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Publications by authors named "Roger Wermuth"

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Novel Indane-Containing NBTIs with Potent Anti-Gram-Negative Activity and Minimal hERG Inhibition.
John G Cumming, Lukas Kreis, Holger Kühne, Roger Wermuth, Maarten Vercruysse

ACS Med Chem Lett· December 2023


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Discovery of a Series of Indane-Containing NBTIs with Activity against Multidrug-Resistant Gram-Negative Pathogens.
John G Cumming, Lukas Kreis, Holger Kühne, Roger Wermuth, Maarten Vercruysse

ACS Med Chem Lett· July 2023


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Discovery of benzoylisoindolines as a novel class of potent, selective and orally active GlyT1 inhibitors.
Emmanuel Pinard, Daniela Alberati, Markus Bender, Edilio Borroni, Virginie Brom, Roger Wermuth

Bioorg Med Chem Lett· December 2010


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Selective GlyT1 inhibitors: discovery of [4-(3-fluoro-5-trifluoromethylpyridin-2-yl)piperazin-1-yl][5-methanesulfonyl-2-((S)-2,2,2-trifluoro-1-methylethoxy)phenyl]methanone (RG1678), a promising novel medicine to treat schizophrenia.
Emmanuel Pinard, Alexander Alanine, Daniela Alberati, Markus Bender, Edilio Borroni, Roger Wermuth

J Med Chem· June 2010


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