Publications by authors named "Ryosuke Watari"

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Discovery of the Clinical Candidate : A Second-Generation of SARS-CoV-2 3CL Protease Inhibitor for Treating COVID-19.
Yuto Unoh, Keiichiro Hirai, Shota Uehara, Sho Kawashima, Haruaki Nobori, Ryosuke Watari

J Med Chem· October 2025

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Investigation of an OATP1B inhibitory effect by a cyclic peptide using the endogenous biomarker coproporphyrin-I in monkeys.
Hiromi Sawada, Yasuto Kido, Makoto Iwasaki, Kimiko Nishida, Kei Mayumi, Ryosuke Watari

Drug Metab Pharmacokinet· August 2025

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Novel Approach to Pre-Exposure Prophylaxis (PrEP) of COVID-19: Development of S-892216 Long-Acting Injectable Suspension.
Ryo Ohashi, Ryosuke Watari, Daisuke Kondo, Shuichi Otake, Tatsuhiko Murata

Chem Pharm Bull (Tokyo)· August 2025

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Minimal Involvement of P-gp and BCRP in Oral Absorption of Ensitrelvir, An Oral SARS-CoV-2 3C-like Protease Inhibitor, in a Non-Clinical Investigation.
Ryosuke Watari, Naomi Tamura, Shinpei Yoshida, Yasuto Kido, Takanobu Matsuzaki

J Pharm Sci· September 2024

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Prediction of drug-drug interaction risk of P-glycoprotein substrate in drug discovery.
Yasuto Kido, Isamu Nanchi, Takanobu Matsuzaki, Ryosuke Watari, Hayato Kiyohara

Drug Metab Pharmacokinet· June 2024

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Prophylactic effect of ensitrelvir in mice infected with SARS-CoV-2.
Haruaki Nobori, Keiko Baba, Takayuki Kuroda, Kaoru Baba, Kazumi Matsumoto, Ryosuke Watari

Antiviral Res· April 2024

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Utility of Coproporphyrin-I Determination in First-in-Human Study for Early Evaluation of OATP1B Inhibitory Potential Based on Investigation of Ensitrelvir, an Oral SARS-CoV-2 3C-Like Protease Inhibitor.
Ryosuke Watari, Hiromi Sawada, Hiroshi Hashimoto, Yasuyuki Kasai, Ryoko Oka

J Pharm Sci· March 2024

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Efficacy comparison of 3CL protease inhibitors ensitrelvir and nirmatrelvir against SARS-CoV-2 in vitro and in vivo.
Takayuki Kuroda, Haruaki Nobori, Keita Fukao, Kaoru Baba, Kazumi Matsumoto, Ryosuke Watari

J Antimicrob Chemother· April 2023

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Quantitative prediction of OATP1B-mediated drug-drug interactions using endogenous biomarker coproporphyrin I.
Hiroaki Takubo, Koji Bessho, Ryosuke Watari, Ryota Shigemi

Xenobiotica· April 2022

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Discovery of 2-Sulfinyl-Diazabicyclooctane Derivatives, Potential Oral β-Lactamase Inhibitors for Infections Caused by Serine β-Lactamase-Producing Enterobacterales.
Motohiro Fujiu, Katsuki Yokoo, Jun Sato, Satoru Shibuya, Kazuo Komano, Ryosuke Watari

J Med Chem· July 2021

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The antagonistic activity profile of naloxone in μ-opioid receptor agonist-induced psychological dependence.
Atsushi Nakamura, Kana Yasufuku, Shinji Shimada, Hiroyuki Aritomi, Youko Furue, Ryosuke Watari

Neurosci Lett· September 2020

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Minimal contribution of P-gp on the low brain distribution of naldemedine, a peripherally acting μ-opioid receptor antagonist.
Ryosuke Watari, Akihiro Matsuda, Shuichi Ohnishi, Hiroshi Hasegawa

Drug Metab Pharmacokinet· April 2019

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Highly Conformationally Restricted Cyclopropane Tethers with Three-Dimensional Structural Diversity Drastically Enhance the Cell Permeability of Cyclic Peptides.
Kouhei Matsui, Yasuto Kido, Ryosuke Watari, Yousuke Kashima, Yutaka Yoshida

Chemistry· March 2017

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Using improved serial blood sampling method of mice to study pharmacokinetics and drug-drug interaction.
Ayahisa Watanabe, Ryosuke Watari, Keiko Ogawa, Ryosuke Shimizu, Yukari Tanaka

J Pharm Sci· March 2015

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Using Improved Serial Blood Sampling Method of Mice to Study Pharmacokinetics and Drug-Drug Interaction.
Ayahisa Watanabe, Ryosuke Watari, Keiko Ogawa, Ryosuke Shimizu, Yukari Tanaka

J Pharm Sci· March 2015

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