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Publications by authors named "Philippe Risch"

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Cellular Potency Optimization of Novel Heme-Binding Imidazo[5,1-]thiazoles, Imidazo[1,5-]pyridines and Pyrazines as Potent IDO1 Inhibitors Devoid of Cytochrome P450 Inhibition.
Sylvaine Cren, Carina Lotz-Jenne, Thierry Kimmerlin, Julien Pothier, Philippe Risch

J Med Chem· October 2025


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Verification of the Major Metabolic Oxidation Path for the Naphthoyl Group in Chemoattractant Receptor-Homologous Molecule Expressed on Th2 Cells (CRTh2) Antagonist 2-(2-(1-Naphthoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5(2H)-yl)acetic Acid (Setipiprant/ACT-129968).
Philippe Risch, Thomas Pfeifer, Jerome Segrestaa, Heinz Fretz, Julien Pothier

J Med Chem· October 2015


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Design of novel aminopyrrolidine factor Xa inhibitors from a screening hit.
Katrin Groebke Zbinden, Lilli Anselm, David W Banner, Jörg Benz, Francesca Blasco, Philippe Risch

Eur J Med Chem· July 2009


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