3 domain using fluorescence polarization.
Zaneta Nikolovska-Coleska, Renxiao Wang, Xueliang Fang, Hongguang Pan, York Tomita, Peter P Roller

Anal Biochem· September 2004

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Structure-based design, synthesis, and evaluation of conformationally constrained mimetics of the second mitochondria-derived activator of caspase that target the X-linked inhibitor of apoptosis protein/caspase-9 interaction site.
Haiying Sun, Zaneta Nikolovska-Coleska, Chao-Yie Yang, Liang Xu, York Tomita, Peter P Roller

J Med Chem· August 2004

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