Publications by authors named "Raphael Rahmani"

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Heterocyclic core modifications in trypanosomacidal 2-[(phenylheteroaryl)ethyl]ureas.
Arthur Toynton, Lori Ferrins, Harriet L Newson, Melissa L Sykes, Swapna Varghese, Raphaël Rahmani

RSC Med Chem· January 2025

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Novel aroyl guanidine anti-trypanosomal compounds that exert opposing effects on parasite energy metabolism.
Swapna Varghese, Anubhav Srivastava, Siu Wai Wong, Thuy Le, Noel Pitcher, Raphael Rahmani

Eur J Med Chem· March 2024

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Structure-Activity Studies of Truncated Latrunculin Analogues with Antimalarial Activity.
Swapna Varghese, Raphaël Rahmani, Damien R Drew, James G Beeson, Jake Baum

ChemMedChem· February 2021

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Hit-to-lead optimization of novel benzimidazole phenylacetamides as broad spectrum trypanosomacides.
Nicole McNamara, Raphael Rahmani, Melissa L Sykes, Vicky M Avery, Jonathan Baell

RSC Med Chem· June 2020

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Discovery of Potent -Ethylurea Pyrazole Derivatives as Dual Inhibitors of and .
Swapna Varghese, Raphaël Rahmani, Stephanie Russell, Girdhar Singh Deora, Lori Ferrins

ACS Med Chem Lett· March 2020

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Crystal structure of the M muscarinic acetylcholine receptor.
Ziva Vuckovic, Patrick R Gentry, Alice E Berizzi, Kunio Hirata, Swapna Varghese, Raphaël Rahmani

Proc Natl Acad Sci U S A· December 2019

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8-Mercaptoguanine Derivatives as Inhibitors of Dihydropteroate Synthase.
Matthew L Dennis, Michael D Lee, Jitendra R Harjani, Mohamed Ahmed, Aaron J DeBono, Raphaël Rahmani

Chemistry· February 2018

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Truncated Latrunculins as Actin Inhibitors Targeting Plasmodium falciparum Motility and Host Cell Invasion.
Swapna Johnson, Raphaël Rahmani, Damien R Drew, Melanie J Williams, Mark Wilkinson

J Med Chem· December 2016

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Hit-to-Lead Optimization of a Novel Class of Potent, Broad-Spectrum Trypanosomacides.
Stephanie Russell, Raphaël Rahmani, Amy J Jones, Harriet L Newson, Kevin Neilde, Marzieh Rahmani Khajouei

J Med Chem· November 2016

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Structural Basis for the Selective Binding of Inhibitors to 6-Hydroxymethyl-7,8-dihydropterin Pyrophosphokinase from Staphylococcus aureus and Escherichia coli.
Matthew L Dennis, Noel P Pitcher, Michael D Lee, Aaron J DeBono, Zhong-Chang Wang, Raphaël Rahmani

J Med Chem· June 2016

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6-Arylpyrazine-2-carboxamides: A New Core for Trypanosoma brucei Inhibitors.
Raphaël Rahmani, Kung Ban, Amy J Jones, Lori Ferrins, Danny Ganame

J Med Chem· September 2015

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Structure-based design and development of functionalized Mercaptoguanine derivatives as inhibitors of the folate biosynthesis pathway enzyme 6-hydroxymethyl-7,8-dihydropterin pyrophosphokinase from Staphylococcus aureus.
Matthew L Dennis, Sandeep Chhabra, Zhong-Chang Wang, Aaron Debono, Olan Dolezal, Raphael Rahmani

J Med Chem· November 2014

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Pyridyl benzamides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei.
Lori Ferrins, Michelle Gazdik, Raphaël Rahmani, Swapna Varghese, Melissa L Sykes

J Med Chem· August 2014

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trans-1,2-Disiloxybenzocyclobutene, an adequate partner for the auto-oxidation: EPR/spin trapping and theoretical studies.
Jean Drujon, Raphaël Rahmani, Virginie Héran, Romain Blanc, Yannick Carissan

Phys Chem Chem Phys· April 2014

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Structural basis for modulation of a G-protein-coupled receptor by allosteric drugs.
Ron O Dror, Hillary F Green, Celine Valant, David W Borhani, James R Valcourt, Raphaël Rahmani

Nature· November 2013

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Drug discovery and human African trypanosomiasis: a disease less neglected?
Lori Ferrins, Raphaël Rahmani, Jonathan B Baell

Future Med Chem· October 2013

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3-(Oxazolo[4,5-b]pyridin-2-yl)anilides as a novel class of potent inhibitors for the kinetoplastid Trypanosoma brucei, the causative agent for human African trypanosomiasis.
Lori Ferrins, Raphaël Rahmani, Melissa L Sykes, Amy J Jones, Vicky M Avery

Eur J Med Chem· August 2013

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Direct-type aldol reactions of fluorenylidene-protected/activated glycine esters with aldehydes for the synthesis of β-hydroxy-α-amino acid derivatives.
Raphaël Rahmani, Masatoshi Matsumoto, Yasuhiro Yamashita, Shū Kobayashi

Chem Asian J· June 2012

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Dramatic influence of the substitution of alkylidene-5H-furan-2-ones in Diels-Alder cycloadditions with o-quinonedimethide as diene partner: en route to the CDEF polycyclic ring system of lactonamycin.
Sébastien Dubois, Fabien Rodier, Romain Blanc, Raphaël Rahmani, Virginie Héran

Org Biomol Chem· June 2012

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Diels-Alder cycloaddition of o-quinonedimethides and alkylidene-5H-furan-2-ones: new and rapid access to lambertellol cores and arthrinone derivatives.
Romain Blanc, Virginie Héran, Raphaël Rahmani, Laurent Commeiras, Jean-Luc Parrain

Org Biomol Chem· December 2010

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